BR9610388A - Composto de pirimidina ou um seu sal de adição de ácido processo para a preparação de uma pirimidina e formulação farmacêutica - Google Patents

Composto de pirimidina ou um seu sal de adição de ácido processo para a preparação de uma pirimidina e formulação farmacêutica

Info

Publication number
BR9610388A
BR9610388A BR9610388A BR9610388A BR9610388A BR 9610388 A BR9610388 A BR 9610388A BR 9610388 A BR9610388 A BR 9610388A BR 9610388 A BR9610388 A BR 9610388A BR 9610388 A BR9610388 A BR 9610388A
Authority
BR
Brazil
Prior art keywords
pyrimidine
preparation
acid addition
pharmaceutical formulation
addition salt
Prior art date
Application number
BR9610388A
Other languages
English (en)
Inventor
Malcom Stuart Noble
Sandra Jane Rodgers
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of BR9610388A publication Critical patent/BR9610388A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BR9610388A 1995-09-05 1996-09-03 Composto de pirimidina ou um seu sal de adição de ácido processo para a preparação de uma pirimidina e formulação farmacêutica BR9610388A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9518027.9A GB9518027D0 (en) 1995-09-05 1995-09-05 Pharmacologically active compound
PCT/EP1996/003856 WO1997009317A2 (en) 1995-09-05 1996-09-03 Optically active phenyl pyrimidine derivative as analgesic agent

Publications (1)

Publication Number Publication Date
BR9610388A true BR9610388A (pt) 1999-07-06

Family

ID=10780172

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9610388A BR9610388A (pt) 1995-09-05 1996-09-03 Composto de pirimidina ou um seu sal de adição de ácido processo para a preparação de uma pirimidina e formulação farmacêutica

Country Status (32)

Country Link
US (1) US6124308A (pt)
EP (1) EP0879230B1 (pt)
JP (1) JPH11512108A (pt)
KR (1) KR19990044397A (pt)
CN (1) CN1200729A (pt)
AP (1) AP640A (pt)
AR (1) AR004192A1 (pt)
AT (1) ATE203523T1 (pt)
AU (1) AU710091B2 (pt)
BG (1) BG65102B1 (pt)
BR (1) BR9610388A (pt)
CA (1) CA2230362A1 (pt)
CO (1) CO4750651A1 (pt)
CZ (1) CZ65598A3 (pt)
DE (1) DE69614150T2 (pt)
EA (1) EA000695B1 (pt)
ES (1) ES2160834T3 (pt)
GB (1) GB9518027D0 (pt)
HR (1) HRP960399A2 (pt)
HU (1) HUP9901260A3 (pt)
ID (1) ID17274A (pt)
IL (1) IL123414A0 (pt)
IS (1) IS4673A (pt)
NO (1) NO980923L (pt)
NZ (1) NZ318390A (pt)
PL (1) PL325329A1 (pt)
SK (1) SK28598A3 (pt)
TR (1) TR199800386T1 (pt)
TW (1) TW367326B (pt)
WO (1) WO1997009317A2 (pt)
YU (1) YU49796A (pt)
ZA (1) ZA967466B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR016212A1 (es) * 1998-04-28 2001-06-20 Astra Ab Uso de compuestos farmaceuticos que tienen una actividad antagonista de nmda para preparar un medicamento para el tratamiento del sindrome de intestino irritable (ibs), y composiciones farmaceuticas
CA2319153A1 (en) * 1998-06-08 1999-12-16 Advanced Medicine, Inc. Novel sodium channel drugs and uses
US6420354B1 (en) 1998-06-08 2002-07-16 Advanced Medicine, Inc. Sodium channel drugs and uses
GB9907965D0 (en) * 1999-04-09 1999-06-02 Glaxo Group Ltd Medical use
US6479498B1 (en) 1999-06-04 2002-11-12 Theravance, Inc. Sodium channel drugs and uses
NZ523851A (en) * 2000-07-21 2004-09-24 Ortho Mcneil Pharm Inc A method for use of carbamate enantiomers in preventing or treating neuropathic pain and cluster and migraine headache-associated pain
WO2003079972A2 (en) 2002-02-22 2003-10-02 New River Parmaceuticals Inc. Active agent delivery systems and methods for protecting and administering active agents
JP2004526714A (ja) * 2001-02-27 2004-09-02 テバ ファーマシューティカル インダストリーズ リミティド ラモトリジンの新しい結晶形およびそれらの調製方法
ATE357217T1 (de) * 2002-04-23 2007-04-15 Teva Pharma Pharmazeutische zusammensetzung enthaltend lamotrigine-partikel mit definierter morphologie
CA2514574A1 (en) * 2003-01-30 2004-08-12 Dynogen Pharmaceuticals, Inc. Use of sodium channel modulators for treating gastrointestinal tract disorders
GB0603087D0 (en) * 2006-02-15 2006-03-29 Glaxo Group Ltd Novel use
CN101641099A (zh) 2007-01-24 2010-02-03 葛兰素集团有限公司 包含3,5-二氨基-6-(2,3-二氯苯基)-1,2,4-三嗪或r(-)-2,4-二氨基-5-(2,3-二氯苯基)-6-氟甲基嘧啶和nk1的药物组合物
GB201111712D0 (en) 2011-07-08 2011-08-24 Gosforth Ct Holdings Pty Ltd Pharmaceutical compositions

