CA2073377A1 - 2-(2-substituted pyrrolidinylthio) carbapenem derivatives - Google Patents
2-(2-substituted pyrrolidinylthio) carbapenem derivativesInfo
- Publication number
- CA2073377A1 CA2073377A1 CA002073377A CA2073377A CA2073377A1 CA 2073377 A1 CA2073377 A1 CA 2073377A1 CA 002073377 A CA002073377 A CA 002073377A CA 2073377 A CA2073377 A CA 2073377A CA 2073377 A1 CA2073377 A1 CA 2073377A1
- Authority
- CA
- Canada
- Prior art keywords
- group
- methyl
- hydroxyethyl
- carbapen
- ylthio
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
- C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
- C07D477/16—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
- C07D477/20—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP194767/1991 | 1991-07-09 | ||
| JP19476791 | 1991-07-09 | ||
| JP34959191 | 1991-12-07 | ||
| JP349591/1991 | 1991-12-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2073377A1 true CA2073377A1 (en) | 1993-01-10 |
Family
ID=26508721
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002073377A Abandoned CA2073377A1 (en) | 1991-07-09 | 1992-07-08 | 2-(2-substituted pyrrolidinylthio) carbapenem derivatives |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0522504A1 (https=) |
| KR (1) | KR930702353A (https=) |
| AU (1) | AU646577B2 (https=) |
| CA (1) | CA2073377A1 (https=) |
| CZ (1) | CZ214492A3 (https=) |
| FI (1) | FI931015A7 (https=) |
| IE (1) | IE922225A1 (https=) |
| IL (1) | IL102453A (https=) |
| NO (1) | NO930844L (https=) |
| TW (1) | TW206226B (https=) |
| WO (1) | WO1993001192A1 (https=) |
| YU (1) | YU68292A (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9216102D0 (en) * | 1992-07-29 | 1992-09-09 | Smithkline Beecham Plc | Pharmaceutical substances |
| KR950014111A (ko) * | 1993-11-23 | 1995-06-15 | 유충식 | 새로운 카바페넴 유도체 및 그 제조방법 |
| KR970010769A (ko) * | 1995-08-01 | 1997-03-27 | 유충식 | 카바페넴 유도체의 제조방법 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1281720C (en) * | 1984-11-08 | 1991-03-19 | Makoto Sunagawa | Carbapenem compounds and production thereof |
| AU631671B2 (en) * | 1989-08-04 | 1992-12-03 | Banyu Pharmaceutical Co., Ltd. | 2-(2-vinylpyrrolidinylthio)carbapenem derivatives |
-
1992
- 1992-07-07 WO PCT/JP1992/000864 patent/WO1993001192A1/en not_active Ceased
- 1992-07-07 TW TW081105391A patent/TW206226B/zh active
- 1992-07-07 EP EP92111497A patent/EP0522504A1/en not_active Withdrawn
- 1992-07-07 AU AU19471/92A patent/AU646577B2/en not_active Ceased
- 1992-07-08 CA CA002073377A patent/CA2073377A1/en not_active Abandoned
- 1992-07-08 YU YU68292A patent/YU68292A/sh unknown
- 1992-07-08 IE IE222592A patent/IE922225A1/en not_active Application Discontinuation
- 1992-07-09 IL IL10245392A patent/IL102453A/en not_active IP Right Cessation
- 1992-07-09 CZ CS922144A patent/CZ214492A3/cs unknown
-
1993
- 1993-03-08 NO NO93930844A patent/NO930844L/no unknown
- 1993-03-08 FI FI931015A patent/FI931015A7/fi not_active Application Discontinuation
- 1993-03-09 KR KR1019930700708A patent/KR930702353A/ko not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| EP0522504A1 (en) | 1993-01-13 |
| WO1993001192A1 (en) | 1993-01-21 |
| IE922225A1 (en) | 1993-01-13 |
| NO930844L (no) | 1993-05-07 |
| TW206226B (https=) | 1993-05-21 |
| KR930702353A (ko) | 1993-09-08 |
| CZ214492A3 (en) | 1993-01-13 |
| IL102453A0 (en) | 1993-01-14 |
| YU68292A (sh) | 1995-03-27 |
| AU1947192A (en) | 1993-01-14 |
| AU646577B2 (en) | 1994-02-24 |
| FI931015A0 (fi) | 1993-03-08 |
| NO930844D0 (no) | 1993-03-08 |
| FI931015A7 (fi) | 1993-03-08 |
| IL102453A (en) | 1996-01-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |