CA1104156A - Analogue de la bestatine - Google Patents

Analogue de la bestatine

Info

Publication number
CA1104156A
CA1104156A CA257,393A CA257393A CA1104156A CA 1104156 A CA1104156 A CA 1104156A CA 257393 A CA257393 A CA 257393A CA 1104156 A CA1104156 A CA 1104156A
Authority
CA
Canada
Prior art keywords
group
amino
benzyl
alkyl
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA257,393A
Other languages
English (en)
Inventor
Hamao Umezawa
Takaaki Aoyagi
Tomohisa Takita
Rinzo Nishizawa
Tetsushi Saino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Microbial Chemistry Research Foundation
Original Assignee
Microbial Chemistry Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Microbial Chemistry Research Foundation filed Critical Microbial Chemistry Research Foundation
Priority to CA363,896A priority Critical patent/CA1104157A/fr
Application granted granted Critical
Publication of CA1104156A publication Critical patent/CA1104156A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA257,393A 1975-07-22 1976-07-20 Analogue de la bestatine Expired CA1104156A (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CA363,896A CA1104157A (fr) 1975-07-22 1980-11-03 Analogues de la bestatine

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB30632/75A GB1510477A (en) 1975-07-22 1975-07-22 Peptides and to amino acid intermediates thereof
GB30632/75 1975-07-22

Publications (1)

Publication Number Publication Date
CA1104156A true CA1104156A (fr) 1981-06-30

Family

ID=10310676

Family Applications (1)

Application Number Title Priority Date Filing Date
CA257,393A Expired CA1104156A (fr) 1975-07-22 1976-07-20 Analogue de la bestatine

Country Status (12)

Country Link
JP (2) JPS52136118A (fr)
AU (1) AU506003B2 (fr)
CA (1) CA1104156A (fr)
CH (1) CH630892A5 (fr)
CS (2) CS201034B2 (fr)
DE (2) DE2660626C2 (fr)
DK (1) DK149110C (fr)
FR (1) FR2318863A1 (fr)
GB (1) GB1510477A (fr)
HU (1) HU183048B (fr)
NL (1) NL7608064A (fr)
SE (3) SE431642B (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2725732C2 (de) 1977-06-07 1983-01-05 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai, Tokyo Bestatin-Analoga, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate
DE2760007C2 (fr) * 1977-06-07 1988-10-06 Microbial Chem Res Found
JPS6026099B2 (ja) * 1977-09-21 1985-06-21 財団法人微生物化学研究会 ペプチド、その酸附加塩およびその製造法
NL188162C (nl) * 1978-11-25 1992-04-16 Nippon Kayaku Kk Werkwijze voor het bereiden van een bestatinederivaat.
US4370318A (en) * 1980-07-07 1983-01-25 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Bestatin-related compounds as immunopotentiator
JPS5767516A (en) * 1980-09-24 1982-04-24 Microbial Chem Res Found Novel analgesic agent
JPH0810855Y2 (ja) * 1989-07-20 1996-03-29 タナシン電機株式会社 オートリバース式テープレコーダ
DE69420524T2 (de) * 1993-06-29 2000-02-17 Kaneka Corp Verfahren zur herstellung von derivaten von 3-amin-2-hydroxy-4-phenylbuttersäure und 1-nitro-4-phenyl-2-butanol zwischenprodukte
ATE284863T1 (de) * 1996-02-08 2005-01-15 Nippon Kayaku Kk Verfahren zur erzeugung optisch aktiver cyanohydrine
US6242494B1 (en) 1998-05-01 2001-06-05 Abbott Laboratories Substituted β-amino acid inhibitors of methionine aminopeptidase-2
SK16282000A3 (sk) * 1998-05-01 2001-05-10 Abbott Laboratories Substituované beta-aminokyselinové inhibítory metionínaminopeptidázy-2

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5439477B2 (fr) * 1974-07-01 1979-11-28

Also Published As

Publication number Publication date
DK331276A (da) 1977-01-23
DK149110B (da) 1986-01-27
JPS52136118A (en) 1977-11-14
GB1510477A (en) 1978-05-10
CH630892A5 (en) 1982-07-15
AU1591276A (en) 1978-01-19
FR2318863B1 (fr) 1980-10-31
DK149110C (da) 1986-09-08
SE8306145L (sv) 1983-11-09
JPS5758338B2 (fr) 1982-12-09
FR2318863A1 (fr) 1977-02-18
CS201034B2 (en) 1980-10-31
AU506003B2 (en) 1979-12-13
JPS5823654A (ja) 1983-02-12
JPS6050780B2 (ja) 1985-11-11
SE8306145D0 (sv) 1983-11-09
SE431642B (sv) 1984-02-20
DE2632396A1 (de) 1977-02-03
DE2660626C2 (de) 1985-07-11
CS201033B2 (en) 1980-10-31
DE2632396C2 (de) 1982-11-25
HU183048B (en) 1984-04-28
SE452318B (sv) 1987-11-23
SE7606736L (sv) 1977-01-23
SE8001959L (sv) 1980-03-13
NL7608064A (nl) 1977-01-25

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Legal Events

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