CA1128041A - 3h-naphtho[1,2-d]imidazoles, processes for preparing them, their use as anti-inflammatory and antimicrobial agents, etc... - Google Patents

3h-naphtho[1,2-d]imidazoles, processes for preparing them, their use as anti-inflammatory and antimicrobial agents, etc...

Info

Publication number
CA1128041A
CA1128041A CA342,360A CA342360A CA1128041A CA 1128041 A CA1128041 A CA 1128041A CA 342360 A CA342360 A CA 342360A CA 1128041 A CA1128041 A CA 1128041A
Authority
CA
Canada
Prior art keywords
formula
alkyl
methyl
naphtho
imidazole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA342,360A
Other languages
English (en)
French (fr)
Inventor
Emilio Toja
Amedeo Omodei-Sale
Domenica Selva
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruppo Lepetit SpA
Original Assignee
Gruppo Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruppo Lepetit SpA filed Critical Gruppo Lepetit SpA
Application granted granted Critical
Publication of CA1128041A publication Critical patent/CA1128041A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA342,360A 1978-12-21 1979-12-20 3h-naphtho[1,2-d]imidazoles, processes for preparing them, their use as anti-inflammatory and antimicrobial agents, etc... Expired CA1128041A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB49690/78 1978-12-21
GB7849690 1978-12-21

Publications (1)

Publication Number Publication Date
CA1128041A true CA1128041A (en) 1982-07-20

Family

ID=10501897

Family Applications (1)

Application Number Title Priority Date Filing Date
CA342,360A Expired CA1128041A (en) 1978-12-21 1979-12-20 3h-naphtho[1,2-d]imidazoles, processes for preparing them, their use as anti-inflammatory and antimicrobial agents, etc...

Country Status (11)

Country Link
US (1) US4340607A (enExample)
EP (1) EP0012866B1 (enExample)
JP (1) JPS5592376A (enExample)
AT (1) ATE2269T1 (enExample)
AU (1) AU532368B2 (enExample)
CA (1) CA1128041A (enExample)
DE (1) DE2964567D1 (enExample)
DK (1) DK157546C (enExample)
IE (1) IE49339B1 (enExample)
NO (1) NO151893C (enExample)
ZA (1) ZA796609B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0034249B1 (en) * 1980-02-08 1984-10-24 Gruppo Lepetit S.P.A. New naphthimidazole and naphthoxazole derivatives, their preparation, and their use in pharmaceuticals
IT1150955B (it) * 1980-06-06 1986-12-17 Lepetit Spa Derivati 3h-naft(1.2-d)-imidazolici il procedimento per la loro preparazione, il loro uso come agenti antiinfiammatori e le composizioni farmaceutiche che li contengono
US4435417A (en) 1981-02-20 1984-03-06 Gruppo Lepetit S.P.A. Antiinflammatory 3H-naphtho[1,2-d]imidazoles
GB8403141D0 (en) * 1984-02-07 1984-03-14 Lepetit Spa Imidazole derivatives
PH26083A (en) * 1987-11-09 1992-02-06 Sandoz Ltd 11, 28-dioxa-4-azatricyclo [22.3.1.04.9) octacos-18-ene derivatives and pharmaceutical compositions containing them and method of use thereof
IT1237805B (it) * 1989-12-21 1993-06-17 Enichem Sintesi Composto fotocromatico, metodo per la sua preparazione e articoli che lo contengono
IT1303672B1 (it) 1998-07-28 2001-02-23 Nicox Sa Sali nitrati di farmaci attivi nei disordini ossei
IT1311924B1 (it) 1999-04-13 2002-03-20 Nicox Sa Composti farmaceutici.
IT1311923B1 (it) 1999-04-13 2002-03-20 Nicox Sa Composti farmaceutici.
IT1314184B1 (it) 1999-08-12 2002-12-06 Nicox Sa Composizioni farmaceutiche per la terapia di condizioni di stressossidativo
US8387749B2 (en) 2004-03-01 2013-03-05 Ykk Corporation Of America Shock absorbing fabric structures
KR20060087386A (ko) * 2005-01-28 2006-08-02 주식회사 대웅제약 신규 벤조이미다졸 유도체 및 이를 함유하는 약제학적조성물
WO2013004462A1 (en) 2011-07-01 2013-01-10 Fondazione Istituto Insubrico Di Ricerca Per La Vita A complex of amorphous tomoxiprole and cyclodextrin with fast dissolution rate and process for the preparation thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL126227C (enExample) * 1958-08-22
GB1484615A (en) * 1974-11-23 1977-09-01 Lepetit Spa Tricyclic n-containing derivatives

Also Published As

Publication number Publication date
NO151893C (no) 1985-06-26
EP0012866A1 (en) 1980-07-09
IE792491L (en) 1980-06-21
JPH0321546B2 (enExample) 1991-03-22
AU532368B2 (en) 1983-09-29
DK157546C (da) 1990-06-25
IE49339B1 (en) 1985-09-18
JPS5592376A (en) 1980-07-12
DK542179A (da) 1980-06-22
US4340607A (en) 1982-07-20
ATE2269T1 (de) 1983-02-15
EP0012866B1 (en) 1983-01-19
NO151893B (no) 1985-03-18
AU5339579A (en) 1980-06-26
DK157546B (da) 1990-01-22
DE2964567D1 (en) 1983-02-24
ZA796609B (en) 1980-11-26
NO794205L (no) 1980-06-24

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