CA1052376A - Process for preparing carboxamides of oxo-1,2-benzothiazine-1,1-dioxides - Google Patents

Process for preparing carboxamides of oxo-1,2-benzothiazine-1,1-dioxides

Info

Publication number
CA1052376A
CA1052376A CA235,575A CA235575A CA1052376A CA 1052376 A CA1052376 A CA 1052376A CA 235575 A CA235575 A CA 235575A CA 1052376 A CA1052376 A CA 1052376A
Authority
CA
Canada
Prior art keywords
pyridyl
methyl
carbon atoms
alkyl
thiazolyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA235,575A
Other languages
English (en)
French (fr)
Inventor
Joseph G. Lombardino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Application granted granted Critical
Publication of CA1052376A publication Critical patent/CA1052376A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/021,2-Thiazines; Hydrogenated 1,2-thiazines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA235,575A 1974-10-15 1975-09-16 Process for preparing carboxamides of oxo-1,2-benzothiazine-1,1-dioxides Expired CA1052376A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US514570A US3892740A (en) 1974-10-15 1974-10-15 Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides

Publications (1)

Publication Number Publication Date
CA1052376A true CA1052376A (en) 1979-04-10

Family

ID=24047770

Family Applications (1)

Application Number Title Priority Date Filing Date
CA235,575A Expired CA1052376A (en) 1974-10-15 1975-09-16 Process for preparing carboxamides of oxo-1,2-benzothiazine-1,1-dioxides

Country Status (28)

Country Link
US (1) US3892740A (US06312121-20011106-C00033.png)
JP (1) JPS5159878A (US06312121-20011106-C00033.png)
AR (1) AR209326A1 (US06312121-20011106-C00033.png)
AT (1) AT356123B (US06312121-20011106-C00033.png)
BE (1) BE834064A (US06312121-20011106-C00033.png)
BG (1) BG35597A3 (US06312121-20011106-C00033.png)
CA (1) CA1052376A (US06312121-20011106-C00033.png)
CH (1) CH609052A5 (US06312121-20011106-C00033.png)
CS (1) CS188254B2 (US06312121-20011106-C00033.png)
DD (1) DD122384A5 (US06312121-20011106-C00033.png)
DE (1) DE2541832A1 (US06312121-20011106-C00033.png)
DK (1) DK146535C (US06312121-20011106-C00033.png)
ES (1) ES441290A1 (US06312121-20011106-C00033.png)
FI (1) FI63573C (US06312121-20011106-C00033.png)
FR (1) FR2287907A1 (US06312121-20011106-C00033.png)
GB (2) GB1505931A (US06312121-20011106-C00033.png)
HU (1) HU172059B (US06312121-20011106-C00033.png)
IE (1) IE41690B1 (US06312121-20011106-C00033.png)
IN (1) IN141982B (US06312121-20011106-C00033.png)
LU (1) LU73491A1 (US06312121-20011106-C00033.png)
NL (1) NL7511492A (US06312121-20011106-C00033.png)
NO (1) NO154395C (US06312121-20011106-C00033.png)
NZ (1) NZ178678A (US06312121-20011106-C00033.png)
PL (1) PL102293B1 (US06312121-20011106-C00033.png)
RO (1) RO68145A (US06312121-20011106-C00033.png)
SE (2) SE423096B (US06312121-20011106-C00033.png)
SU (1) SU664563A3 (US06312121-20011106-C00033.png)
YU (1) YU40127B (US06312121-20011106-C00033.png)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4100347A (en) * 1976-06-10 1978-07-11 Pfizer Inc. 3,4-Dihydro-2-methyl-4-oxo-2H-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide
DE2756113A1 (de) * 1977-12-16 1979-06-21 Thomae Gmbh Dr K Neue 4-hydroxy-2h-1,2-benzothiazin- 3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4213980A (en) * 1978-01-30 1980-07-22 Ciba-Geigy Corporation Azathianaphthalenes
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
JPS57140785A (en) * 1981-02-24 1982-08-31 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation, and pharmaceutical composition containing the same
IN158333B (US06312121-20011106-C00033.png) * 1981-08-03 1986-10-18 Pfizer
IN159273B (US06312121-20011106-C00033.png) * 1981-10-05 1987-04-25 Pfizer
CA1197244A (en) * 1982-04-16 1985-11-26 Medichem, S.A. Process for the preparation of 4-hydroxy-2-methyl-2h- 1,2-benzothiazine-3-carboxamide-1,1-dioxides
US4551452A (en) * 1983-12-21 1985-11-05 Pfizer Inc. Anti-inflammatory 2-methyl-2H-1,2-benzo-(or -thieno-)thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US4683306A (en) * 1984-07-13 1987-07-28 Yuhan Corporation Co., Ltd. Process for the preparation of 3,4-dihydro-2-substituted-2H-1,2-thiazine-carboxylic acid 1,1-dioxide derivatives
US4761424A (en) * 1985-10-01 1988-08-02 Warner-Lambert Company Enolamides, pharmaceutical compositions and methods for treating inflammation
US4829062A (en) * 1986-05-16 1989-05-09 Pfizer Inc. Benzothiazine dioxide derivatives
US5081118A (en) * 1987-10-26 1992-01-14 Pfizer Inc. Benzothiazine dioxide derivatives
WO1990009794A1 (en) * 1989-02-28 1990-09-07 Nippon Hypox Laboratories Incorporated Remedy for diabetes
WO1997046532A1 (en) * 1996-06-03 1997-12-11 Boehringer Ingelheim Pharmaceuticals, Inc. 2-benzyl-4-sulfonyl-4h-isoquinolin-1,3-diones and their use as anti-inflammatory agents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3646020A (en) * 1970-07-16 1972-02-29 Warner Lambert Pharmaceutical 4-acyloxy-3-phenylcarbamyl-2h-1 2-benzothiazine 1 1-dioxides
US3853862A (en) * 1973-04-23 1974-12-10 Pfizer Production of 4-hydroxy-1,2-benzothiazine-3-carboxamides

