CA2387745A1 - Positive modulators of nicotinic receptor agonists - Google Patents
Positive modulators of nicotinic receptor agonists Download PDFInfo
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- CA2387745A1 CA2387745A1 CA002387745A CA2387745A CA2387745A1 CA 2387745 A1 CA2387745 A1 CA 2387745A1 CA 002387745 A CA002387745 A CA 002387745A CA 2387745 A CA2387745 A CA 2387745A CA 2387745 A1 CA2387745 A1 CA 2387745A1
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9903997-6 | 1999-11-03 | ||
| SE9903997A SE9903997D0 (sv) | 1999-11-03 | 1999-11-03 | New compounds |
| PCT/SE2000/002148 WO2001032619A1 (en) | 1999-11-03 | 2000-11-01 | Positive modulators of nicotinic receptor agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2387745A1 true CA2387745A1 (en) | 2001-05-10 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002387745A Abandoned CA2387745A1 (en) | 1999-11-03 | 2000-11-01 | Positive modulators of nicotinic receptor agonists |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US6750242B1 (enExample) |
| EP (1) | EP1230216A1 (enExample) |
| JP (1) | JP2003513071A (enExample) |
| KR (1) | KR20020063176A (enExample) |
| CN (1) | CN1239482C (enExample) |
| AU (1) | AU783507B2 (enExample) |
| BR (1) | BR0015195A (enExample) |
| CA (1) | CA2387745A1 (enExample) |
| CO (1) | CO5251458A1 (enExample) |
| IL (1) | IL149098A0 (enExample) |
| MX (1) | MXPA02004232A (enExample) |
| NO (1) | NO323076B1 (enExample) |
| NZ (2) | NZ518450A (enExample) |
| SE (1) | SE9903997D0 (enExample) |
| WO (1) | WO2001032619A1 (enExample) |
| ZA (1) | ZA200203171B (enExample) |
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| SE9903998D0 (sv) * | 1999-11-03 | 1999-11-03 | Astra Ab | New compounds |
| DE10164139A1 (de) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-Heteroarylcarbonsäureamide |
| DE10234424A1 (de) * | 2002-07-29 | 2004-02-12 | Bayer Ag | Benzothiophen-, Benzofuran- und Indolharnstoffe |
| US7244745B2 (en) | 2002-08-30 | 2007-07-17 | Memory Pharmaceuticals Corp. | Heterocyclic compounds, methods for the preparation thereof, and uses thereof |
| CA2499128C (en) | 2002-09-25 | 2012-07-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof |
| WO2005092890A2 (en) | 2004-03-25 | 2005-10-06 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| ATE489138T1 (de) | 2005-04-13 | 2010-12-15 | Neuraxon Inc | Substituierte indolverbindungen mit nos-hemmender aktivität |
| US20070134169A1 (en) * | 2005-12-11 | 2007-06-14 | Rabinoff Michael D | Methods for smoking cessation or alcohol cessation or other addiction cessation |
| ZA200809659B (en) * | 2006-04-13 | 2010-03-31 | Neuraxon Inc | 1,5 and 3,6-substituted indole compounds having NOS inhibitory activity |
| WO2009062318A1 (en) * | 2007-11-16 | 2009-05-22 | Neuraxon, Inc. | 3,5-substituted indole compounds having nos and norepinephrine reuptake inhibitory activity |
| US20090163451A1 (en) * | 2007-11-16 | 2009-06-25 | Frank Porreca | Methods for treating visceral pain |
| EA201000808A1 (ru) * | 2007-11-16 | 2011-04-29 | Ньюраксон, Инк. | Индольные соединения и способы лечения висцеральной боли |
| US8383657B2 (en) | 2007-12-21 | 2013-02-26 | Abbott Laboratories | Thiazolylidine urea and amide derivatives and methods of use thereof |
| US8536221B2 (en) * | 2008-02-07 | 2013-09-17 | Abbvie Inc. | Amide derivatives as positive allosteric modulators and methods of use thereof |
| ES2392796T3 (es) * | 2008-04-17 | 2012-12-13 | Proximagen Limited | Moduladores de tipo indol del receptor nicotínico de acetilcolina alfa-7 |
| EA019518B1 (ru) * | 2009-04-16 | 2014-04-30 | Проксимаген Лимитед | ПРОИЗВОДНЫЕ ИНДОЛА В КАЧЕСТВЕ МОДУЛЯТОРОВ РЕЦЕПТОРА α7 nAChR |
