BRPI0921879A2 - composto, composição farmacêutica , e, uso de um composto - Google Patents

composto, composição farmacêutica , e, uso de um composto

Info

Publication number
BRPI0921879A2
BRPI0921879A2 BRPI0921879A BRPI0921879A BRPI0921879A2 BR PI0921879 A2 BRPI0921879 A2 BR PI0921879A2 BR PI0921879 A BRPI0921879 A BR PI0921879A BR PI0921879 A BRPI0921879 A BR PI0921879A BR PI0921879 A2 BRPI0921879 A2 BR PI0921879A2
Authority
BR
Brazil
Prior art keywords
compound
pharmaceutical composition
pharmaceutical
composition
Prior art date
Application number
BRPI0921879A
Other languages
English (en)
Portuguese (pt)
Inventor
Swahn Britt-Marie
Rotticci Didier
Lindstrom Johan
Holenz Jorg
Kolmodin Karen
Rakos Laszlo
Soderman Peter
Karlstrom Sofia
Von Berg Stefan
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42170158&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0921879(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0921879A2 publication Critical patent/BRPI0921879A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BRPI0921879A 2008-11-14 2009-11-13 composto, composição farmacêutica , e, uso de um composto BRPI0921879A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US11463408P 2008-11-14 2008-11-14
US13976708P 2008-12-22 2008-12-22
US22165309P 2009-06-30 2009-06-30
PCT/SE2009/051295 WO2010056196A1 (en) 2008-11-14 2009-11-13 New compounds 578

Publications (1)

Publication Number Publication Date
BRPI0921879A2 true BRPI0921879A2 (pt) 2018-10-16

Family

ID=42170158

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0921879A BRPI0921879A2 (pt) 2008-11-14 2009-11-13 composto, composição farmacêutica , e, uso de um composto

Country Status (24)

Country Link
US (2) US8030500B2 (enExample)
EP (1) EP2367814A4 (enExample)
JP (1) JP2012508734A (enExample)
KR (1) KR20110091540A (enExample)
CN (1) CN102282140A (enExample)
AR (1) AR074341A1 (enExample)
AU (1) AU2009314664A1 (enExample)
BR (1) BRPI0921879A2 (enExample)
CA (1) CA2743938A1 (enExample)
CL (1) CL2011001098A1 (enExample)
CO (1) CO6362004A2 (enExample)
CR (1) CR20110255A (enExample)
CU (1) CU20110106A7 (enExample)
DO (1) DOP2011000138A (enExample)
EA (1) EA201190020A1 (enExample)
EC (1) ECSP11011051A (enExample)
IL (1) IL212590A0 (enExample)
MX (1) MX2011004918A (enExample)
NI (1) NI201100099A (enExample)
PE (1) PE20110875A1 (enExample)
TW (1) TW201020244A (enExample)
UY (1) UY32241A (enExample)
WO (1) WO2010056196A1 (enExample)
ZA (1) ZA201104396B (enExample)

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EP2689780A1 (en) 2007-04-24 2014-01-29 Shionogi & Co., Ltd. Intermediates for aminodihydrothiazine derivatives substituted with a cyclic group
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CN103261199A (zh) 2010-10-29 2013-08-21 盐野义制药株式会社 萘啶衍生物
EP2634188A4 (en) 2010-10-29 2014-05-07 Shionogi & Co FUSIONED AMINODIHYDROPYRIMIDINE DERIVATIVE
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CN103608345A (zh) 2011-04-26 2014-02-26 盐野义制药株式会社 噁嗪衍生物和含有该噁嗪衍生物的bace1抑制剂
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CN105272884B (zh) * 2015-11-02 2017-05-24 浙江大学 一种邻氰基二苯甲酮衍生物的制备方法
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Also Published As

Publication number Publication date
EA201190020A1 (ru) 2012-02-28
CL2011001098A1 (es) 2012-02-24
ECSP11011051A (es) 2011-06-30
MX2011004918A (es) 2011-05-30
AR074341A1 (es) 2011-01-12
US20110319426A1 (en) 2011-12-29
IL212590A0 (en) 2011-07-31
CA2743938A1 (en) 2010-05-20
DOP2011000138A (es) 2011-06-30
EP2367814A4 (en) 2012-07-04
CN102282140A (zh) 2011-12-14
CO6362004A2 (es) 2012-01-20
CU20110106A7 (es) 2012-01-31
TW201020244A (en) 2010-06-01
NI201100099A (es) 2012-03-19
PE20110875A1 (es) 2012-01-11
UY32241A (es) 2010-06-30
CR20110255A (es) 2011-07-04
AU2009314664A1 (en) 2011-06-23
JP2012508734A (ja) 2012-04-12
EP2367814A1 (en) 2011-09-28
ZA201104396B (en) 2012-03-28
WO2010056196A1 (en) 2010-05-20
US20100125082A1 (en) 2010-05-20
KR20110091540A (ko) 2011-08-11
US8030500B2 (en) 2011-10-04

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