BR9809702A - Derivado de ciclobutilamina substituìdo - Google Patents
Derivado de ciclobutilamina substituìdoInfo
- Publication number
- BR9809702A BR9809702A BR9809702-4A BR9809702A BR9809702A BR 9809702 A BR9809702 A BR 9809702A BR 9809702 A BR9809702 A BR 9809702A BR 9809702 A BR9809702 A BR 9809702A
- Authority
- BR
- Brazil
- Prior art keywords
- derivative
- cyclobutylamine
- resistant
- derivatives
- bacteria
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
"DERIVADO DE CICLOBUTILAMINA SUBSTITUìDO". Derivadosde ciclobutilamina substituídos com novas estruturasrepresentadas pela fórmula geral (I), na qual cada um de R^ 1^ aR^ 4^ e Q representa um substituinte especifico e, em particular, Qrepresenta um derivado de quinolina de uma estrutura específica.Esses derivados são úteis como compostos antibacterianos, quetêm excelentes ações antibacterianas por um grande âmbito debactérias, incluindo aquelas gram-negativas e gram-positivas,exercem potentes atividade antibacterianas, particularmente, emStaphylococcus aureus resistente à meticilina (MRSA),Streptococcus pneumoniae resistente à penicilina e bactériasresistentes à quinolona e são excelentes em dinâmica e segurançain vivo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP14139897 | 1997-05-30 | ||
PCT/JP1998/002359 WO1998054169A1 (fr) | 1997-05-30 | 1998-05-28 | Derives substitues de la cyclobutylamine |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9809702A true BR9809702A (pt) | 2001-12-11 |
Family
ID=15291079
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9809702-4A BR9809702A (pt) | 1997-05-30 | 1998-05-28 | Derivado de ciclobutilamina substituìdo |
Country Status (20)
Country | Link |
---|---|
US (1) | US6448266B1 (pt) |
EP (1) | EP0990654B1 (pt) |
JP (1) | JP4357598B2 (pt) |
KR (1) | KR100551462B1 (pt) |
CN (1) | CN1191245C (pt) |
AR (1) | AR012883A1 (pt) |
AT (1) | ATE378327T1 (pt) |
AU (1) | AU732175B2 (pt) |
BR (1) | BR9809702A (pt) |
CA (1) | CA2292580A1 (pt) |
DE (1) | DE69838716T2 (pt) |
DK (1) | DK0990654T3 (pt) |
ES (1) | ES2297885T3 (pt) |
ID (1) | ID23696A (pt) |
IL (1) | IL133123A (pt) |
MY (1) | MY119816A (pt) |
NO (1) | NO318143B1 (pt) |
RU (1) | RU2205829C2 (pt) |
WO (1) | WO1998054169A1 (pt) |
ZA (1) | ZA984527B (pt) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1015445B1 (en) | 1997-09-15 | 2009-02-25 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
KR100768034B1 (ko) | 1999-03-17 | 2007-10-17 | 다이이찌 세이야꾸 가부시기가이샤 | 의약 조성물 |
KR100777149B1 (ko) | 2000-11-20 | 2007-11-19 | 다이이찌 세이야꾸 가부시기가이샤 | 데할로게노 화합물 |
AU3089102A (en) | 2000-12-14 | 2002-06-24 | Procter & Gamble | Antimicrobial quinolones |
IL155678A0 (en) | 2000-12-14 | 2003-11-23 | Procter & Gamble | Antimicrobial 2-pyridones, their compositions and uses |
EP1669354B1 (en) * | 2003-09-29 | 2013-03-20 | Daiichi Sankyo Company, Limited | 8-cyanoquinolonecarboxylic acid derivative |
US7456279B2 (en) | 2006-03-28 | 2008-11-25 | The Procter & Gamble Company | Coupling process for preparing quinolone intermediates |
SMP200800058B (it) | 2006-03-28 | 2009-09-07 | Procter & Gamble | Sali e polimorfi malati di un acido (3s, 5s) -7- [3-ammino-5-metilpiperidinil]-1-ciclopropil-1,4-diidro-8-metossi-4-osso-3-chinolincarbossilico |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL79189A (en) * | 1985-06-26 | 1990-07-12 | Daiichi Seiyaku Co | Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them |
JPH0827728A (ja) * | 1990-02-13 | 1996-01-30 | Sf Marina System Ab | ポンツーンの昇降案内装置 |
JP3745433B2 (ja) * | 1995-02-02 | 2006-02-15 | 第一製薬株式会社 | 複素環式化合物 |
EP1304329B1 (en) * | 1995-02-02 | 2008-10-15 | Daiichi Sankyo Company, Limited | Pyridonecarboxylic acid derivatives and their use as antibacterial agents |
ES2258780T3 (es) * | 1995-11-22 | 2006-09-01 | Daiichi Pharmaceutical Co., Ltd. | Derivados de aminocicloalquilpirrolidina sustituidos. |
-
1998
- 1998-05-27 MY MYPI98002358A patent/MY119816A/en unknown
- 1998-05-27 ZA ZA984527A patent/ZA984527B/xx unknown
- 1998-05-28 ID IDW991489A patent/ID23696A/id unknown
- 1998-05-28 JP JP50048599A patent/JP4357598B2/ja not_active Expired - Fee Related
- 1998-05-28 DK DK98921863T patent/DK0990654T3/da active
- 1998-05-28 WO PCT/JP1998/002359 patent/WO1998054169A1/ja active IP Right Grant
- 1998-05-28 AT AT98921863T patent/ATE378327T1/de not_active IP Right Cessation
- 1998-05-28 ES ES98921863T patent/ES2297885T3/es not_active Expired - Lifetime
