CA2096238A1 - Process for the production of 4,5,6,7-tetrahydroimidazo-(4,5,ljk)(1,4)-benzodiazepine-2-( 1 h)-thiones as well as intermediate products - Google Patents

Process for the production of 4,5,6,7-tetrahydroimidazo-(4,5,ljk)(1,4)-benzodiazepine-2-( 1 h)-thiones as well as intermediate products

Info

Publication number
CA2096238A1
CA2096238A1 CA002096238A CA2096238A CA2096238A1 CA 2096238 A1 CA2096238 A1 CA 2096238A1 CA 002096238 A CA002096238 A CA 002096238A CA 2096238 A CA2096238 A CA 2096238A CA 2096238 A1 CA2096238 A1 CA 2096238A1
Authority
CA
Canada
Prior art keywords
denotes
compounds
residue
formula
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002096238A
Other languages
English (en)
French (fr)
Inventor
Herbert Leinert
Alfred Mertens
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roche Diagnostics GmbH
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2096238A1 publication Critical patent/CA2096238A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/26—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
    • C07C211/29—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA002096238A 1990-11-16 1991-10-29 Process for the production of 4,5,6,7-tetrahydroimidazo-(4,5,ljk)(1,4)-benzodiazepine-2-( 1 h)-thiones as well as intermediate products Abandoned CA2096238A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4036552A DE4036552C1 (enExample) 1990-11-16 1990-11-16
DEP4036552.2 1990-11-16

Publications (1)

Publication Number Publication Date
CA2096238A1 true CA2096238A1 (en) 1992-05-17

Family

ID=6418388

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002096238A Abandoned CA2096238A1 (en) 1990-11-16 1991-10-29 Process for the production of 4,5,6,7-tetrahydroimidazo-(4,5,ljk)(1,4)-benzodiazepine-2-( 1 h)-thiones as well as intermediate products

Country Status (9)

Country Link
EP (1) EP0557307A1 (enExample)
JP (1) JPH06502400A (enExample)
AU (1) AU8855991A (enExample)
CA (1) CA2096238A1 (enExample)
DE (1) DE4036552C1 (enExample)
IE (1) IE913979A1 (enExample)
IL (1) IL100033A0 (enExample)
WO (1) WO1992008706A1 (enExample)
ZA (1) ZA919050B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ238664A (en) * 1990-07-06 1992-12-23 Janssen Pharmaceutica Nv Substituted tetrahydroimidazo(1,4)benzodiazepin-2-(thi)ones and pharmaceutical anti-viral compositions
US5463049A (en) * 1991-09-24 1995-10-31 Janssen Pharmaceutica N.V. Process for preparing enantiomerically pure imidazo[4,5,1-JK][1,4]-benzodiazepin-2(1H)-thiones
UA56197C2 (uk) 1996-11-08 2003-05-15 Зенека Лімітед Гетероциклічні похідні

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8806449D0 (en) * 1988-03-18 1988-04-20 Janssen Pharmaceutica Nv Antiviral hexahydroimiazo(1 4)benzodiazepin-2-ones
IL93136A (en) * 1989-02-23 1995-01-24 Janssen Pharmaceutica Nv Tetrahydroimidazo (1,4) benzodiazepin-2-thione derivatives, their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
EP0557307A1 (de) 1993-09-01
ZA919050B (en) 1992-08-26
AU8855991A (en) 1992-06-11
IE913979A1 (en) 1992-05-20
WO1992008706A1 (de) 1992-05-29
IL100033A0 (en) 1992-08-18
DE4036552C1 (enExample) 1992-02-06
JPH06502400A (ja) 1994-03-17

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Legal Events

Date Code Title Description
FZDE Discontinued