AT306930B - Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen - Google Patents
Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinenInfo
- Publication number
- AT306930B AT306930B AT439269A AT439269A AT306930B AT 306930 B AT306930 B AT 306930B AT 439269 A AT439269 A AT 439269A AT 439269 A AT439269 A AT 439269A AT 306930 B AT306930 B AT 306930B
- Authority
- AT
- Austria
- Prior art keywords
- azacytosines
- glycosyl
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/12—Triazine radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS339968 | 1968-05-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AT306930B true AT306930B (de) | 1973-04-25 |
Family
ID=5373920
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT439269A AT306930B (de) | 1968-05-08 | 1969-05-07 | Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen |
Country Status (12)
| Country | Link |
|---|---|
| JP (1) | JPS4916435B1 (de) |
| AT (1) | AT306930B (de) |
| BE (1) | BE732268A (de) |
| BR (1) | BR6908600D0 (de) |
| CA (1) | CA921904A (de) |
| CH (1) | CH527207A (de) |
| DE (1) | DE1922702A1 (de) |
| ES (1) | ES366910A1 (de) |
| FR (1) | FR2008048A1 (de) |
| GB (1) | GB1227691A (de) |
| IT (1) | IT1037009B (de) |
| NL (1) | NL6906909A (de) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2012888C3 (de) * | 1970-03-14 | 1981-04-02 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden |
| US6905669B2 (en) | 2001-04-24 | 2005-06-14 | Supergen, Inc. | Compositions and methods for reestablishing gene transcription through inhibition of DNA methylation and histone deacetylase |
| US6982253B2 (en) | 2002-06-05 | 2006-01-03 | Supergen, Inc. | Liquid formulation of decitabine and use of the same |
| US6887855B2 (en) | 2003-03-17 | 2005-05-03 | Pharmion Corporation | Forms of 5-azacytidine |
| US6943249B2 (en) | 2003-03-17 | 2005-09-13 | Ash Stevens, Inc. | Methods for isolating crystalline Form I of 5-azacytidine |
| US7038038B2 (en) | 2003-03-17 | 2006-05-02 | Pharmion Corporation | Synthesis of 5-azacytidine |
| US20060014949A1 (en) * | 2004-07-13 | 2006-01-19 | Supergen Inc. | Compositions and formulations of decitabine polymorphs and methods of use thereof |
| US7250416B2 (en) | 2005-03-11 | 2007-07-31 | Supergen, Inc. | Azacytosine analogs and derivatives |
| US7700567B2 (en) | 2005-09-29 | 2010-04-20 | Supergen, Inc. | Oligonucleotide analogues incorporating 5-aza-cytosine therein |
| JP5528806B2 (ja) | 2006-10-12 | 2014-06-25 | アステックス、セラピューティックス、リミテッド | 複合薬剤 |
| EP2073807A1 (de) | 2006-10-12 | 2009-07-01 | Astex Therapeutics Limited | Pharmazeutische kombinationen |
| PT3782611T (pt) | 2008-05-15 | 2022-11-18 | Celgene Corp | Formulações orais de análogos da citidina e métodos de utilização dos mesmos |
| JP5650643B2 (ja) | 2008-08-08 | 2015-01-07 | サイノファーム タイワン リミテッド | ５−アザシトシンヌクレオシド及びその誘導体の製造方法 |
| BR112013025167A2 (pt) | 2011-03-31 | 2019-09-24 | Celgene Int Sarl | processo para preparar 5-azacitidina, ou um sal, solvato, hidrato, ou seu polimorfo, sal de 5-azacitidina, 5-azacitidina, ou um sal, solvato, hidrato, ou polimorfo |
| EP2750768B1 (de) | 2011-08-30 | 2018-10-03 | Astex Pharmaceuticals, Inc. | Decitabin-derivat zubereitungen |