- 1998-05-28 CA CA002292580A patent/CA2292580A1/en not_active Abandoned
- 1998-05-28 RU RU99125325/04A patent/RU2205829C2/ru not_active IP Right Cessation
- 1998-05-28 AU AU74539/98A patent/AU732175B2/en not_active Ceased
- 1998-05-28 IL IL13312398A patent/IL133123A/en not_active IP Right Cessation
- 1998-05-28 DE DE69838716T patent/DE69838716T2/de not_active Expired - Fee Related
- 1998-05-28 EP EP98921863A patent/EP0990654B1/en not_active Expired - Lifetime
- 1998-05-28 US US09/424,780 patent/US6448266B1/en not_active Expired - Fee Related
- 1998-05-28 CN CNB988078066A patent/CN1191245C/zh not_active Expired - Fee Related
- 1998-05-28 BR BR9809702-4A patent/BR9809702A/pt not_active Application Discontinuation
- 1998-05-28 KR KR1019997011191A patent/KR100551462B1/ko not_active IP Right Cessation
- 1998-05-29 AR ARP980102496A patent/AR012883A1/es active IP Right Grant
-
1999
- 1999-11-29 NO NO19995839A patent/NO318143B1/no unknown
Also Published As
Publication number | Publication date |
---|---|
WO1998054169A1 (fr) | 1998-12-03 |
ID23696A (id) | 2000-05-11 |
CA2292580A1 (en) | 1998-12-03 |
DK0990654T3 (da) | 2008-01-21 |
AR012883A1 (es) | 2000-11-22 |
CN1191245C (zh) | 2005-03-02 |
US6448266B1 (en) | 2002-09-10 |
EP0990654A1 (en) | 2000-04-05 |
KR100551462B1 (ko) | 2006-02-14 |
CN1265659A (zh) | 2000-09-06 |
IL133123A0 (en) | 2001-03-19 |
DE69838716D1 (de) | 2007-12-27 |
IL133123A (en) | 2005-12-18 |
EP0990654B1 (en) | 2007-11-14 |
NO995839L (no) | 2000-01-28 |
ZA984527B (en) | 1998-12-03 |
ATE378327T1 (de) | 2007-11-15 |
MY119816A (en) | 2005-07-29 |
KR20010013204A (ko) | 2001-02-26 |
JP4357598B2 (ja) | 2009-11-04 |
EP0990654A4 (en) | 2004-09-15 |
NO318143B1 (no) | 2005-02-07 |
NO995839D0 (no) | 1999-11-29 |
ES2297885T3 (es) | 2008-05-01 |
AU732175B2 (en) | 2001-04-12 |
AU7453998A (en) | 1998-12-30 |
RU2205829C2 (ru) | 2003-06-10 |
DE69838716T2 (de) | 2008-10-30 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
WO2005070945A8 (ja) | メチシリン耐性黄色ブドウ球菌(mrsa)に有効な新規アミノグリコシド系抗生物質 | |
TR199901127T2 (xx) | Antibakteriyel etkili 6-O-ikameli ketolitler. | |
ATE480538T1 (de) | 2-arylmethylazetidincarbapenemderivate und deren herstellung | |
PT718293E (pt) | Composto ciclodepsipeptidico | |
NZ545472A (en) | 7-(4-substituted-3-cyclopropylaminomethyl-1-pyrrolidinyl)quinolonecarboxylic acid derivative | |
BR9809702A (pt) | Derivado de ciclobutilamina substituìdo | |
DE602004004808D1 (de) | Acyloxymethylcarbamat-prodrugs von oxazolidinonen | |
WO2005070922A3 (en) | Bis-indole pyrroles useful as antimicrobials agents | |
DK1096952T3 (da) | Polysaccharidvaccine mod stafylokok-infektioner | |
MXPA03004437A (es) | Compuestos de deshalogeno. | |
WO2004016632A8 (en) | Lincomycin derivatives possessing antibacterial activity | |
CA2189995A1 (en) | Novel carbapenem derivatives | |
WO2005007665A8 (en) | Lincomycin derivatives possessing antibacterial activity | |
DK206888D0 (da) | Thiadiazolylacetamidcephemderivat | |
EP0947517A4 (en) | CEPHEM DERIVATIVES | |
WO2004004646A3 (en) | O-derivatized nocathiacin derivatives | |
DE60115851D1 (de) | Anti-infektionsmittel, die gegen gegenüber mehreren arzneimitteln resistente bakterienstämme nützlich sind | |
WO2002057286A3 (en) | 9-amino erythromycin derivatives with antibacterial activity | |
BR0312246A (pt) | derivados oxazolidinona glicoloil substituìdo como agentes antibacterianos | |
ES2195411T3 (es) | Compuestos antibacterianos de carbapenem, composiciones que contienen tales compuestos y procedimientos de tratamiento. | |
RU94028649A (ru) | Оксимные производные с цефалоспорановой структурой, способ их получения и промежуточные соединения | |
BRPI0411537A (pt) | derivados de lincomicina que possuem atividade antibacteriana | |
GR1003521B (el) | Μεθοδοι χρησεως ενωσεων φλουοροκινολονης εναντια κατα gram θετικων παθογονων βακτηριδιων | |
WO2003068791A3 (en) | Macrolides with activity against methicillin-resistant staphylococcus aureus | |
AR022098A1 (es) | Uso de compuestos de quinolona para la manufactura de un medicamento contra bacterias patogenas gram positivas |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B15K | Others concerning applications: alteration of classification |
Free format text: ALTERADA DE INT.CL: C07D 401/04, C07D 498/06, A61K 31/4709, A61P 31/04 Ipc: C07D 401/04 (2008.01), C07D 498/06 (2008.01) |
|
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFERIMENTO DE ACORDO COM ART. 8O DA LPI. |