BRPI0814251A2 - derivados de ácido heterociclil-carboxílicos heterociclicamente substituídos - Google Patents
derivados de ácido heterociclil-carboxílicos heterociclicamente substituídosInfo
- Publication number
- BRPI0814251A2 BRPI0814251A2 BRPI0814251A BRPI0814251A BRPI0814251A2 BR PI0814251 A2 BRPI0814251 A2 BR PI0814251A2 BR PI0814251 A BRPI0814251 A BR PI0814251A BR PI0814251 A BRPI0814251 A BR PI0814251A BR PI0814251 A2 BRPI0814251 A2 BR PI0814251A2
- Authority
- BR
- Brazil
- Prior art keywords
- carboxylic acid
- acid derivatives
- substituted heterocyclyl
- heterocyclically substituted
- heterocyclyl carboxylic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pretreatment Of Seeds And Plants (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07110228A EP2014661A1 (de) | 2007-06-13 | 2007-06-13 | Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate |
PCT/EP2008/004352 WO2008151735A2 (de) | 2007-06-13 | 2008-05-31 | Heterocyclisch substituierte heterocyclyl-carbonsäurederivate |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0814251A2 true BRPI0814251A2 (pt) | 2018-08-14 |
Family
ID=38646606
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0814251A BRPI0814251A2 (pt) | 2007-06-13 | 2008-05-31 | derivados de ácido heterociclil-carboxílicos heterociclicamente substituídos |
Country Status (9)
Country | Link |
---|---|
US (1) | US20100167931A1 (pt) |
EP (2) | EP2014661A1 (pt) |
JP (1) | JP2010532750A (pt) |
CN (1) | CN101679443A (pt) |
AR (1) | AR066945A1 (pt) |
BR (1) | BRPI0814251A2 (pt) |
CL (1) | CL2008001628A1 (pt) |
TW (1) | TW200911122A (pt) |
WO (1) | WO2008151735A2 (pt) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI482771B (zh) * | 2009-05-04 | 2015-05-01 | Du Pont | 磺醯胺殺線蟲劑 |
JP2014517079A (ja) | 2011-06-22 | 2014-07-17 | バーテックス ファーマシューティカルズ インコーポレイテッド | Atrキナーゼ阻害剤として有用な化合物 |
ES2884030T3 (es) | 2012-12-07 | 2021-12-10 | Vertex Pharma | 2-amino-N-(piperidin-1-il-piridin-3-il)pirazolo[1,5alfa]pirimidin-3-carboxamida como inhibidor de ATR quinasa |
EP2970288A1 (en) | 2013-03-15 | 2016-01-20 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
WO2014143241A1 (en) | 2013-03-15 | 2014-09-18 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
JP2016512815A (ja) | 2013-03-15 | 2016-05-09 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | Atrキナーゼの阻害剤として有用な縮合ピラゾロピリミジン誘導体 |
JP6543252B2 (ja) | 2013-12-06 | 2019-07-10 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | ATRキナーゼ阻害剤として有用な2−アミノ−6−フルオロ−N−[5−フルオロ−ピリジン−3−イル]ピラゾロ[1,5−a]ピリミジン−3−カルボキサミド化合物、その調製、その異なる固体形態および放射性標識された誘導体 |
RS60013B1 (sr) | 2014-06-05 | 2020-04-30 | Vertex Pharma | Radioaktivno obeleženi derivati jedinjenja 2-amino-6-fluoro-n-[5-fluoropiridin-3-il]pirazolo[1,5-a]pirimidin-3-karboksamida, korisnog kao inhibitora atr kinaze, dobijanje pomenutog jedinjenja i njegovi različiti čvrsti oblici |
SG10201811175WA (en) | 2014-06-17 | 2019-01-30 | Vertex Pharma | Method for treating cancer using a combination of chk1 and atr inhibitors |
EP3355926A4 (en) | 2015-09-30 | 2019-08-21 | Vertex Pharmaceuticals Inc. | METHOD FOR THE TREATMENT OF CANCER WITH A COMBINATION OF DNA DAMAGING AGENTS AND ATR INHIBITORS |
AR121344A1 (es) * | 2020-02-18 | 2022-05-11 | Pi Industries Ltd | Compuestos heterocíclicos fusionados y su uso como agentes para el control de plagas |
WO2023230217A1 (en) * | 2022-05-25 | 2023-11-30 | Trustees Of Boston University | Antileishmanial compounds, compositions and use thereof |
CN116969954B (zh) * | 2023-09-21 | 2023-11-28 | 广东省农业科学院农业质量标准与监测技术研究所 | 一类含内酰胺的三环稠合杂环化合物及其应用 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20070037828A1 (en) * | 2003-06-27 | 2007-02-15 | Olaf Gebauer | Pyrazolopyrimidines |
DE102004008807A1 (de) * | 2004-02-20 | 2005-09-08 | Bayer Cropscience Ag | Pyrazolopyrimidine |
DE102005007534A1 (de) * | 2005-02-17 | 2006-08-31 | Bayer Cropscience Ag | Pyrazolopyrimidine |
WO2007023020A1 (de) * | 2005-07-13 | 2007-03-01 | Basf Aktiengeseelschaft | 7-amino-6-heteroaryl-1,2,4-triazolo[1,5-a]pyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen |
-
2007
- 2007-06-13 EP EP07110228A patent/EP2014661A1/de not_active Ceased
-
2008
- 2008-05-31 US US12/663,218 patent/US20100167931A1/en not_active Abandoned
- 2008-05-31 EP EP08801444A patent/EP2158204A2/de not_active Withdrawn
- 2008-05-31 WO PCT/EP2008/004352 patent/WO2008151735A2/de active Application Filing
- 2008-05-31 BR BRPI0814251A patent/BRPI0814251A2/pt not_active IP Right Cessation
- 2008-05-31 CN CN200880020002A patent/CN101679443A/zh active Pending
- 2008-05-31 JP JP2010511521A patent/JP2010532750A/ja not_active Withdrawn
- 2008-06-04 CL CL2008001628A patent/CL2008001628A1/es unknown
- 2008-06-10 AR ARP080102467A patent/AR066945A1/es unknown
- 2008-06-12 TW TW097121828A patent/TW200911122A/zh unknown
Also Published As
Publication number | Publication date |
---|---|
EP2014661A1 (de) | 2009-01-14 |
WO2008151735A3 (de) | 2009-07-02 |
TW200911122A (en) | 2009-03-16 |
WO2008151735A2 (de) | 2008-12-18 |
US20100167931A1 (en) | 2010-07-01 |
CN101679443A (zh) | 2010-03-24 |
CL2008001628A1 (es) | 2008-12-19 |
EP2158204A2 (de) | 2010-03-03 |
JP2010532750A (ja) | 2010-10-14 |
AR066945A1 (es) | 2009-09-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: application dismissed [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2485 DE 21-08-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |
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B350 | Update of information on the portal [chapter 15.35 patent gazette] |