Also Published As

Publication number Publication date
NO154395B (no) 1986-06-02
AR209326A1 (es) 1977-04-15
SE423096B (sv) 1982-04-13
BG35597A3 (en) 1984-05-15
JPS5159878A (en) 1976-05-25
FR2287907B1 (US06312121-20011106-C00033.png) 1979-09-14
PL102293B1 (pl) 1979-03-31
FI63573C (fi) 1985-05-15
IN141982B (US06312121-20011106-C00033.png) 1977-05-14
DK146535C (da) 1986-11-17
HU172059B (hu) 1978-05-28
LU73491A1 (US06312121-20011106-C00033.png) 1976-08-19
DK440275A (da) 1976-04-16
SE446266B (sv) 1986-08-25
RO68145A (ro) 1980-01-15
NO753250L (US06312121-20011106-C00033.png) 1976-04-21
IE41690B1 (en) 1980-02-27
FI752717A (US06312121-20011106-C00033.png) 1976-04-16
GB1505932A (en) 1978-04-05
ATA731175A (de) 1979-09-15
NL7511492A (nl) 1976-04-21
FR2287907A1 (fr) 1976-05-14
SU664563A3 (ru) 1979-05-25
CH609052A5 (US06312121-20011106-C00033.png) 1979-02-15
JPS5337354B2 (US06312121-20011106-C00033.png) 1978-10-07
AT356123B (de) 1980-04-10
IE41690L (en) 1976-04-15
NZ178678A (en) 1978-03-06
DK146535B (da) 1983-10-31
SE7510041L (sv) 1976-04-20
ES441290A1 (es) 1977-04-01
BE834064A (fr) 1976-04-01
NO154395C (no) 1986-09-10
US3892740A (en) 1975-07-01
YU242875A (en) 1982-05-31
DD122384A5 (US06312121-20011106-C00033.png) 1976-10-05
YU40127B (en) 1985-08-31
DE2541832A1 (de) 1976-04-22
CS188254B2 (en) 1979-02-28
FI63573B (fi) 1983-03-31
GB1505931A (en) 1978-04-05
SE7901131L (sv) 1979-02-08

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