DK145578C - Analogifremgangsmaade til fremstilling af klormetyl-17alfa-acetoxy-9alfa-fluor-11beta-hydroxy-16beta-metyl-3-oxoandrosta-1,4-dien-17beta-karboxylat - Google Patents

Analogifremgangsmaade til fremstilling af klormetyl-17alfa-acetoxy-9alfa-fluor-11beta-hydroxy-16beta-metyl-3-oxoandrosta-1,4-dien-17beta-karboxylat

Info

Publication number
DK145578C
DK145578C DK50179A DK50179A DK145578C DK 145578 C DK145578 C DK 145578C DK 50179 A DK50179 A DK 50179A DK 50179 A DK50179 A DK 50179A DK 145578 C DK145578 C DK 145578C
Authority
DK
Denmark
Prior art keywords
9alfa
chlorometyl
17alfa
16beta
oxoandrosta
Prior art date
Application number
DK50179A
Other languages
English (en)
Other versions
DK50179A (da
DK145578B (da
Inventor
G H Phillipps
B M Bain
A F English
A F Woolett
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of DK50179A publication Critical patent/DK50179A/da
Publication of DK145578B publication Critical patent/DK145578B/da
Application granted granted Critical
Publication of DK145578C publication Critical patent/DK145578C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
DK50179A 1978-02-08 1979-02-07 Analogifremgangsmaade til fremstilling af klormetyl-17alfa-acetoxy-9alfa-fluor-11beta-hydroxy-16beta-metyl-3-oxoandrosta-1,4-dien-17beta-karboxylat DK145578C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB513178 1978-02-08
GB513178 1978-02-08

Publications (3)

Publication Number Publication Date
DK50179A DK50179A (da) 1979-08-09
DK145578B DK145578B (da) 1982-12-13
DK145578C true DK145578C (da) 1983-05-09

Family

ID=9790294

Family Applications (1)

Application Number Title Priority Date Filing Date
DK50179A DK145578C (da) 1978-02-08 1979-02-07 Analogifremgangsmaade til fremstilling af klormetyl-17alfa-acetoxy-9alfa-fluor-11beta-hydroxy-16beta-metyl-3-oxoandrosta-1,4-dien-17beta-karboxylat

Country Status (20)

Country Link
JP (1) JPS54145648A (da)
AT (1) AT367771B (da)
AU (1) AU520827B2 (da)
BE (1) BE873996A (da)
CA (1) CA1129407A (da)
CH (1) CH639669A5 (da)
DE (1) DE2904614A1 (da)
DK (1) DK145578C (da)
ES (1) ES477523A1 (da)
FI (1) FI790403A (da)
FR (1) FR2422688A1 (da)
IE (1) IE47814B1 (da)
IL (1) IL56613A (da)
IT (1) IT1114534B (da)
NL (1) NL7900967A (da)
NZ (1) NZ189586A (da)
PT (1) PT69192A (da)
SE (1) SE435626B (da)
YU (1) YU26779A (da)
ZA (1) ZA79538B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE449106B (sv) * 1980-07-10 1987-04-06 Otsuka Pharma Co Ltd Steroid med anti-inflammatorisk verkan samt komposition innehallande denna
US5237070A (en) * 1985-07-22 1993-08-17 Riker Laboratories, Inc. Substituted DI-t-butylphenols
JP4847112B2 (ja) * 2005-11-29 2011-12-28 株式会社マキタ 園芸バリカン
WO2012056201A2 (en) 2010-10-27 2012-05-03 Hovione Inter Limited Electrophilic reagents for monohalomethylation,their preparation and their uses

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1384372A (en) * 1971-01-20 1975-02-19 Glaxo Lab Ltd Dereivatives of 17alpha-hydroxyandrost-4-ene-17beta-carboxylic acids
GB1438940A (en) * 1972-07-19 1976-06-09 Glaxo Lab Ltd 17beta-haloalkoxycarbonyl-17alpha-oxysteroids