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI67844C (fi) * 1979-06-01 1985-06-10 Wellcome Found Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 3,5-diamino-6-(substituerad fenyl)-1,2,4-triazinderivat
FI895821A0 (fi) * 1988-12-07 1989-12-05 Wellcome Found Farmaceutiskt aktiva cns foereningar.

Also Published As

Publication number Publication date
BG65102B1 (bg) 2007-02-28
JPH11512108A (ja) 1999-10-19
AU710091B2 (en) 1999-09-16
AU6986596A (en) 1997-03-27
TR199800386T1 (xx) 1998-05-21
ID17274A (id) 1997-12-18
CZ65598A3 (cs) 1998-07-15
KR19990044397A (ko) 1999-06-25
US6124308A (en) 2000-09-26
HUP9901260A2 (hu) 1999-09-28
CO4750651A1 (es) 1999-03-31
AP640A (en) 1998-04-14
HUP9901260A3 (en) 2001-04-28
ZA967466B (en) 1998-04-06
AR004192A1 (es) 1998-11-04
EA199800189A1 (ru) 1998-10-29
NO980923D0 (no) 1998-03-04
YU49796A (sh) 1999-07-28
NZ318390A (en) 1999-02-25
IL123414A0 (en) 1998-09-24
WO1997009317A3 (en) 1997-04-03
HRP960399A2 (en) 1998-04-30
WO1997009317A2 (en) 1997-03-13
MX9801680A (es) 1998-05-31
BG102342A (en) 1998-09-30
ATE203523T1 (de) 2001-08-15
EP0879230A2 (en) 1998-11-25
NO980923L (no) 1998-05-04
IS4673A (is) 1998-02-23
GB9518027D0 (en) 1995-11-08
CA2230362A1 (en) 1997-03-13
DE69614150T2 (de) 2001-11-22
ES2160834T3 (es) 2001-11-16
TW367326B (en) 1999-08-21
DE69614150D1 (de) 2001-08-30
EP0879230B1 (en) 2001-07-25
EA000695B1 (ru) 2000-02-28
AP9600857A0 (en) 1996-10-31
CN1200729A (zh) 1998-12-02
SK28598A3 (en) 1998-09-09
PL325329A1 (en) 1998-07-20

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Legal Events

Date Code Title Description
FB34 Technical and formal requirements: requirement - article 34 of industrial property law
FA14 Dismissal: dismissal - article 34 of industrial property law
B11T Dismissal of application maintained [chapter 11.20 patent gazette]