BR6908600D0 - Processo de preparar-1-glicosel-5-azacitosinas - Google Patents
Processo de preparar-1-glicosel-5-azacitosinasInfo
- Publication number
- BR6908600D0 BR6908600D0 BR20860069A BR20860069A BR6908600D0 BR 6908600 D0 BR6908600 D0 BR 6908600D0 BR 20860069 A BR20860069 A BR 20860069A BR 20860069 A BR20860069 A BR 20860069A BR 6908600 D0 BR6908600 D0 BR 6908600D0
- Authority
- BR
- Brazil
- Prior art keywords
- glycosel
- azacytosins
- preparing
- Prior art date
Links
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CS339968 | 1968-05-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR6908600D0 true BR6908600D0 (pt) | 1973-02-22 |
Family
ID=5373920
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR20860069A BR6908600D0 (pt) | 1968-05-08 | 1969-05-07 | Processo de preparar-1-glicosel-5-azacitosinas |
Country Status (12)
Country | Link |
---|---|
JP (1) | JPS4916435B1 (ja) |
AT (1) | AT306930B (ja) |
BE (1) | BE732268A (ja) |
BR (1) | BR6908600D0 (ja) |
CA (1) | CA921904A (ja) |
CH (1) | CH527207A (ja) |
DE (1) | DE1922702A1 (ja) |
ES (1) | ES366910A1 (ja) |
FR (1) | FR2008048A1 (ja) |
GB (1) | GB1227691A (ja) |
IT (1) | IT1037009B (ja) |
NL (1) | NL6906909A (ja) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2012888C3 (de) * | 1970-03-14 | 1981-04-02 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden |
US6905669B2 (en) | 2001-04-24 | 2005-06-14 | Supergen, Inc. | Compositions and methods for reestablishing gene transcription through inhibition of DNA methylation and histone deacetylase |
US6982253B2 (en) | 2002-06-05 | 2006-01-03 | Supergen, Inc. | Liquid formulation of decitabine and use of the same |
US6887855B2 (en) * | 2003-03-17 | 2005-05-03 | Pharmion Corporation | Forms of 5-azacytidine |
US6943249B2 (en) | 2003-03-17 | 2005-09-13 | Ash Stevens, Inc. | Methods for isolating crystalline Form I of 5-azacytidine |
US7038038B2 (en) | 2003-03-17 | 2006-05-02 | Pharmion Corporation | Synthesis of 5-azacytidine |
US20060014949A1 (en) * | 2004-07-13 | 2006-01-19 | Supergen Inc. | Compositions and formulations of decitabine polymorphs and methods of use thereof |
US7250416B2 (en) | 2005-03-11 | 2007-07-31 | Supergen, Inc. | Azacytosine analogs and derivatives |
US7700567B2 (en) | 2005-09-29 | 2010-04-20 | Supergen, Inc. | Oligonucleotide analogues incorporating 5-aza-cytosine therein |
JP5528806B2 (ja) | 2006-10-12 | 2014-06-25 | アステックス、セラピューティックス、リミテッド | 複合薬剤 |
WO2008044045A1 (en) | 2006-10-12 | 2008-04-17 | Astex Therapeutics Limited | Pharmaceutical combinations |
ES2969144T3 (es) | 2008-05-15 | 2024-05-16 | Celgene Corp | Formulaciones orales de análogos de citidina y métodos de uso de los mismos |
WO2010017547A1 (en) | 2008-08-08 | 2010-02-11 | Scinopharm Taiwan Ldt. | Process for making 5-azacytosine nucleosides and their derivatives |
JP6289361B2 (ja) | 2011-03-31 | 2018-03-07 | セルジーン インターナショナル サルル | 5−アザシチジンの合成 |
EP2750768B1 (en) | 2011-08-30 | 2018-10-03 | Astex Pharmaceuticals, Inc. | Decitabine derivative formulations |
JP6768722B2 (ja) | 2015-07-02 | 2020-10-14 | 大塚製薬株式会社 | 凍結乾燥医薬組成物 |
WO2017090264A1 (ja) | 2015-11-27 | 2017-06-01 | 大原薬品工業株式会社 | 5-アザシチジン又は其の2'-デオキシ体の5'位ジベンジル燐酸エステル |
JP6162349B1 (ja) | 2016-04-21 | 2017-07-12 | 大原薬品工業株式会社 | 5−アザシチジン類の糖部シリルエーテル誘導体 |
WO2017183215A1 (ja) | 2016-04-21 | 2017-10-26 | 大原薬品工業株式会社 | 5-アザシチジン類の糖部シリルエーテル誘導体 |
US10227374B2 (en) | 2016-04-21 | 2019-03-12 | Ohara Pharmaceutical Co., Ltd. | Silyl etherified derivatives of 5-azacytidines in carbohydrate moiety |
AU2018310857A1 (en) | 2017-08-03 | 2020-02-13 | Otsuka Pharmaceutical Co., Ltd. | Drug compound and purification methods thereof |
-
1969
- 1969-04-23 CH CH619669A patent/CH527207A/de not_active IP Right Cessation
- 1969-04-24 GB GB1227691D patent/GB1227691A/en not_active Expired
- 1969-04-29 BE BE732268D patent/BE732268A/xx unknown
- 1969-04-29 IT IT1620369A patent/IT1037009B/it active
- 1969-05-03 DE DE19691922702 patent/DE1922702A1/de active Pending
- 1969-05-06 NL NL6906909A patent/NL6906909A/xx unknown
- 1969-05-07 ES ES366910A patent/ES366910A1/es not_active Expired
- 1969-05-07 FR FR6914547A patent/FR2008048A1/fr active Pending
- 1969-05-07 BR BR20860069A patent/BR6908600D0/pt unknown
- 1969-05-07 AT AT439269A patent/AT306930B/de not_active IP Right Cessation
- 1969-05-08 CA CA050902A patent/CA921904A/en not_active Expired
- 1969-05-08 JP JP3545969A patent/JPS4916435B1/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
GB1227691A (ja) | 1971-04-07 |
CA921904A (en) | 1973-02-27 |
NL6906909A (ja) | 1969-11-11 |
FR2008048A1 (ja) | 1970-01-16 |
JPS4916435B1 (ja) | 1974-04-22 |
BE732268A (ja) | 1969-10-01 |
AT306930B (de) | 1973-04-25 |
CH527207A (de) | 1972-08-31 |
DE1922702A1 (de) | 1969-11-20 |
IT1037009B (it) | 1979-11-10 |
ES366910A1 (es) | 1971-03-16 |
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