BRPI0611747A2 - composto ou um sal farmaceuticamente aceitÁvel do mesmo ou n-àxidos do mesmo, composiÇço farmacÊutica, mÉtodos para tratar uma infecÇço bacteriana e para inibir o dna girase bacteriana em um animal de sangue quente, uso de um composto ou um sal farmaceuticamente aceitÁvel do mesmo, e, processo para fabricar um composto ou um sal farmaceuticamente aceitÁvel do mesmo - Google Patents

composto ou um sal farmaceuticamente aceitÁvel do mesmo ou n-àxidos do mesmo, composiÇço farmacÊutica, mÉtodos para tratar uma infecÇço bacteriana e para inibir o dna girase bacteriana em um animal de sangue quente, uso de um composto ou um sal farmaceuticamente aceitÁvel do mesmo, e, processo para fabricar um composto ou um sal farmaceuticamente aceitÁvel do mesmo

Info

Publication number
BRPI0611747A2
BRPI0611747A2 BRPI0611747-3A BRPI0611747A BRPI0611747A2 BR PI0611747 A2 BRPI0611747 A2 BR PI0611747A2 BR PI0611747 A BRPI0611747 A BR PI0611747A BR PI0611747 A2 BRPI0611747 A2 BR PI0611747A2
Authority
BR
Brazil
Prior art keywords
pharmaceutically acceptable
compound
acceptable salt
warm
treating
Prior art date
Application number
BRPI0611747-3A
Other languages
English (en)
Inventor
Gloria Breault
Charles Joseph Eyermann
Bolin Geng
Marshall Morningstar
Folkert Reck
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36956054&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0611747(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0611747A2 publication Critical patent/BRPI0611747A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

COMPOSTO OU UM SAL FARMACEUTICAMENTE ACEITÁVEL DO MESMO OU N-àXIDOS DO MESMO, COMPOSIÇçO FARMACÊUTICA, MÉTODOS PARA TRATAR UMA INFECÇçO BACTERIANA E PARA INIBIR O DNA GIRASE BACTERIANA EM UM ANIMAL DE SANGUE QUENTE, USO DE UM COMPOSTO OU UM SAL FARMACEUTICAMENTE ACEITÁVEL DO MESMO, E, PROCESSO PARA FABRICAR UM COMPOSTO OU UM SAL FARMACEUTICAMENTE ACEITÁVEL DO MESMO. A presente invenção diz respeito aos compostos que demonstram atividade anti-bacteriana, aos processos para prepará-los, às composições farmacêuticas que os contenham como ingrediente ativo, ao uso destes como medicamentos e ao uso destes na fabricação de medicamentos para o uso no tratamento de infecções bacterianas em animais de sangue quente tal como os seres humanos. Em particular esta invenção diz respeito aos compostos úteis para o tratamento de infecções bacterianas em animais de sangue quente tais como seres humanos, mais particularmente ao uso destes compostos na fabricação de medicamentos para o uso no tratamento de infecções bacterianas em animais de sangue quente tal como seres humanos.
BRPI0611747-3A 2005-06-16 2006-06-16 composto ou um sal farmaceuticamente aceitÁvel do mesmo ou n-àxidos do mesmo, composiÇço farmacÊutica, mÉtodos para tratar uma infecÇço bacteriana e para inibir o dna girase bacteriana em um animal de sangue quente, uso de um composto ou um sal farmaceuticamente aceitÁvel do mesmo, e, processo para fabricar um composto ou um sal farmaceuticamente aceitÁvel do mesmo BRPI0611747A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69134005P 2005-06-16 2005-06-16
PCT/GB2006/002207 WO2006134378A1 (en) 2005-06-16 2006-06-16 Compounds for the treatment of multi-drug resistant bacterial infections

Publications (1)

Publication Number Publication Date
BRPI0611747A2 true BRPI0611747A2 (pt) 2008-12-02

Family

ID=36956054

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0611747-3A BRPI0611747A2 (pt) 2005-06-16 2006-06-16 composto ou um sal farmaceuticamente aceitÁvel do mesmo ou n-àxidos do mesmo, composiÇço farmacÊutica, mÉtodos para tratar uma infecÇço bacteriana e para inibir o dna girase bacteriana em um animal de sangue quente, uso de um composto ou um sal farmaceuticamente aceitÁvel do mesmo, e, processo para fabricar um composto ou um sal farmaceuticamente aceitÁvel do mesmo

Country Status (20)

Country Link
US (3) US7875715B2 (pt)
EP (2) EP1893599A1 (pt)
JP (1) JP5204649B2 (pt)
KR (2) KR101351160B1 (pt)
CN (1) CN101243068B (pt)
AR (1) AR054781A1 (pt)
AU (1) AU2006258879C1 (pt)
BR (1) BRPI0611747A2 (pt)
CA (1) CA2610900A1 (pt)
EC (1) ECSP088102A (pt)
IL (1) IL187581A0 (pt)
MX (1) MX2007015297A (pt)
MY (1) MY150958A (pt)
NO (1) NO20080338L (pt)
NZ (1) NZ565110A (pt)
RU (1) RU2008100306A (pt)
TW (1) TW200716623A (pt)
UY (1) UY29608A1 (pt)
WO (1) WO2006134378A1 (pt)
ZA (1) ZA200710563B (pt)

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NO20080338L (no) 2008-02-29
US20100152441A1 (en) 2010-06-17
AU2006258879B2 (en) 2009-11-19
CN101243068A (zh) 2008-08-13
RU2008100306A (ru) 2009-07-27
ECSP088102A (es) 2008-02-20
JP5204649B2 (ja) 2013-06-05
ZA200710563B (en) 2008-12-31
EP1893599A1 (en) 2008-03-05
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MY150958A (en) 2014-03-31
AU2006258879A1 (en) 2006-12-21
AR054781A1 (es) 2007-07-18
EP2289890A1 (en) 2011-03-02
US8124602B2 (en) 2012-02-28
JP2008543819A (ja) 2008-12-04
MX2007015297A (es) 2008-02-21
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NZ565110A (en) 2011-05-27
IL187581A0 (en) 2008-03-20
WO2006134378A1 (en) 2006-12-21
KR20130108468A (ko) 2013-10-02
US20120108577A1 (en) 2012-05-03
CA2610900A1 (en) 2006-12-21
UY29608A1 (es) 2007-01-31
TW200716623A (en) 2007-05-01

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