BR9809702A - Derivado de ciclobutilamina substituìdo - Google Patents

Derivado de ciclobutilamina substituìdo

Info

Publication number
BR9809702A
BR9809702A BR9809702-4A BR9809702A BR9809702A BR 9809702 A BR9809702 A BR 9809702A BR 9809702 A BR9809702 A BR 9809702A BR 9809702 A BR9809702 A BR 9809702A
Authority
BR
Brazil
Prior art keywords
derivative
cyclobutylamine
resistant
derivatives
bacteria
Prior art date
Application number
BR9809702-4A
Other languages
English (en)
Inventor
Makota Takemura
Hisashi Takahashi
Kazuyuki Sugita
Rie Miyauchi
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of BR9809702A publication Critical patent/BR9809702A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"DERIVADO DE CICLOBUTILAMINA SUBSTITUìDO". Derivadosde ciclobutilamina substituídos com novas estruturasrepresentadas pela fórmula geral (I), na qual cada um de R^ 1^ aR^ 4^ e Q representa um substituinte especifico e, em particular, Qrepresenta um derivado de quinolina de uma estrutura específica.Esses derivados são úteis como compostos antibacterianos, quetêm excelentes ações antibacterianas por um grande âmbito debactérias, incluindo aquelas gram-negativas e gram-positivas,exercem potentes atividade antibacterianas, particularmente, emStaphylococcus aureus resistente à meticilina (MRSA),Streptococcus pneumoniae resistente à penicilina e bactériasresistentes à quinolona e são excelentes em dinâmica e segurançain vivo.
BR9809702-4A 1997-05-30 1998-05-28 Derivado de ciclobutilamina substituìdo BR9809702A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP14139897 1997-05-30
PCT/JP1998/002359 WO1998054169A1 (fr) 1997-05-30 1998-05-28 Derives substitues de la cyclobutylamine

Publications (1)

Publication Number Publication Date
BR9809702A true BR9809702A (pt) 2001-12-11

Family

ID=15291079

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9809702-4A BR9809702A (pt) 1997-05-30 1998-05-28 Derivado de ciclobutilamina substituìdo

Country Status (20)

Country Link
US (1) US6448266B1 (pt)
EP (1) EP0990654B1 (pt)
JP (1) JP4357598B2 (pt)
KR (1) KR100551462B1 (pt)
CN (1) CN1191245C (pt)
AR (1) AR012883A1 (pt)
AT (1) ATE378327T1 (pt)
AU (1) AU732175B2 (pt)
BR (1) BR9809702A (pt)
CA (1) CA2292580A1 (pt)
DE (1) DE69838716T2 (pt)
DK (1) DK0990654T3 (pt)
ES (1) ES2297885T3 (pt)
ID (1) ID23696A (pt)
IL (1) IL133123A (pt)
MY (1) MY119816A (pt)
NO (1) NO318143B1 (pt)
RU (1) RU2205829C2 (pt)
WO (1) WO1998054169A1 (pt)
ZA (1) ZA984527B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1015445B1 (en) 1997-09-15 2009-02-25 The Procter & Gamble Company Antimicrobial quinolones, their compositions and uses
KR100768034B1 (ko) 1999-03-17 2007-10-17 다이이찌 세이야꾸 가부시기가이샤 의약 조성물
KR100777149B1 (ko) 2000-11-20 2007-11-19 다이이찌 세이야꾸 가부시기가이샤 데할로게노 화합물
AU3089102A (en) 2000-12-14 2002-06-24 Procter & Gamble Antimicrobial quinolones
IL155678A0 (en) 2000-12-14 2003-11-23 Procter & Gamble Antimicrobial 2-pyridones, their compositions and uses
EP1669354B1 (en) * 2003-09-29 2013-03-20 Daiichi Sankyo Company, Limited 8-cyanoquinolonecarboxylic acid derivative
US7456279B2 (en) 2006-03-28 2008-11-25 The Procter & Gamble Company Coupling process for preparing quinolone intermediates
SMP200800058B (it) 2006-03-28 2009-09-07 Procter & Gamble Sali e polimorfi malati di un acido (3s, 5s) -7- [3-ammino-5-metilpiperidinil]-1-ciclopropil-1,4-diidro-8-metossi-4-osso-3-chinolincarbossilico

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL79189A (en) * 1985-06-26 1990-07-12 Daiichi Seiyaku Co Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them
JPH0827728A (ja) * 1990-02-13 1996-01-30 Sf Marina System Ab ポンツーンの昇降案内装置
JP3745433B2 (ja) * 1995-02-02 2006-02-15 第一製薬株式会社 複素環式化合物
EP1304329B1 (en) * 1995-02-02 2008-10-15 Daiichi Sankyo Company, Limited Pyridonecarboxylic acid derivatives and their use as antibacterial agents
ES2258780T3 (es) * 1995-11-22 2006-09-01 Daiichi Pharmaceutical Co., Ltd. Derivados de aminocicloalquilpirrolidina sustituidos.

Also Published As

Publication number Publication date
WO1998054169A1 (fr) 1998-12-03
ID23696A (id) 2000-05-11
CA2292580A1 (en) 1998-12-03
DK0990654T3 (da) 2008-01-21
AR012883A1 (es) 2000-11-22
CN1191245C (zh) 2005-03-02
US6448266B1 (en) 2002-09-10
EP0990654A1 (en) 2000-04-05
KR100551462B1 (ko) 2006-02-14
CN1265659A (zh) 2000-09-06
IL133123A0 (en) 2001-03-19
DE69838716D1 (de) 2007-12-27
IL133123A (en) 2005-12-18
EP0990654B1 (en) 2007-11-14
NO995839L (no) 2000-01-28
ZA984527B (en) 1998-12-03
ATE378327T1 (de) 2007-11-15
MY119816A (en) 2005-07-29
KR20010013204A (ko) 2001-02-26
JP4357598B2 (ja) 2009-11-04
EP0990654A4 (en) 2004-09-15
NO318143B1 (no) 2005-02-07
NO995839D0 (no) 1999-11-29
ES2297885T3 (es) 2008-05-01
AU732175B2 (en) 2001-04-12
AU7453998A (en) 1998-12-30
RU2205829C2 (ru) 2003-06-10
DE69838716T2 (de) 2008-10-30

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DE INT.CL: C07D 401/04, C07D 498/06, A61K 31/4709, A61P 31/04

Ipc: C07D 401/04 (2008.01), C07D 498/06 (2008.01)

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFERIMENTO DE ACORDO COM ART. 8O DA LPI.