CA1129407A - Antiinflammatory steroid of the androstane series - Google Patents

Antiinflammatory steroid of the androstane series

Info

Publication number
CA1129407A
CA1129407A CA321,032A CA321032A CA1129407A CA 1129407 A CA1129407 A CA 1129407A CA 321032 A CA321032 A CA 321032A CA 1129407 A CA1129407 A CA 1129407A
Authority
CA
Canada
Prior art keywords
beta
alpha
methyl
fluoro
diene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA321,032A
Other languages
English (en)
French (fr)
Inventor
Gordon H. Phillipps
Edward A. Woollett
Brian M. Bain
Alan F. English
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of CA1129407A publication Critical patent/CA1129407A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
CA321,032A 1978-02-08 1979-02-07 Antiinflammatory steroid of the androstane series Expired CA1129407A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB5131/78 1978-02-08
GB513178 1978-02-08

Publications (1)

Publication Number Publication Date
CA1129407A true CA1129407A (en) 1982-08-10

Family

ID=9790294

Family Applications (1)

Application Number Title Priority Date Filing Date
CA321,032A Expired CA1129407A (en) 1978-02-08 1979-02-07 Antiinflammatory steroid of the androstane series

Country Status (20)

Country Link
JP (1) JPS54145648A (de)
AT (1) AT367771B (de)
AU (1) AU520827B2 (de)
BE (1) BE873996A (de)
CA (1) CA1129407A (de)
CH (1) CH639669A5 (de)
DE (1) DE2904614A1 (de)
DK (1) DK145578C (de)
ES (1) ES477523A1 (de)
FI (1) FI790403A (de)
FR (1) FR2422688A1 (de)
IE (1) IE47814B1 (de)
IL (1) IL56613A (de)
IT (1) IT1114534B (de)
NL (1) NL7900967A (de)
NZ (1) NZ189586A (de)
PT (1) PT69192A (de)
SE (1) SE435626B (de)
YU (1) YU26779A (de)
ZA (1) ZA79538B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE449106B (sv) * 1980-07-10 1987-04-06 Otsuka Pharma Co Ltd Steroid med anti-inflammatorisk verkan samt komposition innehallande denna
US5237070A (en) * 1985-07-22 1993-08-17 Riker Laboratories, Inc. Substituted DI-t-butylphenols
JP4847112B2 (ja) * 2005-11-29 2011-12-28 株式会社マキタ 園芸バリカン
WO2012056201A2 (en) 2010-10-27 2012-05-03 Hovione Inter Limited Electrophilic reagents for monohalomethylation,their preparation and their uses

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1384372A (en) * 1971-01-20 1975-02-19 Glaxo Lab Ltd Dereivatives of 17alpha-hydroxyandrost-4-ene-17beta-carboxylic acids
GB1438940A (en) * 1972-07-19 1976-06-09 Glaxo Lab Ltd 17beta-haloalkoxycarbonyl-17alpha-oxysteroids

Also Published As

Publication number Publication date
IL56613A0 (en) 1979-05-31
YU26779A (en) 1983-01-21
DK145578C (da) 1983-05-09
DE2904614A1 (de) 1979-08-09
SE435626B (sv) 1984-10-08
AU520827B2 (en) 1982-03-04
IE47814B1 (en) 1984-06-27
ES477523A1 (es) 1979-07-16
BE873996A (fr) 1979-08-07
AT367771B (de) 1982-07-26
FR2422688B1 (de) 1982-07-16
CH639669A5 (en) 1983-11-30
DK50179A (da) 1979-08-09
IT1114534B (it) 1986-01-27
AU4408479A (en) 1979-08-16
IL56613A (en) 1982-12-31
ATA92379A (de) 1981-12-15
ZA79538B (en) 1980-02-27
NL7900967A (nl) 1979-08-10
FI790403A (fi) 1979-08-09
FR2422688A1 (fr) 1979-11-09
JPS54145648A (en) 1979-11-14
IE790236L (en) 1979-08-08
NZ189586A (en) 1981-01-23
IT7947909A0 (it) 1979-02-06
DK145578B (da) 1982-12-13
SE7901100L (sv) 1979-08-09
PT69192A (en) 1979-03-01

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Legal Events

Date Code Title Description
MKEX Expiry