CA2117075A1 - Quinazoline derivatives and their preparation - Google Patents

Quinazoline derivatives and their preparation

Info

Publication number
CA2117075A1
CA2117075A1 CA002117075A CA2117075A CA2117075A1 CA 2117075 A1 CA2117075 A1 CA 2117075A1 CA 002117075 A CA002117075 A CA 002117075A CA 2117075 A CA2117075 A CA 2117075A CA 2117075 A1 CA2117075 A1 CA 2117075A1
Authority
CA
Canada
Prior art keywords
compound
salts
alkyl
formula
hydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002117075A
Other languages
English (en)
French (fr)
Inventor
Norihiko Shimazaki
Yoshikuni Itoh
Takumi Yatabe
Hitoshi Yamazaki
Masashi Hashimoto
Hirokazu Tanaka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/755,747 external-priority patent/US5296487A/en
Application filed by Individual filed Critical Individual
Publication of CA2117075A1 publication Critical patent/CA2117075A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA002117075A 1991-09-06 1992-09-02 Quinazoline derivatives and their preparation Abandoned CA2117075A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP07/755,747 1991-09-06
US07/755,747 US5296487A (en) 1990-01-02 1991-09-06 Quinazoline derivatives and their preparation
PCT/JP1992/001117 WO1993005035A1 (en) 1991-09-06 1992-09-02 Quinazoline derivatives and their preparation
CN93102096A CN1092067A (zh) 1991-09-06 1993-03-05 喹唑啉衍生物及其制备

Publications (1)

Publication Number Publication Date
CA2117075A1 true CA2117075A1 (en) 1993-03-18

Family

ID=36808717

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002117075A Abandoned CA2117075A1 (en) 1991-09-06 1992-09-02 Quinazoline derivatives and their preparation

Country Status (6)

Country Link
EP (1) EP0602125A1 (ja)
JP (1) JPH06510538A (ja)
CN (1) CN1092067A (ja)
AU (1) AU2500992A (ja)
CA (1) CA2117075A1 (ja)
WO (1) WO1993005035A1 (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9205702D0 (en) * 1992-03-16 1992-04-29 Fujisawa Pharmaceutical Co A new use of a quinazoline derivative
US5565454A (en) * 1995-05-31 1996-10-15 Ergo Science, Incorporated Method for preventing intervention-associated stenosis and other symptoms associated with stenosis of blood vessels following non-bypass, invasive interventions
US6521630B1 (en) * 1999-08-31 2003-02-18 Pfizer Inc. Tetrahydroquinazoline-2,4-diones and therapeutic uses thereof
KR100950629B1 (ko) * 2005-06-27 2010-04-01 에프. 호프만-라 로슈 아게 8-알콕시-4-메틸-3,4-다이하이드로-퀴나졸린-2-일 아민 및5-ｈｔ5ａ 수용체 리간드로서의 이의 용도

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE126796T1 (de) * 1990-01-02 1995-09-15 Fujisawa Pharmaceutical Co Quinazolinderivate und ihre herstellung.

Also Published As

Publication number Publication date
AU2500992A (en) 1993-04-05
EP0602125A1 (en) 1994-06-22
JPH06510538A (ja) 1994-11-24
CN1092067A (zh) 1994-09-14
WO1993005035A1 (en) 1993-03-18

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Legal Events

Date Code Title Description
FZDE Dead