BRPI0909813A2 - processo para a preparação de derivados de ácido ciclohexanocarboxílico - Google Patents
processo para a preparação de derivados de ácido ciclohexanocarboxílicoInfo
- Publication number
- BRPI0909813A2 BRPI0909813A2 BRPI0909813A BRPI0909813A BRPI0909813A2 BR PI0909813 A2 BRPI0909813 A2 BR PI0909813A2 BR PI0909813 A BRPI0909813 A BR PI0909813A BR PI0909813 A BRPI0909813 A BR PI0909813A BR PI0909813 A2 BRPI0909813 A2 BR PI0909813A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- acid derivatives
- cyclohexanecarboxylic acid
- cyclohexanecarboxylic
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/57—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C233/58—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C253/00—Preparation of carboxylic acid nitriles
- C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/06—Preparation of carboxylic acids or their salts, halides or anhydrides from carboxylic acid amides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP08154078.3 | 2008-04-04 | ||
EP08154078 | 2008-04-04 | ||
EP09151065.1 | 2009-01-22 | ||
EP09151065 | 2009-01-22 | ||
PCT/EP2009/053581 WO2009121788A1 (en) | 2008-04-04 | 2009-03-26 | New process for the preparatiion of cyclohexanecarboxylic acid dericatives |
Publications (2)
Publication Number | Publication Date |
---|---|
BRPI0909813A2 true BRPI0909813A2 (pt) | 2015-10-06 |
BRPI0909813B1 BRPI0909813B1 (pt) | 2018-01-02 |
Family
ID=40749840
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0909813-5A BRPI0909813B1 (pt) | 2008-04-04 | 2009-03-26 | "processos para preparação de derivados de ácido ciclo-hexanocarboxílico, e intermediário" |
Country Status (12)
Country | Link |
---|---|
US (1) | US8143442B2 (pt) |
EP (1) | EP2274278B1 (pt) |
JP (1) | JP5564487B2 (pt) |
KR (1) | KR101279751B1 (pt) |
CN (1) | CN101981001B (pt) |
AU (1) | AU2009231423B2 (pt) |
BR (1) | BRPI0909813B1 (pt) |
CA (1) | CA2717955C (pt) |
ES (1) | ES2592727T3 (pt) |
IL (1) | IL207431A (pt) |
MX (1) | MX2010009926A (pt) |
WO (1) | WO2009121788A1 (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20130100124A (ko) * | 2010-09-16 | 2013-09-09 | 에프. 호프만-라 로슈 아게 | 신규 방법 |
MX2013006038A (es) | 2010-12-16 | 2013-08-01 | Hoffmann La Roche | Proceso para la preparacion de derivados de tiol aromaticos por hidrogenacion de disulfuros. |
US8975438B2 (en) * | 2011-07-13 | 2015-03-10 | Hoffmann-La Roche Inc. | Process for the preparation of cyclohexanecarboxylic acid derivatives |
JP6449235B2 (ja) | 2013-03-27 | 2019-01-09 | エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft | 治療に対する応答性を予測するための遺伝マーカー |
CN105277462A (zh) * | 2014-06-19 | 2016-01-27 | 浙江海洋学院 | 一种罐底老化油泥的组成含量分析方法 |
PT3174995T (pt) | 2014-07-30 | 2020-10-15 | Hoffmann La Roche | Marcadores genéticos para prever o tipo de resposta ao tratamento com um fármaco de aumento do hdl ou mimetizador do hdl |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2899458A (en) * | 1959-08-11 | Process for producing oxy aromatic | ||
US4129595A (en) * | 1978-03-29 | 1978-12-12 | Chevron Research Company | Preparation of chloroacetyl chloride |
CH641756A5 (fr) * | 1978-04-27 | 1984-03-15 | Sanofi Sa | Composes derives de l'acide cyclohexylcarboxylique, et medicaments les contenant. |
DE3218540A1 (de) * | 1982-05-17 | 1983-11-24 | Hoechst Ag, 6230 Frankfurt | Spiro-2-aza-alkan-3-carbonitrile, verfahren zu ihrer herstellung und ihre verwendung |
JP2894445B2 (ja) * | 1997-02-12 | 1999-05-24 | 日本たばこ産業株式会社 | Cetp活性阻害剤として有効な化合物 |
IT1292037B1 (it) | 1997-05-30 | 1999-01-25 | Bracco Spa | Processo per la preparazione di 5-(acetil 62,3-diidrossipropil)- ammino)-n,n'-bis(2,3-diidrossipropil)-2,4,6-triiodo-1,3-benzen- |
GB0229803D0 (en) | 2002-12-20 | 2003-01-29 | Syngenta Ltd | Chemical process |
ITMI20031333A1 (it) | 2003-06-30 | 2005-01-01 | Erregierre Spa | Processo di preparazione di raloxifene cloridrato. |
US7435849B2 (en) * | 2005-10-31 | 2008-10-14 | Hoffmann-La Roche Inc. | Process for the production of acid chlorides |
EP1935867A1 (en) * | 2006-12-20 | 2008-06-25 | F. Hoffmann-La Roche Ag | Process for preparing 1-(2-ethyl-butyl)-cyclohexanecarboxylic acid |
JP5526120B2 (ja) * | 2008-04-04 | 2014-06-18 | エフ.ホフマン−ラ ロシュ アーゲー | 対応するシクロヘキサンカルボキシアミド誘導体を経るシクロヘキサンカルボン酸誘導体の新規な製造方法 |
-
2009
- 2009-03-26 WO PCT/EP2009/053581 patent/WO2009121788A1/en active Application Filing
- 2009-03-26 MX MX2010009926A patent/MX2010009926A/es active IP Right Grant
- 2009-03-26 EP EP09728035.8A patent/EP2274278B1/en active Active
- 2009-03-26 KR KR1020107021983A patent/KR101279751B1/ko active IP Right Grant
- 2009-03-26 AU AU2009231423A patent/AU2009231423B2/en active Active
- 2009-03-26 CN CN200980111292.3A patent/CN101981001B/zh active Active
- 2009-03-26 ES ES09728035.8T patent/ES2592727T3/es active Active
- 2009-03-26 JP JP2011502347A patent/JP5564487B2/ja active Active
- 2009-03-26 BR BRPI0909813-5A patent/BRPI0909813B1/pt active IP Right Grant
- 2009-03-26 CA CA2717955A patent/CA2717955C/en active Active
- 2009-03-31 US US12/414,698 patent/US8143442B2/en active Active
-
2010
- 2010-08-05 IL IL207431A patent/IL207431A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
JP2011516447A (ja) | 2011-05-26 |
MX2010009926A (es) | 2010-09-28 |
BRPI0909813B1 (pt) | 2018-01-02 |
JP5564487B2 (ja) | 2014-07-30 |
EP2274278B1 (en) | 2016-08-17 |
WO2009121788A1 (en) | 2009-10-08 |
ES2592727T3 (es) | 2016-12-01 |
EP2274278A1 (en) | 2011-01-19 |
IL207431A (en) | 2014-11-30 |
US20090253928A1 (en) | 2009-10-08 |
US8143442B2 (en) | 2012-03-27 |
KR101279751B1 (ko) | 2013-07-04 |
IL207431A0 (en) | 2010-12-30 |
CA2717955A1 (en) | 2009-10-08 |
KR20100120311A (ko) | 2010-11-15 |
AU2009231423B2 (en) | 2014-01-30 |
CN101981001B (zh) | 2016-06-08 |
CA2717955C (en) | 2016-08-09 |
AU2009231423A1 (en) | 2009-10-08 |
CN101981001A (zh) | 2011-02-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |