BR9908960A - Amino guanidinas cìclicas - Google Patents

Amino guanidinas cìclicas

Info

Publication number
BR9908960A
BR9908960A BR9908960-2A BR9908960A BR9908960A BR 9908960 A BR9908960 A BR 9908960A BR 9908960 A BR9908960 A BR 9908960A BR 9908960 A BR9908960 A BR 9908960A
Authority
BR
Brazil
Prior art keywords
cyclic guanidine
cyclic
amino
guanidine amino
substituents
Prior art date
Application number
BR9908960-2A
Other languages
English (en)
Inventor
Gerd Ascher
Werner Heilamayer
Johannes Ludescher
Johannes Hilderbrandt
Michael Schranz
Josef Wieser
Original Assignee
Biochemie Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biochemie Gmbh filed Critical Biochemie Gmbh
Publication of BR9908960A publication Critical patent/BR9908960A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Patente de Invenção: <B>"AMINO GUANIDINAS CìCLICAS"<D>. Composto de fórmula onde R~ 2~ juntamente com o átomo de nitrogênio ao qual ele está ligado forma um grupo aminoguanidino cíclico ou derivado do mesmo, sendo que os outros substituintes possuem vários significados, útil como produto farmacêutico.
BR9908960-2A 1998-03-23 1999-03-19 Amino guanidinas cìclicas BR9908960A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT0051598A AT406772B (de) 1998-03-23 1998-03-23 Antibakterielle 7-acylamino-3-iminomethyl- cephalosporine und verfahren zu deren herstellung
PCT/EP1999/001853 WO1999048896A1 (en) 1998-03-23 1999-03-19 Cephalosporines having cyclic aminoguanidine substituents as antibiotics

Publications (1)

Publication Number Publication Date
BR9908960A true BR9908960A (pt) 2000-12-05

Family

ID=3492649

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9908960-2A BR9908960A (pt) 1998-03-23 1999-03-19 Amino guanidinas cìclicas

Country Status (25)

Country Link
US (1) US6440957B1 (pt)
EP (2) EP1930335A1 (pt)
JP (1) JP2002507616A (pt)
KR (1) KR100696422B1 (pt)
CN (1) CN1188418C (pt)
AR (1) AR015248A1 (pt)
AT (1) AT406772B (pt)
AU (1) AU749735B2 (pt)
BR (1) BR9908960A (pt)
CA (1) CA2324953C (pt)
CO (1) CO5080739A1 (pt)
HU (1) HUP0101603A3 (pt)
ID (1) ID26567A (pt)
IL (2) IL138477A0 (pt)
MY (1) MY119841A (pt)
NO (1) NO20004760L (pt)
NZ (1) NZ506908A (pt)
PE (1) PE20000360A1 (pt)
PL (1) PL343094A1 (pt)
RU (1) RU2245884C2 (pt)
SK (1) SK14152000A3 (pt)
TR (1) TR200002749T2 (pt)
TW (1) TWI250983B (pt)
WO (1) WO1999048896A1 (pt)
ZA (1) ZA200004850B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020115852A1 (en) * 1997-04-01 2002-08-22 Gerd Ascher Antibacterial substituted 7-acylamino-3-(methylhydrazono) methyl-cephalosporins and intermediates
DE102007052891A1 (de) 2007-11-02 2009-05-07 Evonik Degussa Gmbh Verfahren zur Stabilisierung von olefinisch ungesättigten Monomeren
DE102013204950A1 (de) 2013-03-20 2014-09-25 Evonik Industries Ag Verfahren und Zusammensetzung zur Inhibierung der Polymerisation von Cyclopentadienverbindungen
EP2993164B1 (de) 2014-09-08 2017-02-15 Evonik Degussa GmbH Phenolische (Thio)Acetale als Inhibitoren der Polymerisation von olefinisch ungesättigten Monomeren
TWI669317B (zh) 2014-09-22 2019-08-21 德商贏創德固賽有限責任公司 反應性單體的改良製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE943408C (de) * 1953-03-31 1956-05-17 Bayer Ag Verfahren zur Darstellung von Bisguanylhydrazonen
FI851934L (fi) * 1984-05-30 1985-12-01 Ici Plc Kefalosporinderivat.
CA2219656C (en) * 1995-05-11 2008-08-19 Gerd Ascher Antibacterial cephalosporins
PL200130B1 (pl) * 1997-04-01 2008-12-31 Nabriva Therapeutics Forschung Podstawione pochodne 7-acyloamino-3-(metylohydrazono)metylocefalosporyny, sposób ich wytwarzania, kompozycja farmaceutyczna zawierająca takie pochodne, zastosowania tych pochodnych oraz związki pośrednie służące do otrzymywania podstawionych 7-acyloamino-3-(metylohydrazono)metylocefalosporyn

