BRPI0909813A2 - processo para a preparação de derivados de ácido ciclohexanocarboxílico - Google Patents

processo para a preparação de derivados de ácido ciclohexanocarboxílico

Info

Publication number
BRPI0909813A2
BRPI0909813A2 BRPI0909813A BRPI0909813A BRPI0909813A2 BR PI0909813 A2 BRPI0909813 A2 BR PI0909813A2 BR PI0909813 A BRPI0909813 A BR PI0909813A BR PI0909813 A BRPI0909813 A BR PI0909813A BR PI0909813 A2 BRPI0909813 A2 BR PI0909813A2
Authority
BR
Brazil
Prior art keywords
preparation
acid derivatives
cyclohexanecarboxylic acid
cyclohexanecarboxylic
derivatives
Prior art date
Application number
BRPI0909813A
Other languages
English (en)
Inventor
Dennis Smith Consulting Limited
Gerald John Harnett
Helmut Stahr
Michael Jansen
Reinhard Reents
Tim Sattelkau
Ursula Hoffmann
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0909813A2 publication Critical patent/BRPI0909813A2/pt
Publication of BRPI0909813B1 publication Critical patent/BRPI0909813B1/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/57Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C233/58Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00Preparation of carboxylic acid nitriles
    • C07C253/30Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/06Preparation of carboxylic acids or their salts, halides or anhydrides from carboxylic acid amides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BRPI0909813-5A 2008-04-04 2009-03-26 "processos para preparação de derivados de ácido ciclo-hexanocarboxílico, e intermediário" BRPI0909813B1 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP08154078.3 2008-04-04
EP08154078 2008-04-04
EP09151065.1 2009-01-22
EP09151065 2009-01-22
PCT/EP2009/053581 WO2009121788A1 (en) 2008-04-04 2009-03-26 New process for the preparatiion of cyclohexanecarboxylic acid dericatives

Publications (2)

Publication Number Publication Date
BRPI0909813A2 true BRPI0909813A2 (pt) 2015-10-06
BRPI0909813B1 BRPI0909813B1 (pt) 2018-01-02

Family

ID=40749840

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0909813-5A BRPI0909813B1 (pt) 2008-04-04 2009-03-26 "processos para preparação de derivados de ácido ciclo-hexanocarboxílico, e intermediário"

Country Status (12)

Country Link
US (1) US8143442B2 (pt)
EP (1) EP2274278B1 (pt)
JP (1) JP5564487B2 (pt)
KR (1) KR101279751B1 (pt)
CN (1) CN101981001B (pt)
AU (1) AU2009231423B2 (pt)
BR (1) BRPI0909813B1 (pt)
CA (1) CA2717955C (pt)
ES (1) ES2592727T3 (pt)
IL (1) IL207431A (pt)
MX (1) MX2010009926A (pt)
WO (1) WO2009121788A1 (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20130100124A (ko) * 2010-09-16 2013-09-09 에프. 호프만-라 로슈 아게 신규 방법
MX2013006038A (es) 2010-12-16 2013-08-01 Hoffmann La Roche Proceso para la preparacion de derivados de tiol aromaticos por hidrogenacion de disulfuros.
US8975438B2 (en) * 2011-07-13 2015-03-10 Hoffmann-La Roche Inc. Process for the preparation of cyclohexanecarboxylic acid derivatives
JP6449235B2 (ja) 2013-03-27 2019-01-09 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft 治療に対する応答性を予測するための遺伝マーカー
CN105277462A (zh) * 2014-06-19 2016-01-27 浙江海洋学院 一种罐底老化油泥的组成含量分析方法
PT3174995T (pt) 2014-07-30 2020-10-15 Hoffmann La Roche Marcadores genéticos para prever o tipo de resposta ao tratamento com um fármaco de aumento do hdl ou mimetizador do hdl

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2899458A (en) * 1959-08-11 Process for producing oxy aromatic
US4129595A (en) * 1978-03-29 1978-12-12 Chevron Research Company Preparation of chloroacetyl chloride
CH641756A5 (fr) * 1978-04-27 1984-03-15 Sanofi Sa Composes derives de l'acide cyclohexylcarboxylique, et medicaments les contenant.
DE3218540A1 (de) * 1982-05-17 1983-11-24 Hoechst Ag, 6230 Frankfurt Spiro-2-aza-alkan-3-carbonitrile, verfahren zu ihrer herstellung und ihre verwendung
JP2894445B2 (ja) * 1997-02-12 1999-05-24 日本たばこ産業株式会社 Cetp活性阻害剤として有効な化合物
IT1292037B1 (it) 1997-05-30 1999-01-25 Bracco Spa Processo per la preparazione di 5-(acetil 62,3-diidrossipropil)- ammino)-n,n'-bis(2,3-diidrossipropil)-2,4,6-triiodo-1,3-benzen-
GB0229803D0 (en) 2002-12-20 2003-01-29 Syngenta Ltd Chemical process
ITMI20031333A1 (it) 2003-06-30 2005-01-01 Erregierre Spa Processo di preparazione di raloxifene cloridrato.
US7435849B2 (en) * 2005-10-31 2008-10-14 Hoffmann-La Roche Inc. Process for the production of acid chlorides
EP1935867A1 (en) * 2006-12-20 2008-06-25 F. Hoffmann-La Roche Ag Process for preparing 1-(2-ethyl-butyl)-cyclohexanecarboxylic acid
JP5526120B2 (ja) * 2008-04-04 2014-06-18 エフ.ホフマン−ラ ロシュ アーゲー 対応するシクロヘキサンカルボキシアミド誘導体を経るシクロヘキサンカルボン酸誘導体の新規な製造方法

Also Published As

Publication number Publication date
JP2011516447A (ja) 2011-05-26
MX2010009926A (es) 2010-09-28
BRPI0909813B1 (pt) 2018-01-02
JP5564487B2 (ja) 2014-07-30
EP2274278B1 (en) 2016-08-17
WO2009121788A1 (en) 2009-10-08
ES2592727T3 (es) 2016-12-01
EP2274278A1 (en) 2011-01-19
IL207431A (en) 2014-11-30
US20090253928A1 (en) 2009-10-08
US8143442B2 (en) 2012-03-27
KR101279751B1 (ko) 2013-07-04
IL207431A0 (en) 2010-12-30
CA2717955A1 (en) 2009-10-08
KR20100120311A (ko) 2010-11-15
AU2009231423B2 (en) 2014-01-30
CN101981001B (zh) 2016-06-08
CA2717955C (en) 2016-08-09
AU2009231423A1 (en) 2009-10-08
CN101981001A (zh) 2011-02-23

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]