Also Published As

Publication number Publication date
IL56613A0 (en) 1979-05-31
YU26779A (en) 1983-01-21
CA1129407A (en) 1982-08-10
DE2904614A1 (de) 1979-08-09
SE435626B (sv) 1984-10-08
AU520827B2 (en) 1982-03-04
IE47814B1 (en) 1984-06-27
ES477523A1 (es) 1979-07-16
BE873996A (fr) 1979-08-07
AT367771B (de) 1982-07-26
FR2422688B1 (da) 1982-07-16
CH639669A5 (en) 1983-11-30
DK50179A (da) 1979-08-09
IT1114534B (it) 1986-01-27
AU4408479A (en) 1979-08-16
IL56613A (en) 1982-12-31
ATA92379A (de) 1981-12-15
ZA79538B (en) 1980-02-27
NL7900967A (nl) 1979-08-10
FI790403A (fi) 1979-08-09
FR2422688A1 (fr) 1979-11-09
JPS54145648A (en) 1979-11-14
IE790236L (en) 1979-08-08
NZ189586A (en) 1981-01-23
IT7947909A0 (it) 1979-02-06
DK145578B (da) 1982-12-13
SE7901100L (sv) 1979-08-09
PT69192A (en) 1979-03-01

Similar Documents

Publication Publication Date Title
DK158788C (da) Analogifremgangsmaade til fremstilling af tetrazolylalkoxycarbostyrilderivater
DK149023C (da) Analogifremgangsmaade til fremstilling af tiazolidinderivater
DK153552C (da) Analogifremgangsmaade til fremstilling af 1,8-naphthyridinderivater
DK147912C (da) Fremgangsmaade til fremstilling af 1alfa-hydroxylerede vitamin d-forbindelser
DK281079A (da) Fremgangsmaade til fremstilling af 4,5-diaryl-2-nitroimidazoler
DK364579A (da) Fremgangsmaade til fremstilling af n2-arylsulfonyl-l-arginiamider
DK148480C (da) Analogifremgangsmaade til fremstilling af cycloalkyltriazoler
DK151013C (da) Analogifremgangsmaade til fremstilling af 5-methyl-isoxazol-4-carboxylsyreanilider
DK147178C (da) Fremgangsmaade til 1-hydroxylering af 5,6-trans-vitamin d-forbindelser
DK153844C (da) Analogifremgangsmaade til fremstilling af 1,2,3,5-tetrahydroimidazothienopyrimidin-2-oner
DK46777A (da) Fremgangsmade til fremstilling af meta-aryloxybenzaldehyder
DK504979A (da) Fremgangsmaade til fremstilling af 1,2,4,5-tetraalkyl-4-arylpiperidiner
DK145698C (da) Analogifremgangsmaade til fremstilling af 2-alkoxyadeninderivater
DK444479A (da) Fremgangsmaade til fremstilling af 3,4-dihydro-3-oxo-2-quinoxaliner
DK147145C (da) Analogifremgangsmaade til fremstilling af chlorambucilderivater
DK161198C (da) Analogifremgangsmaade til fremstilling af substituerede omega-aroylpropionyl-l-proliner
DK165687C (da) Fremgangsmaade til fremstilling af 2-chlorsulfinylazetidinoner
DK150479C (da) Fremgangsmaade til fremstilling af 2-chlor-5-trifluormethylpyridin
DK151256C (da) Analogifremgangsmaade til fremstilling af alkylendioxybenzenderivater
DK139029B (da) Analogifremgangsmåde til fremstilling af 5-m-tolyloxyuracil.
DK454579A (da) Fremgangsmaade til fremstilling af 6-piperidino-2,4-diaminopyrimidin-3-oxid
DK150147C (da) Analogifremgangsmaade til fremstilling af forbindelser af muramyldipeptidtypen
DK153838C (da) Analogifremgangsmaade til fremstilling af 2,4-dichlor-alfa-(n-imidazolylmethyl)-dibenzylethere
DK145578C (da) Analogifremgangsmaade til fremstilling af klormetyl-17alfa-acetoxy-9alfa-fluor-11beta-hydroxy-16beta-metyl-3-oxoandrosta-1,4-dien-17beta-karboxylat
DK165325C (da) Analogifremgangsmaade til fremstilling af 4-aza-17-substituerede 5alfa-androstan-3-oner