BRPI0817839A2 - Método para produzir derivado de anel fundido de pirazol - Google Patents
Método para produzir derivado de anel fundido de pirazolInfo
- Publication number
- BRPI0817839A2 BRPI0817839A2 BRPI0817839-9A BRPI0817839A BRPI0817839A2 BR PI0817839 A2 BRPI0817839 A2 BR PI0817839A2 BR PI0817839 A BRPI0817839 A BR PI0817839A BR PI0817839 A2 BRPI0817839 A2 BR PI0817839A2
- Authority
- BR
- Brazil
- Prior art keywords
- pyrazole ring
- ring derivative
- producing fused
- fused pyrazole
- producing
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
- 125000003226 pyrazolyl group Chemical group 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2007271068 | 2007-10-18 | ||
JP2008107868 | 2008-04-17 | ||
PCT/JP2008/068822 WO2009051210A1 (ja) | 2007-10-18 | 2008-10-17 | ピラゾール縮合環誘導体の製造方法 |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0817839A2 true BRPI0817839A2 (pt) | 2015-06-16 |
Family
ID=40567471
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0817839-9A BRPI0817839A2 (pt) | 2007-10-18 | 2008-10-17 | Método para produzir derivado de anel fundido de pirazol |
Country Status (10)
Country | Link |
---|---|
US (1) | US20100217001A1 (pt) |
EP (1) | EP2202233A4 (pt) |
JP (1) | JPWO2009051210A1 (pt) |
CN (1) | CN101827843A (pt) |
BR (1) | BRPI0817839A2 (pt) |
CA (1) | CA2702958A1 (pt) |
IL (1) | IL204822A0 (pt) |
MX (1) | MX2010004135A (pt) |
RU (1) | RU2010119706A (pt) |
WO (1) | WO2009051210A1 (pt) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0313976B8 (pt) * | 2002-10-22 | 2021-05-25 | Eisai Co Ltd | compostos de 7-fenilpirazolopiridina e uso dos mesmos na preparação de agente terapêutico ou profilático para doenças associadas com o crf ou seus receptores |
JP4832743B2 (ja) * | 2004-03-29 | 2011-12-07 | ケンブリッジユニバーシティテクニカルサービスリミテッド | 化合物の合成方法および合成反応触媒 |
US7411082B2 (en) * | 2004-03-29 | 2008-08-12 | Cambridge University Technical Services Ltd. | Synthesizing method for compound, and catalyst for synthesis reaction |
JP4927537B2 (ja) * | 2004-04-12 | 2012-05-09 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピラゾール縮合環誘導体の製造方法 |
-
2008
- 2008-10-17 MX MX2010004135A patent/MX2010004135A/es unknown
- 2008-10-17 WO PCT/JP2008/068822 patent/WO2009051210A1/ja active Application Filing
- 2008-10-17 US US12/738,514 patent/US20100217001A1/en not_active Abandoned
- 2008-10-17 JP JP2009538156A patent/JPWO2009051210A1/ja active Pending
- 2008-10-17 CN CN200880111926A patent/CN101827843A/zh active Pending
- 2008-10-17 CA CA2702958A patent/CA2702958A1/en not_active Abandoned
- 2008-10-17 RU RU2010119706/04A patent/RU2010119706A/ru unknown
- 2008-10-17 BR BRPI0817839-9A patent/BRPI0817839A2/pt not_active IP Right Cessation
- 2008-10-17 EP EP08840583A patent/EP2202233A4/en not_active Withdrawn
-
2010
- 2010-03-28 IL IL204822A patent/IL204822A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP2202233A1 (en) | 2010-06-30 |
IL204822A0 (en) | 2010-11-30 |
JPWO2009051210A1 (ja) | 2011-03-03 |
CN101827843A (zh) | 2010-09-08 |
WO2009051210A1 (ja) | 2009-04-23 |
MX2010004135A (es) | 2010-04-30 |
RU2010119706A (ru) | 2011-11-27 |
EP2202233A4 (en) | 2010-11-10 |
CA2702958A1 (en) | 2009-04-23 |
US20100217001A1 (en) | 2010-08-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 4A, 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |