BRPI1013871A2 - Processo para a preparação de derivados de ácido propiônico. - Google Patents

Processo para a preparação de derivados de ácido propiônico.

Info

Publication number
BRPI1013871A2
BRPI1013871A2 BRPI1013871-4A BRPI1013871A BRPI1013871A2 BR PI1013871 A2 BRPI1013871 A2 BR PI1013871A2 BR PI1013871 A BRPI1013871 A BR PI1013871A BR PI1013871 A2 BRPI1013871 A2 BR PI1013871A2
Authority
BR
Brazil
Prior art keywords
preparation
propionic acid
acid derivatives
derivatives
propionic
Prior art date
Application number
BRPI1013871-4A
Other languages
English (en)
Inventor
Kurt Puentener
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42110388&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI1013871(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI1013871A2 publication Critical patent/BRPI1013871A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BRPI1013871-4A 2009-03-24 2010-03-19 Processo para a preparação de derivados de ácido propiônico. BRPI1013871A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09156074 2009-03-24
EP09178220 2009-12-07
PCT/EP2010/053598 WO2010108861A1 (en) 2009-03-24 2010-03-19 Process for the preparation of propionic acid derivatives

Publications (1)

Publication Number Publication Date
BRPI1013871A2 true BRPI1013871A2 (pt) 2015-08-25

Family

ID=42110388

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1013871-4A BRPI1013871A2 (pt) 2009-03-24 2010-03-19 Processo para a preparação de derivados de ácido propiônico.

Country Status (23)

Country Link
US (4) US8450496B2 (pt)
EP (1) EP2411385B1 (pt)
JP (1) JP5479572B2 (pt)
KR (1) KR101368501B1 (pt)
CN (1) CN102361866B (pt)
AR (1) AR075915A1 (pt)
AU (1) AU2010227650B2 (pt)
BR (1) BRPI1013871A2 (pt)
CA (1) CA2754103C (pt)
CL (1) CL2011002345A1 (pt)
DK (1) DK2411385T3 (pt)
ES (1) ES2548502T3 (pt)
HK (1) HK1166065A1 (pt)
IL (1) IL214849A (pt)
MX (1) MX2011009898A (pt)
PE (1) PE20120643A1 (pt)
PL (1) PL2411385T3 (pt)
RU (1) RU2544989C2 (pt)
SG (1) SG174536A1 (pt)
SI (1) SI2411385T1 (pt)
TW (1) TWI415848B (pt)
WO (1) WO2010108861A1 (pt)
ZA (1) ZA201106628B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8450496B2 (en) 2009-03-24 2013-05-28 Hoffman-La Roche Inc. Process for the preparation of propionic acid derivatives
DK2585452T3 (en) * 2009-12-07 2015-10-12 Hoffmann La Roche PROCESS FOR THE PREPARATION OF propionic
WO2013181384A1 (en) 2012-05-31 2013-12-05 Ratiopharm Gmbh Solid state forms of aleglitazar sodium
EP2895469B1 (en) * 2012-09-12 2017-10-18 F. Hoffmann-La Roche AG Solid forms of (s)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzo[b]thiophen-7-yl}-propionic acid and of salts thereof
WO2015137496A1 (ja) * 2014-03-14 2015-09-17 武田薬品工業株式会社 複素環化合物の製造法
CN106582852B (zh) * 2016-12-09 2019-04-05 黑龙江省科学院石油化学研究院 一种二茂铁双膦-铑(ⅰ)手性催化剂的制备方法
NL2024731B1 (en) 2020-01-22 2021-09-09 Sonova Ag Acoustic device with deformable shape as valve
NL2024842B1 (en) 2020-02-05 2021-09-13 Sonova Ag Acoustic device with sma microspring switch

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE59309554D1 (de) * 1992-04-02 1999-06-10 Novartis Ag Ferrocenyldiphosphine als Liganden für homogene Katalysatoren
DE59410267D1 (de) * 1993-02-26 2003-05-15 Syngenta Participations Ag Ferrocenyldiphosphine als Liganden für homogene Katalysatoren
NZ529033A (en) 2001-05-15 2005-06-24 F Carboxylic acid substituted oxazole derivatives for use as PPAR-alpha and -gamma activators in the treatment of diabetes
EP1622920B1 (en) * 2003-05-09 2006-08-23 Umicore AG & Co. KG Substituted ferrocenyldiphosphines as ligands for homogeneous hydrogenation catalysts
US7262303B2 (en) * 2003-09-29 2007-08-28 Hoffman-La Roche Inc. Process for the production of chiral propionic acid derivatives
GB0500700D0 (en) * 2005-01-14 2005-02-23 Stylacats Ltd Process for the manufacture of 2-alkyl-3-phenylpropionic acids and alcohols
CN100432083C (zh) * 2006-07-11 2008-11-12 南开大学 螺环膦-噁唑啉配体及其在不对称催化氢化中的应用
EP1939182A1 (de) * 2006-12-22 2008-07-02 Speedel Experimenta AG Verfahren zur Herstellung von (R oder S)-2-Alkyl-3-heterocyclyl-1-propanolen
US7977499B2 (en) * 2007-02-20 2011-07-12 Solvias Ag Bis(ferrocenylphosphino) ferrocene ligands used in asymmetric hydrogenation reactions
PE20091364A1 (es) * 2008-01-17 2009-10-13 Novartis Ag Proceso para la preparacion de inhibidores de nep
CN101565434B (zh) 2008-04-25 2012-05-30 浙江九洲药业股份有限公司 螺环膦-噁唑啉和制备方法及其应用
US8450496B2 (en) 2009-03-24 2013-05-28 Hoffman-La Roche Inc. Process for the preparation of propionic acid derivatives

