BRPI1013871A2 - Processo para a preparação de derivados de ácido propiônico. - Google Patents
Processo para a preparação de derivados de ácido propiônico.Info
- Publication number
- BRPI1013871A2 BRPI1013871A2 BRPI1013871-4A BRPI1013871A BRPI1013871A2 BR PI1013871 A2 BRPI1013871 A2 BR PI1013871A2 BR PI1013871 A BRPI1013871 A BR PI1013871A BR PI1013871 A2 BRPI1013871 A2 BR PI1013871A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- propionic acid
- acid derivatives
- derivatives
- propionic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP09156074 | 2009-03-24 | ||
EP09178220 | 2009-12-07 | ||
PCT/EP2010/053598 WO2010108861A1 (en) | 2009-03-24 | 2010-03-19 | Process for the preparation of propionic acid derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI1013871A2 true BRPI1013871A2 (pt) | 2015-08-25 |
Family
ID=42110388
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI1013871-4A BRPI1013871A2 (pt) | 2009-03-24 | 2010-03-19 | Processo para a preparação de derivados de ácido propiônico. |
Country Status (23)
Country | Link |
---|---|
US (4) | US8450496B2 (pt) |
EP (1) | EP2411385B1 (pt) |
JP (1) | JP5479572B2 (pt) |
KR (1) | KR101368501B1 (pt) |
CN (1) | CN102361866B (pt) |
AR (1) | AR075915A1 (pt) |
AU (1) | AU2010227650B2 (pt) |
BR (1) | BRPI1013871A2 (pt) |
CA (1) | CA2754103C (pt) |
CL (1) | CL2011002345A1 (pt) |
DK (1) | DK2411385T3 (pt) |
ES (1) | ES2548502T3 (pt) |
HK (1) | HK1166065A1 (pt) |
IL (1) | IL214849A (pt) |
MX (1) | MX2011009898A (pt) |
PE (1) | PE20120643A1 (pt) |
PL (1) | PL2411385T3 (pt) |
RU (1) | RU2544989C2 (pt) |
SG (1) | SG174536A1 (pt) |
SI (1) | SI2411385T1 (pt) |
TW (1) | TWI415848B (pt) |
WO (1) | WO2010108861A1 (pt) |
ZA (1) | ZA201106628B (pt) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8450496B2 (en) | 2009-03-24 | 2013-05-28 | Hoffman-La Roche Inc. | Process for the preparation of propionic acid derivatives |
DK2585452T3 (en) * | 2009-12-07 | 2015-10-12 | Hoffmann La Roche | PROCESS FOR THE PREPARATION OF propionic |
WO2013181384A1 (en) | 2012-05-31 | 2013-12-05 | Ratiopharm Gmbh | Solid state forms of aleglitazar sodium |
EP2895469B1 (en) * | 2012-09-12 | 2017-10-18 | F. Hoffmann-La Roche AG | Solid forms of (s)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzo[b]thiophen-7-yl}-propionic acid and of salts thereof |
WO2015137496A1 (ja) * | 2014-03-14 | 2015-09-17 | 武田薬品工業株式会社 | 複素環化合物の製造法 |
CN106582852B (zh) * | 2016-12-09 | 2019-04-05 | 黑龙江省科学院石油化学研究院 | 一种二茂铁双膦-铑(ⅰ)手性催化剂的制备方法 |
NL2024731B1 (en) | 2020-01-22 | 2021-09-09 | Sonova Ag | Acoustic device with deformable shape as valve |
NL2024842B1 (en) | 2020-02-05 | 2021-09-13 | Sonova Ag | Acoustic device with sma microspring switch |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE59309554D1 (de) * | 1992-04-02 | 1999-06-10 | Novartis Ag | Ferrocenyldiphosphine als Liganden für homogene Katalysatoren |
DE59410267D1 (de) * | 1993-02-26 | 2003-05-15 | Syngenta Participations Ag | Ferrocenyldiphosphine als Liganden für homogene Katalysatoren |
NZ529033A (en) | 2001-05-15 | 2005-06-24 | F | Carboxylic acid substituted oxazole derivatives for use as PPAR-alpha and -gamma activators in the treatment of diabetes |
