BR6908600D0 - Processo de preparar-1-glicosel-5-azacitosinas - Google Patents

Processo de preparar-1-glicosel-5-azacitosinas

Info

Publication number
BR6908600D0
BR6908600D0 BR20860069A BR20860069A BR6908600D0 BR 6908600 D0 BR6908600 D0 BR 6908600D0 BR 20860069 A BR20860069 A BR 20860069A BR 20860069 A BR20860069 A BR 20860069A BR 6908600 D0 BR6908600 D0 BR 6908600D0
Authority
BR
Brazil
Prior art keywords
glycosel
azacytosins
preparing
Prior art date
Application number
BR20860069A
Other languages
English (en)
Portuguese (pt)
Inventor
F Sorns
A Piskala
Original Assignee
Ceskoslovenska Akademie Ved
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ceskoslovenska Akademie Ved filed Critical Ceskoslovenska Akademie Ved
Publication of BR6908600D0 publication Critical patent/BR6908600D0/pt

Links

BR20860069A 1968-05-08 1969-05-07 Processo de preparar-1-glicosel-5-azacitosinas BR6908600D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS339968 1968-05-08

Publications (1)

Publication Number Publication Date
BR6908600D0 true BR6908600D0 (pt) 1973-02-22

Family

ID=5373920

Family Applications (1)

Application Number Title Priority Date Filing Date
BR20860069A BR6908600D0 (pt) 1968-05-08 1969-05-07 Processo de preparar-1-glicosel-5-azacitosinas

Country Status (12)

Country Link
JP (1) JPS4916435B1 (ja)
AT (1) AT306930B (ja)
BE (1) BE732268A (ja)
BR (1) BR6908600D0 (ja)
CA (1) CA921904A (ja)
CH (1) CH527207A (ja)
DE (1) DE1922702A1 (ja)
ES (1) ES366910A1 (ja)
FR (1) FR2008048A1 (ja)
GB (1) GB1227691A (ja)
IT (1) IT1037009B (ja)
NL (1) NL6906909A (ja)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2012888C3 (de) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden
US6905669B2 (en) 2001-04-24 2005-06-14 Supergen, Inc. Compositions and methods for reestablishing gene transcription through inhibition of DNA methylation and histone deacetylase
US6982253B2 (en) 2002-06-05 2006-01-03 Supergen, Inc. Liquid formulation of decitabine and use of the same
US6887855B2 (en) * 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US6943249B2 (en) 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US7038038B2 (en) 2003-03-17 2006-05-02 Pharmion Corporation Synthesis of 5-azacytidine
US20060014949A1 (en) * 2004-07-13 2006-01-19 Supergen Inc. Compositions and formulations of decitabine polymorphs and methods of use thereof
US7250416B2 (en) 2005-03-11 2007-07-31 Supergen, Inc. Azacytosine analogs and derivatives
US7700567B2 (en) 2005-09-29 2010-04-20 Supergen, Inc. Oligonucleotide analogues incorporating 5-aza-cytosine therein
JP5528806B2 (ja) 2006-10-12 2014-06-25 アステックス、セラピューティックス、リミテッド 複合薬剤
WO2008044045A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
ES2969144T3 (es) 2008-05-15 2024-05-16 Celgene Corp Formulaciones orales de análogos de citidina y métodos de uso de los mismos
WO2010017547A1 (en) 2008-08-08 2010-02-11 Scinopharm Taiwan Ldt. Process for making 5-azacytosine nucleosides and their derivatives
JP6289361B2 (ja) 2011-03-31 2018-03-07 セルジーン インターナショナル サルル 5−アザシチジンの合成
EP2750768B1 (en) 2011-08-30 2018-10-03 Astex Pharmaceuticals, Inc. Decitabine derivative formulations
JP6768722B2 (ja) 2015-07-02 2020-10-14 大塚製薬株式会社 凍結乾燥医薬組成物
WO2017090264A1 (ja) 2015-11-27 2017-06-01 大原薬品工業株式会社 5-アザシチジン又は其の2'-デオキシ体の5'位ジベンジル燐酸エステル
JP6162349B1 (ja) 2016-04-21 2017-07-12 大原薬品工業株式会社 5−アザシチジン類の糖部シリルエーテル誘導体
WO2017183215A1 (ja) 2016-04-21 2017-10-26 大原薬品工業株式会社 5-アザシチジン類の糖部シリルエーテル誘導体
US10227374B2 (en) 2016-04-21 2019-03-12 Ohara Pharmaceutical Co., Ltd. Silyl etherified derivatives of 5-azacytidines in carbohydrate moiety
AU2018310857A1 (en) 2017-08-03 2020-02-13 Otsuka Pharmaceutical Co., Ltd. Drug compound and purification methods thereof

Also Published As

Publication number Publication date
GB1227691A (ja) 1971-04-07
CA921904A (en) 1973-02-27
NL6906909A (ja) 1969-11-11
FR2008048A1 (ja) 1970-01-16
JPS4916435B1 (ja) 1974-04-22
BE732268A (ja) 1969-10-01
AT306930B (de) 1973-04-25
CH527207A (de) 1972-08-31
DE1922702A1 (de) 1969-11-20
IT1037009B (it) 1979-11-10
ES366910A1 (es) 1971-03-16

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