Also Published As

Publication number Publication date
IL214849A0 (en) 2011-11-30
DK2411385T3 (en) 2015-08-17
TWI415848B (zh) 2013-11-21
KR101368501B1 (ko) 2014-02-27
CN102361866A (zh) 2012-02-22
US20130184468A1 (en) 2013-07-18
ES2548502T3 (es) 2015-10-19
CA2754103A1 (en) 2010-09-30
JP5479572B2 (ja) 2014-04-23
US8450496B2 (en) 2013-05-28
JP2012521385A (ja) 2012-09-13
AU2010227650B2 (en) 2015-06-04
AU2010227650A1 (en) 2011-09-22
CN102361866B (zh) 2015-03-25
US20100249428A1 (en) 2010-09-30
IL214849A (en) 2015-10-29
SI2411385T1 (sl) 2015-10-30
KR20110130500A (ko) 2011-12-05
AR075915A1 (es) 2011-05-04
RU2544989C2 (ru) 2015-03-20
WO2010108861A1 (en) 2010-09-30
CA2754103C (en) 2017-07-11
CL2011002345A1 (es) 2012-03-30
ZA201106628B (en) 2012-05-30
MX2011009898A (es) 2011-09-30
RU2011142614A (ru) 2013-04-27
SG174536A1 (en) 2011-10-28
HK1166065A1 (en) 2012-10-19
PL2411385T3 (pl) 2016-01-29
EP2411385A1 (en) 2012-02-01
PE20120643A1 (es) 2012-05-31
US20190106416A1 (en) 2019-04-11
US20150025249A1 (en) 2015-01-22
EP2411385B1 (en) 2015-08-05
TW201036963A (en) 2010-10-16

Similar Documents

Publication Publication Date Title
BRPI0909655A2 (pt) Processo para a preparação regioseletiva de derivados de ácido 1-alquil-3-haloalquil-pirazol-4carboxílico
BRPI1011936A2 (pt) métodos biológicos para a preparação de ácido adípico
BRPI0914917A2 (pt) processo para a produção de ácidos carboxílicos livres.
BR112012014490A2 (pt) processo para a preparação substituída de 1-o-acil-2-desóxi-2-fluoro-4-tio-beta-d-arabinofuranoses
BRPI0911759A2 (pt) microorganismo para a produção de ácido metacrílico
DOP2011000086A (es) Derivados de acido 1-amino-2-ciclobutiletilboronico
BRPI1013561A2 (pt) Processo para a preparação de alogliptina
BRPI0817747A2 (pt) Processo para a preparação de derivados de ácido 2-di-halogenoacil-3-amino-acrílico
BRPI0916360A2 (pt) processo para preparar derivados de ácido r-beta-amino fenilbutírico
BR112013013256A2 (pt) método para a produção de ácido 2-bromo-4,5-dialcoxi- benzóico
BRPI1014812A2 (pt) Processo para a produção de alacoóis
BRPI1013871A2 (pt) Processo para a preparação de derivados de ácido propiônico.
BR112012000210A2 (pt) processo para a produção de heterodímeoros de ácido glutâmico.
BR112012016247A2 (pt) processo contínuo para a produção de derivados de ácidos carboxílicos saturados
BR112012002500A2 (pt) Processo para o preparo de derivados de ácido 1- (2-halobifenil-4-yl) - ciclopropanocarboxílico
BRPI1014691A2 (pt) Composto, e, processo para a preparação de um composto.
BR112014001571A2 (pt) processo para preparar derivados de ácido carboxílico
BR112012001274A2 (pt) processo para produção de ácidos decancarboxílicos
BR112012001731A2 (pt) Processo para a preparação de 1-benzil-3-hidroximetil-1h-indazol
BRPI0821752A2 (pt) Processo para preparar derivados de ácido 22-fluoracil-3-amino-acrílico
BRPI1010571A2 (pt) processo para a preparação de um composto útil como um inibidor de tafla.
BRPI0913644A2 (pt) processo para a prepração de derivados de pirimidina substituída.
BRPI0914792A2 (pt) processo para a preparação de polióis
BRPI0909813A2 (pt) processo para a preparação de derivados de ácido ciclohexanocarboxílico
BRPI1008557A2 (pt) processo para a preparação de 5-/6-nitrofluoresceína

Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06T Formal requirements before examination [chapter 6.20 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B11D Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time