BRPI0619551A2 - derivados de jasmonato aprimorados, composições farmacêuticas e métodos de uso dos mesmos - Google Patents
derivados de jasmonato aprimorados, composições farmacêuticas e métodos de uso dos mesmos Download PDFInfo
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- BRPI0619551A2 BRPI0619551A2 BRPI0619551-2A BRPI0619551A BRPI0619551A2 BR PI0619551 A2 BRPI0619551 A2 BR PI0619551A2 BR PI0619551 A BRPI0619551 A BR PI0619551A BR PI0619551 A2 BRPI0619551 A2 BR PI0619551A2
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74287505P | 2005-12-07 | 2005-12-07 | |
| US60/742.875 | 2005-12-07 | ||
| US77258206P | 2006-02-13 | 2006-02-13 | |
| US60/772.582 | 2006-02-13 | ||
| US83066606P | 2006-07-14 | 2006-07-14 | |
| US60/830.666 | 2006-07-14 | ||
| PCT/IL2006/001409 WO2007066337A2 (en) | 2005-12-07 | 2006-12-07 | Jasmonate derivatives, pharmaceutical compositions and methods of use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0619551A2 true BRPI0619551A2 (pt) | 2011-10-04 |
Family
ID=38123294
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0619551-2A BRPI0619551A2 (pt) | 2005-12-07 | 2006-12-07 | derivados de jasmonato aprimorados, composições farmacêuticas e métodos de uso dos mesmos |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8247439B2 (enExample) |
| EP (1) | EP1968959A2 (enExample) |
| JP (1) | JP2009520692A (enExample) |
| AU (1) | AU2006322845A1 (enExample) |
| BR (1) | BRPI0619551A2 (enExample) |
| CA (1) | CA2630666A1 (enExample) |
| WO (1) | WO2007066337A2 (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9284274B2 (en) | 2005-12-07 | 2016-03-15 | Ramot At Tel-Aviv University Ltd. | Chemical derivatives of jasmonate, pharmaceutical compositions and methods of use thereof |
| CN101511351A (zh) * | 2006-07-10 | 2009-08-19 | 雷蒙特亚特特拉维夫大学有限公司 | 治疗癌症的组合方法 |
| JP2010521149A (ja) | 2007-03-15 | 2010-06-24 | ラモット アット テル−アヴィヴ ユニヴァーシティ リミテッド | ミトコンドリア結合ヘキソキナーゼを選択的に阻害する化合物の同定のためのジャスモン酸エステルに基づくアッセイ |
| WO2009120826A1 (en) * | 2008-03-27 | 2009-10-01 | Wyeth | 2-aryl- and 2-heteroarylthiazolyl compounds, methods for their preparation and use thereof |
| US9284252B2 (en) | 2009-06-09 | 2016-03-15 | Sepal Pharma Ltd. | Use of jasmonate ester derivatives for treating benign hyperproliferative skin disorders |
| AU2012221877A1 (en) | 2011-02-25 | 2013-09-19 | Nanocare Technologies, Inc. | Pharmaceutical formulation comprising compounds of the jasmonate family |
| US8883220B2 (en) | 2011-09-16 | 2014-11-11 | Nanocare Technologies, Inc. | Compositions of jasmonate compounds |
| BR112017014229A2 (pt) * | 2014-12-31 | 2018-03-06 | Nanocare Technologies, Inc. | conjugado, composição, e, método para tratamento de um distúrbio. |
| US20200297620A1 (en) | 2016-03-28 | 2020-09-24 | Vidac Pharma Ltd | Stable pharmaceutical compositions for topical administration and uses thereof |
| WO2018083704A1 (en) | 2016-11-07 | 2018-05-11 | Vidac Pharma Ltd. | Use of hexokinase 2/mitochondria-detaching compounds for activating immune responses |
| WO2018083705A1 (en) | 2016-11-07 | 2018-05-11 | Vidac Pharma Ltd. | Use of hexokinase 2/mitochondria-detaching compounds for treating hexokinase-2 (hk2)-expressing cancers |
| WO2019135243A1 (en) * | 2018-01-07 | 2019-07-11 | Vidac Pharma Ltd | Methods for preparation of jasmonate compounds |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS63122669A (ja) * | 1986-10-25 | 1988-05-26 | メルク・パテント・ゲゼルシヤフト・ミツト・ベシユレンクテル・ハフツング | 複素環状液晶化合物 |
| US5476945A (en) * | 1992-11-17 | 1995-12-19 | Fuji Photo Film Co., Ltd. | Water-soluble methine derivatives of thiazole |
| JPH07308196A (ja) * | 1994-05-18 | 1995-11-28 | Mitsui Petrochem Ind Ltd | タキサン型ジテルペンの製造方法 |
| EP1348764A1 (en) * | 1993-11-15 | 2003-10-01 | Mitsui Chemicals, Inc. | A Method of Producing a Taxane-Type Diterpene and Method of Obtaining Cultured Cells which Produce the Taxane-Type Diterpene at a High Rate |
| AU2002254342A1 (en) * | 2001-03-23 | 2002-10-08 | The Board Of Trustees Of The University Of Illinois | Compounds capable of modulating the activity of multidrug transporters and therapeutic use of the same |
| US6469061B1 (en) * | 2001-04-04 | 2002-10-22 | Ramot University Authority For Applied Research And Industrial Development Limited | Jasmonate pharmaceutical composition for treatment of cancer |
| FR2825926A1 (fr) * | 2001-06-14 | 2002-12-20 | Sod Conseils Rech Applic | Derives d'imidazoles modulant les canaux sodiques |
| AU2003296405A1 (en) * | 2003-01-06 | 2004-08-10 | Eli Lilly And Company | Fused heterocyclic derivatives as ppar modulators |
| WO2005054172A2 (en) | 2003-12-02 | 2005-06-16 | Ramot At Tel-Aviv University Ltd. | Jasmonate derivative compounds, pharmaceuticals compositions and methods of use thereof |
-
2006
- 2006-12-07 EP EP06821627A patent/EP1968959A2/en not_active Withdrawn
- 2006-12-07 AU AU2006322845A patent/AU2006322845A1/en not_active Abandoned
- 2006-12-07 BR BRPI0619551-2A patent/BRPI0619551A2/pt not_active IP Right Cessation
- 2006-12-07 CA CA002630666A patent/CA2630666A1/en not_active Abandoned
- 2006-12-07 WO PCT/IL2006/001409 patent/WO2007066337A2/en not_active Ceased
- 2006-12-07 JP JP2008544003A patent/JP2009520692A/ja active Pending
- 2006-12-07 US US12/096,111 patent/US8247439B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2009520692A (ja) | 2009-05-28 |
| EP1968959A2 (en) | 2008-09-17 |
| US8247439B2 (en) | 2012-08-21 |
| AU2006322845A1 (en) | 2007-06-14 |
| WO2007066337A2 (en) | 2007-06-14 |
| US20090197927A1 (en) | 2009-08-06 |
| CA2630666A1 (en) | 2007-06-14 |
| WO2007066337A3 (en) | 2007-11-15 |
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| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A ANUIDADE. |
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| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012. |