CA1175807A - SULFONE DE L'ACIDE 2-.beta.-CHLOROMETHYL-2.alpha.- METHYLPENAM-3.alpha.-CARBOXYLIQUE - Google Patents

SULFONE DE L'ACIDE 2-.beta.-CHLOROMETHYL-2.alpha.- METHYLPENAM-3.alpha.-CARBOXYLIQUE

Info

Publication number
CA1175807A
CA1175807A CA000368537A CA368537A CA1175807A CA 1175807 A CA1175807 A CA 1175807A CA 000368537 A CA000368537 A CA 000368537A CA 368537 A CA368537 A CA 368537A CA 1175807 A CA1175807 A CA 1175807A
Authority
CA
Canada
Prior art keywords
acid
ester
salt
formula
produce
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000368537A
Other languages
English (en)
Inventor
William J. Gottstein
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/214,833 external-priority patent/US4340539A/en
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Priority to CA000424446A priority Critical patent/CA1175808A/fr
Priority to CA000426209A priority patent/CA1175809A/fr
Application granted granted Critical
Publication of CA1175807A publication Critical patent/CA1175807A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Cephalosporin Compounds (AREA)
CA000368537A 1980-01-21 1981-01-15 SULFONE DE L'ACIDE 2-.beta.-CHLOROMETHYL-2.alpha.- METHYLPENAM-3.alpha.-CARBOXYLIQUE Expired CA1175807A (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
CA000424446A CA1175808A (fr) 1980-01-21 1983-03-24 DERIVES SULFONES DE L'ACIDE 2-.beta.-CHLOROMETHYL-2.alpha.- METHYLPENAM-3.alpha.-CARBOXYLIQUE
CA000426209A CA1175809A (fr) 1980-01-21 1983-04-19 2.beta.-CHLOROMETHYL-2.alpha.-METHYLPENAM-3.alpha.-ACIDE CARBOXYLIQUE SULFONE ET SELS, AINSI QUE LEURS ESTERS

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US11389480A 1980-01-21 1980-01-21
US113,894 1980-01-21
US21483180A 1980-12-11 1980-12-11
US214,833 1980-12-11
US06/214,833 US4340539A (en) 1980-01-21 1980-12-11 Derivatives of 6-bromo penicillanic acid
US214,831 1980-12-11

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CA000426209A Division CA1175809A (fr) 1980-01-21 1983-04-19 2.beta.-CHLOROMETHYL-2.alpha.-METHYLPENAM-3.alpha.-ACIDE CARBOXYLIQUE SULFONE ET SELS, AINSI QUE LEURS ESTERS

Publications (1)

Publication Number Publication Date
CA1175807A true CA1175807A (fr) 1984-10-09

Family

ID=27381401

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000368537A Expired CA1175807A (fr) 1980-01-21 1981-01-15 SULFONE DE L'ACIDE 2-.beta.-CHLOROMETHYL-2.alpha.- METHYLPENAM-3.alpha.-CARBOXYLIQUE

Country Status (12)

Country Link
KR (1) KR850001066B1 (fr)
CA (1) CA1175807A (fr)
CH (2) CH649087A5 (fr)
DE (1) DE3101527A1 (fr)
DK (3) DK162717C (fr)
GB (1) GB2070592B (fr)
HU (2) HU184380B (fr)
IL (1) IL61880A (fr)
NL (1) NL8100209A (fr)
NO (5) NO160298C (fr)
OA (1) OA06748A (fr)
SE (5) SE455702B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA826687B (en) * 1981-09-14 1983-07-27 Pfizer Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor
DE3372068D1 (en) * 1983-09-15 1987-07-23 Bristol Myers Co Pharmaceutical compositions for treating resistant bacteria including anaerobes
GB2157286B (en) * 1984-04-12 1987-12-31 Leo Pharm Prod Ltd B-lactam antibiotic potentiators

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2912511C2 (de) * 1977-06-07 1982-06-24 Pfizer Inc., 10017 New York, N.Y. Pharmazeutische Zusammensetzung, enthaltend Penicillansäure
IN149747B (fr) * 1977-06-07 1982-04-03 Pfizer
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
GB2045236A (en) * 1979-03-26 1980-10-29 Hoechst Uk Ltd Oxapenem derivatives
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide

Also Published As

Publication number Publication date
SE9000189D0 (sv) 1990-01-19
NO861945L (no) 1981-07-22
NL8100209A (nl) 1981-08-17
SE9000189L (sv) 1991-07-20
DE3101527A1 (de) 1982-02-18
NO161677B (no) 1989-06-05
OA06748A (fr) 1982-06-30
DK162769C (da) 1992-04-27
DK285890D0 (da) 1990-11-30
NO164300B (no) 1990-06-11
IL61880A (en) 1984-11-30
SE9000190D0 (sv) 1990-01-19
NO861946L (no) 1981-07-22
DK162717C (da) 1992-04-21
KR850001465A (ko) 1985-03-18
SE8100339L (sv) 1981-09-01
NO164299C (no) 1990-09-19
DK21881A (da) 1981-07-22
DK162717B (da) 1991-12-02
CH649087A5 (de) 1985-04-30
SE466203B (sv) 1992-01-13
DK162769B (da) 1991-12-09
NO164299B (no) 1990-06-11
KR850001066B1 (ko) 1985-07-25
SE9000190L (sv) 1991-07-20
NO853450L (no) 1981-07-22
NO164298B (no) 1990-06-11
NO164300C (no) 1990-09-19
DK164938B (da) 1992-09-14
SE8502286L (sv) 1985-05-08
SE8502286D0 (sv) 1985-05-08
GB2070592B (en) 1983-05-11
NO164298C (no) 1990-09-19
HU184380B (en) 1984-08-28
GB2070592A (en) 1981-09-09
SE8502285D0 (sv) 1985-05-08
NO161677C (no) 1989-09-13
CH651571A5 (de) 1985-09-30
NO861944L (no) 1981-07-22
DK285890A (da) 1990-11-30
SE455702B (sv) 1988-08-01
NO160298C (no) 1989-04-05
DK164938C (da) 1993-02-01
DK285790D0 (da) 1990-11-30
NO160298B (no) 1988-12-27
SE8502285L (sv) 1985-05-08
NO810166L (no) 1981-07-22
HU188606B (en) 1986-04-28
DK285790A (da) 1990-11-30

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Legal Events

Date Code Title Description
MKEX Expiry