CA2191999A1 - Hydrazides d'acide carboxylique de carbamyle et leur utilisation contre les champignons - Google Patents

Hydrazides d'acide carboxylique de carbamyle et leur utilisation contre les champignons

Info

Publication number
CA2191999A1
CA2191999A1 CA002191999A CA2191999A CA2191999A1 CA 2191999 A1 CA2191999 A1 CA 2191999A1 CA 002191999 A CA002191999 A CA 002191999A CA 2191999 A CA2191999 A CA 2191999A CA 2191999 A1 CA2191999 A1 CA 2191999A1
Authority
CA
Canada
Prior art keywords
alkyl
aryl
alkoxy
cyano
carry
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002191999A
Other languages
English (en)
Inventor
Oliver Wagner
Frank Wetterich
Karl Eicken
Eberhard Ammermann
Gisela Lorenz
Thomas Muller
John-Bryan Speakman
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE4419516A external-priority patent/DE4419516A1/de
Priority claimed from DE1995104423 external-priority patent/DE19504423A1/de
Application filed by Individual filed Critical Individual
Publication of CA2191999A1 publication Critical patent/CA2191999A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/40—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/42—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/54—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/12—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, neither directly attached to a ring nor the nitrogen atom being a member of a heterocyclic ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22—O-Aryl or S-Aryl esters thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/24—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing the groups, or; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C243/24—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids
    • C07C243/26—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C243/34—Hydrazines having nitrogen atoms of hydrazine groups acylated by carboxylic acids with acylating carboxyl groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of a carbon skeleton further substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/60—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups having oxygen atoms of carbamate groups bound to nitrogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des hydrazides d'acide carboxylique de carbamyle de la formule (I) ainsi que leurs sels, dont les restes ont les notations suivantes: R?1¿ désigne alkyle, alcényle, alcinyle, cycloalkyle, cycloalcényle, aryle ou hétéroaryle éventuellement substitué ou un carbo- ou hétérocycle non aromatique éventuellement substitué, W?1¿W?2¿C=N-, où W?1¿ désigne alkyle, alcényle, alcinyle, cycloalkyle, cycloalcényle, aryle ou hétéroaryle éventuellement substitué et W?2¿ désigne hydrogène ou W?1¿; R?2¿ désigne hydrogène ou alkyle ou cycloalkyle éventuellement substitué; R?3¿ désigne alkyle, cycloalkyle ou phénylalkyle éventuellement substitué; R?4¿ désigne hydrogène ou un des restes R?3¿ ou R?3¿ et R?4¿ désignent conjointement avec l'atome de C auquel ils sont liés, un carbo- ou hétérocycle saturé éventuellement substitué; R?5¿ désigne un des restes R?2¿; R?6¿ désigne alkyle, alcényle, alcinyle, cycloalkyle, cycloalcényle, aryle ou hétéroaryle éventuellement substitué, un carbo- ou hétérocycle non aromatique éventuellement substitué ou hydrogène si R?3¿ désigne iso-propyle; R?7¿ désigne un des restes R?6¿, à l'exception d'hydrogène; X?1¿, X?2¿, X?3¿ désigne chacun oxygène ou soufre. L'invention concerne également leurs procédés de préparation, des agents qui les contiennent, leur utilisation et de plus des intermédiaires de la formule (IV) dans lesquels X?3¿ désigne oxygène et R?3¿ désigne un groupe CH(CH¿3?)¿2?, CH¿2?CH(CH¿3?)2 ou CH(CH¿3?)C¿2?H¿5?.
CA002191999A 1994-06-03 1995-05-20 Hydrazides d'acide carboxylique de carbamyle et leur utilisation contre les champignons Abandoned CA2191999A1 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE4419516A DE4419516A1 (de) 1994-06-03 1994-06-03 Carbamoylcarbonsäurehydrazide
DEP4419516.8 1994-06-03
DE1995104423 DE19504423A1 (de) 1995-02-10 1995-02-10 Carbamoylcarbonsäurehydrazide
DE19504423.1 1995-02-10

Publications (1)

Publication Number Publication Date
CA2191999A1 true CA2191999A1 (fr) 1995-12-14

Family

ID=25937165

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002191999A Abandoned CA2191999A1 (fr) 1994-06-03 1995-05-20 Hydrazides d'acide carboxylique de carbamyle et leur utilisation contre les champignons

Country Status (8)

Country Link
EP (1) EP0763014A1 (fr)
JP (1) JPH10501215A (fr)
KR (1) KR970703306A (fr)
AU (1) AU685957B2 (fr)
BR (1) BR9507914A (fr)
CA (1) CA2191999A1 (fr)
IL (1) IL113916A0 (fr)
WO (1) WO1995033710A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI297335B (en) 2001-07-10 2008-06-01 Synta Pharmaceuticals Corp Taxol enhancer compounds
TWI252847B (en) 2001-07-10 2006-04-11 Synta Pharmaceuticals Corp Synthesis of taxol enhancers
TWI332943B (en) 2001-07-10 2010-11-11 Synta Pharmaceuticals Corp Taxol enhancer compounds
TWI330079B (en) * 2003-01-15 2010-09-11 Synta Pharmaceuticals Corp Treatment for cancers
JP5362986B2 (ja) 2004-06-23 2013-12-11 シンタ ファーマスーティカルズ コーポレイション 癌治療のためのビス（チオ‐ヒドラジドアミド）塩
BRPI0610219A2 (pt) 2005-04-15 2010-06-08 Synta Pharmaceuticals Corp métodos de tratamento de um ser humano com cáncer e composição de farmacêutica
KR20090045354A (ko) 2006-08-21 2009-05-07 신타 파마슈티칼스 코프. 증식성 장애를 치료하기 위한 화합물
AU2007290490B2 (en) 2006-08-31 2011-09-08 Synta Pharmaceuticals Corp. Combination with bis(thiohydrazide amides) for treating cancer
TW200829543A (en) 2006-09-15 2008-07-16 Synta Pharmaceuticals Corp Purification of bis(thiohydrazide amides)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1199540B (de) * 1963-12-27 1965-08-26 Schering Ag Mittel mit Wirkung gegen echten Mehltau

Also Published As

Publication number Publication date
IL113916A0 (en) 1995-08-31
AU2735395A (en) 1996-01-04
BR9507914A (pt) 1997-09-23
KR970703306A (ko) 1997-07-03
AU685957B2 (en) 1998-01-29
EP0763014A1 (fr) 1997-03-19
WO1995033710A1 (fr) 1995-12-14
JPH10501215A (ja) 1998-02-03

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Legal Events

Date Code Title Description
FZDE Discontinued