Also Published As

Publication number Publication date
TWI250983B (en) 2006-03-11
RU2245884C2 (ru) 2005-02-10
EP1082326A1 (en) 2001-03-14
CN1188418C (zh) 2005-02-09
KR100696422B1 (ko) 2007-03-20
PL343094A1 (en) 2001-07-30
ZA200004850B (en) 2002-02-27
CO5080739A1 (es) 2001-09-25
IL138477A0 (en) 2001-10-31
NZ506908A (en) 2003-04-29
US6440957B1 (en) 2002-08-27
NO20004760L (no) 2000-11-21
EP1930335A1 (en) 2008-06-11
AU749735B2 (en) 2002-07-04
MY119841A (en) 2005-07-29
IL138477A (en) 2007-06-17
AR015248A1 (es) 2001-04-18
PE20000360A1 (es) 2000-05-17
JP2002507616A (ja) 2002-03-12
AT406772B (de) 2000-08-25
SK14152000A3 (sk) 2001-05-10
TR200002749T2 (tr) 2000-12-21
KR20010074666A (ko) 2001-08-08
CN1294593A (zh) 2001-05-09
CA2324953A1 (en) 1999-09-30
ATA51598A (de) 2000-01-15
NO20004760D0 (no) 2000-09-22
AU3518899A (en) 1999-10-18
HUP0101603A2 (hu) 2001-12-28
CA2324953C (en) 2008-05-13
WO1999048896A1 (en) 1999-09-30
HUP0101603A3 (en) 2002-10-28
ID26567A (id) 2001-01-18

Similar Documents

Publication Publication Date Title
CY1120169T1 (el) Παραγωγο αμιδιου και φαρμακο
BR0012880A (pt) Derivados de mutilina e seu uso como antibacterianos
HUP9802859A2 (hu) Acil-amino-szalicilsav-amid-származékok és alkalmazásuk peszticidként
DK1265606T3 (da) Celleadhæsionsinhibitorer
BR9907429A (pt) Composto de hidrazida, processo para sua preparação e composições farmacêuticas contendo os mesmos
BR9900443A (pt) Esteres de ácido aril acrìlico.
BR0009641A (pt) Derivados de 1,4-benzotiazepin-1,1-dióxido, substituìdos com radicais de açúcar, processo para produção dos mesmos, medicamentos contendo esses compostos e sua utilização
PT1063228E (pt) Derivados de cicloalcenos processo para a sua preparacao e utilizacao
CY1109882T1 (el) Νεα αλατα ατορβαστατινης και φαρμακευτικες συνθεσεις που τα περιεχουν
BR9916328A (pt) Inibidores de transferase de farnesila
ATE316531T1 (de) Kondensierte dihydrochinolinon-derivate zur hemmung von mrp1
WO2005002508A3 (en) Macromolecular platinum chelates
BR0007890A (pt) Compostos de uracila e uso dos mesmos
HUP0201475A2 (hu) Heteroarilamidin-, metilamidin- és guanidinszármazékok, előállításuk és alkalmazásuk, valamint e vegyületeket tartalmazó gyógyászati készítmények
DE69208408T2 (de) Phenylthioharnstoffderivate und ihre pharmazeutische Verwendung
BR0213990A (pt) Derivados de piperazina tendo atividade antagonìstica de sst1
BR9908960A (pt) Amino guanidinas cìclicas
AR044175A1 (es) Compuestos de cefemo
BR0309130A (pt) Derivados de acil-3-carboxifenil-uréia, processo para a sua preparação e sua aplicação
DE69915514D1 (de) Prenyltransferase-inhibitoren
DE602004025935D1 (de) Histondeacetylaseinhibitor und verfahren zu dessen herstellung
ATE325116T1 (de) Farnesyltransferasehemmende 4- heterocyclylchinolin- und chinazolinderivate
NO20060884L (no) Adhesiv samensetning omfattende et formaldehydinneholdende aminoplastresin og en katalyserende forbindelse
BRPI0406840A (pt) Derivados de acil-fenil-uréia substituìdos por carbonilamino, processos para a sua preparação e sua aplicação
ATE434615T1 (de) Farnesyltransferase hemmende benzoheterocyclische derivate

Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: C07D 501/46, A61K 31/545, A61P 31/04

Ipc: C07D 501/46 (2009.01), A61K 31/545 (2009.01)

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO DE ACORDO COM OS ARTIGOS 8O, 10 (VIII), 11, 13, 24 E 25 DA LPI.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.