EP1622920B1 (en) * | 2003-05-09 | 2006-08-23 | Umicore AG & Co. KG | Substituted ferrocenyldiphosphines as ligands for homogeneous hydrogenation catalysts |
US7262303B2 (en) * | 2003-09-29 | 2007-08-28 | Hoffman-La Roche Inc. | Process for the production of chiral propionic acid derivatives |
GB0500700D0 (en) * | 2005-01-14 | 2005-02-23 | Stylacats Ltd | Process for the manufacture of 2-alkyl-3-phenylpropionic acids and alcohols |
CN100432083C (zh) * | 2006-07-11 | 2008-11-12 | 南开大学 | 螺环膦-噁唑啉配体及其在不对称催化氢化中的应用 |
EP1939182A1 (de) * | 2006-12-22 | 2008-07-02 | Speedel Experimenta AG | Verfahren zur Herstellung von (R oder S)-2-Alkyl-3-heterocyclyl-1-propanolen |
US7977499B2 (en) * | 2007-02-20 | 2011-07-12 | Solvias Ag | Bis(ferrocenylphosphino) ferrocene ligands used in asymmetric hydrogenation reactions |
PE20091364A1 (es) * | 2008-01-17 | 2009-10-13 | Novartis Ag | Proceso para la preparacion de inhibidores de nep |
CN101565434B (zh) | 2008-04-25 | 2012-05-30 | 浙江九洲药业股份有限公司 | 螺环膦-噁唑啉和制备方法及其应用 |
US8450496B2 (en) | 2009-03-24 | 2013-05-28 | Hoffman-La Roche Inc. | Process for the preparation of propionic acid derivatives |
-
2010
- 2010-03-17 US US12/725,480 patent/US8450496B2/en not_active Expired - Fee Related
- 2010-03-19 RU RU2011142614/04A patent/RU2544989C2/ru not_active IP Right Cessation
- 2010-03-19 PL PL10709535T patent/PL2411385T3/pl unknown
- 2010-03-19 JP JP2012501258A patent/JP5479572B2/ja not_active Expired - Fee Related
- 2010-03-19 CA CA2754103A patent/CA2754103C/en not_active Expired - Fee Related
- 2010-03-19 ES ES10709535.8T patent/ES2548502T3/es active Active
- 2010-03-19 WO PCT/EP2010/053598 patent/WO2010108861A1/en active Application Filing
- 2010-03-19 PE PE2011001680A patent/PE20120643A1/es active IP Right Grant
- 2010-03-19 EP EP10709535.8A patent/EP2411385B1/en not_active Not-in-force
- 2010-03-19 CN CN201080013420.3A patent/CN102361866B/zh not_active Expired - Fee Related
- 2010-03-19 DK DK10709535.8T patent/DK2411385T3/en active
- 2010-03-19 KR KR1020117024733A patent/KR101368501B1/ko active IP Right Grant
- 2010-03-19 BR BRPI1013871-4A patent/BRPI1013871A2/pt active Search and Examination
- 2010-03-19 AU AU2010227650A patent/AU2010227650B2/en not_active Ceased
- 2010-03-19 SG SG2011068939A patent/SG174536A1/en unknown
- 2010-03-19 MX MX2011009898A patent/MX2011009898A/es active IP Right Grant
- 2010-03-19 SI SI201031004T patent/SI2411385T1/sl unknown
- 2010-03-22 AR ARP100100913A patent/AR075915A1/es unknown
- 2010-03-22 TW TW099108411A patent/TWI415848B/zh not_active IP Right Cessation
-
2011
- 2011-08-25 IL IL214849A patent/IL214849A/en not_active IP Right Cessation
- 2011-09-09 ZA ZA2011/06628A patent/ZA201106628B/en unknown
- 2011-09-23 CL CL2011002345A patent/CL2011002345A1/es unknown
-
2012
- 2012-07-09 HK HK12106673.7A patent/HK1166065A1/xx not_active IP Right Cessation
-
2013
- 2013-03-11 US US13/792,292 patent/US20130184468A1/en not_active Abandoned
-
2014
- 2014-10-08 US US14/509,763 patent/US20150025249A1/en not_active Abandoned
-
2018
- 2018-12-11 US US16/216,214 patent/US20190106416A1/en not_active Abandoned
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B11D | Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time |