| TWI519532B (zh) * | 2010-05-17 | 2016-02-01 | 艾維沃製藥公司 | （Ｒ）－７－氯－Ｎ－（啶－３－基）苯並［b］噻吩－２－羧醯胺鹽酸鹽單水合物之結晶形體 |
| TW201245185A (en) | 2011-04-01 | 2012-11-16 | Lundbeck & Co As H | New positive allosteric modulators of nicotinic acetylcholine receptor |
| AR086791A1 (es) | 2011-07-01 | 2014-01-22 | Lundbeck & Co As H | Moduladores alostericos positivos del receptor de acetilcolina nicotinico |
| RU2017136693A (ru) | 2012-05-08 | 2019-02-08 | Форум Фармасьютикалз, Инк. | Способы поддержания, лечения или улучшения когнитивной функции |
| KR102242658B1 (ko) * | 2018-08-29 | 2021-04-21 | 숙명여자대학교산학협력단 | 치환된 인돌 유도체, 이의 제조방법 및 이를 유효성분으로 포함하는 PPARα, PPARγ 및 PPARδ 관련 질환의 예방 또는 치료용 약학적 조성물 |
Family Cites Families (9)
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|---|---|---|---|---|
| US2787551A (en) * | 1954-02-24 | 1957-04-02 | Eastman Kodak Co | Compositions stabilized with hydroxyindole |
| BE758766A (fr) * | 1969-11-17 | 1971-05-10 | Ici Ltd | Nouveaux derives de la morpholine et de la |
| US4704390A (en) * | 1986-02-13 | 1987-11-03 | Warner-Lambert Company | Phenyl and heterocyclic tetrahydropyridyl alkoxy-benzheterocyclic compounds as antipsychotic agents |
| JPH06500551A (ja) * | 1990-09-13 | 1994-01-20 | ビーチャム・グループ・パブリック・リミテッド・カンパニー | ５ｈｔ受容体アンタゴニストとしてのインドールウレア |
| CA2124206C (en) * | 1991-11-25 | 2001-02-27 | John Eugene Macor | Indole derivatives |
| WO1993018026A1 (en) * | 1992-03-04 | 1993-09-16 | Beecham Group Plc | Indole ureas as 5-ht1c receptor antogonists |
| US5504101A (en) * | 1994-05-06 | 1996-04-02 | Allelix Biopharmaceuticals, Inc. | 5-HT-1D receptor ligands |
| FR2722686B1 (fr) * | 1994-07-22 | 1996-08-30 | Oreal | Set, procede, dispositif et composition de teinture des fibres keratiniques |
| US5576321A (en) * | 1995-01-17 | 1996-11-19 | Eli Lilly And Company | Compounds having effects on serotonin-related systems |
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- 2000-11-01 AU AU14264/01A patent/AU783507B2/en not_active Ceased
- 2000-11-01 CN CNB008154414A patent/CN1239482C/zh not_active Expired - Fee Related
- 2000-11-01 CO CO00083175A patent/CO5251458A1/es not_active Application Discontinuation
- 2000-11-01 MX MXPA02004232A patent/MXPA02004232A/es unknown
- 2000-11-01 NZ NZ518450A patent/NZ518450A/en unknown
- 2000-11-01 WO PCT/SE2000/002148 patent/WO2001032619A1/en not_active Ceased
- 2000-11-01 CA CA002387745A patent/CA2387745A1/en not_active Abandoned
- 2000-11-01 BR BR0015195-5A patent/BR0015195A/pt not_active IP Right Cessation
- 2000-11-01 KR KR1020027005706A patent/KR20020063176A/ko not_active Ceased
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- 2000-11-01 IL IL14909800A patent/IL149098A0/xx unknown
- 2000-11-01 NZ NZ530161A patent/NZ530161A/en unknown
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- 2002-04-26 NO NO20022009A patent/NO323076B1/no unknown
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| EP1230216A1 (en) | 2002-08-14 |
| NZ518450A (en) | 2004-04-30 |
| AU1426401A (en) | 2001-05-14 |
| NO20022009L (no) | 2002-07-02 |
| CO5251458A1 (es) | 2003-02-28 |
| NO323076B1 (no) | 2006-12-27 |
| AU783507B2 (en) | 2005-11-03 |
| US6750242B1 (en) | 2004-06-15 |
| MXPA02004232A (es) | 2002-10-17 |
| SE9903997D0 (sv) | 1999-11-03 |
| IL149098A0 (en) | 2002-11-10 |
| ZA200203171B (en) | 2003-09-23 |
| BR0015195A (pt) | 2002-06-18 |
| KR20020063176A (ko) | 2002-08-01 |
| CN1239482C (zh) | 2006-02-01 |
| NO20022009D0 (no) | 2002-04-26 |
| WO2001032619A1 (en) | 2001-05-10 |
| JP2003513071A (ja) | 2003-04-08 |
| CN1387512A (zh) | 2002-12-25 |
| NZ530161A (en) | 2005-08-26 |
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