| KR20180024010A (ko) | 2015-07-02 | 2018-03-07 | 오쓰까 세이야꾸 가부시키가이샤 | 동결건조된 약제학적 조성물 |
| WO2017090264A1 (ja) | 2015-11-27 | 2017-06-01 | 大原薬品工業株式会社 | ５－アザシチジン又は其の２'－デオキシ体の５'位ジベンジル燐酸エステル |
| WO2017183215A1 (ja) | 2016-04-21 | 2017-10-26 | 大原薬品工業株式会社 | ５－アザシチジン類の糖部シリルエーテル誘導体 |
| JP6162349B1 (ja) | 2016-04-21 | 2017-07-12 | 大原薬品工業株式会社 | ５−アザシチジン類の糖部シリルエーテル誘導体 |
| US10227374B2 (en) | 2016-04-21 | 2019-03-12 | Ohara Pharmaceutical Co., Ltd. | Silyl etherified derivatives of 5-azacytidines in carbohydrate moiety |
| EP3661522A2 (de) | 2017-08-03 | 2020-06-10 | Otsuka Pharmaceutical Co., Ltd. | Arzneimittelverbindung und reinigungsverfahren dafür |
| US20220332737A1 (en) * | 2019-06-07 | 2022-10-20 | Ludwig-Maximilians-Universität München | Carbocyclic nucleoside analogue |
-
1969
- 1969-04-23 CH CH619669A patent/CH527207A/de not_active IP Right Cessation
- 1969-04-24 GB GB1227691D patent/GB1227691A/en not_active Expired
- 1969-04-29 IT IT1620369A patent/IT1037009B/it active
- 1969-04-29 BE BE732268D patent/BE732268A/xx unknown
- 1969-05-03 DE DE19691922702 patent/DE1922702A1/de active Pending
- 1969-05-06 NL NL6906909A patent/NL6906909A/xx unknown
- 1969-05-07 ES ES366910A patent/ES366910A1/es not_active Expired
- 1969-05-07 FR FR6914547A patent/FR2008048A1/fr active Pending
- 1969-05-07 BR BR20860069A patent/BR6908600D0/pt unknown
- 1969-05-07 AT AT439269A patent/AT306930B/de not_active IP Right Cessation
- 1969-05-08 JP JP3545969A patent/JPS4916435B1/ja active Pending
- 1969-05-08 CA CA050902A patent/CA921904A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FR2008048A1 (de) | 1970-01-16 |
| ES366910A1 (es) | 1971-03-16 |
| IT1037009B (it) | 1979-11-10 |
| CA921904A (en) | 1973-02-27 |
| DE1922702A1 (de) | 1969-11-20 |
| CH527207A (de) | 1972-08-31 |
| GB1227691A (de) | 1971-04-07 |
| JPS4916435B1 (de) | 1974-04-22 |
| BE732268A (de) | 1969-10-01 |
| BR6908600D0 (pt) | 1973-02-22 |
| NL6906909A (de) | 1969-11-11 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CH507249A (de) | Verfahren zur Herstellung von 2-Brom-a-ergokryptin | |
| AT306930B (de) | Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen | |
| AT291254B (de) | Verfahren zur herstellung von 3-amino-4jod-5-methyllisoxazolen | |
| AT296964B (de) | Verfahren zur Herstellung von 1-Hydroxyphenyl-2-aminoäthanolen | |
| CH501573A (de) | Verfahren zur Herstellung von Trimethyl-p-benzochinon | |
| AT294064B (de) | Verfahren zur Herstellung von 1-Alkyl-2-aminomethylpyrrolidinen | |
| CH520135A (de) | Verfahren zur Herstellung von Erythromycylamin | |
| CH516529A (de) | Verfahren zur Herstellung von 4-Cyano-4-phenyl-aminocyclohexanen | |
| AT296254B (de) | Verfahren zur Herstellung von 2-Acyloxythionobenzamiden | |
| CH486444A (de) | Verfahren zur Herstellung von 7-Cyan-cumarinen | |
| CH513141A (de) | Verfahren zur Herstellung von Glyoxaldithiosemicarbazonen | |
| CH520672A (de) | Verfahren zur Herstellung von Chlorfluorpyridinen | |
| AT314097B (de) | Verfahren zur Herstellung von 19-Norsteroiden | |
| AT286252B (de) | Verfahren zur Herstellung von 3-Aminopropanolen | |
| AT292205B (de) | Verfahren zur Herstellung von 1-Peracylglykosyl-5-azacytosinen | |
| AT289737B (de) | Verfahren zur Herstellung von Sulfatobetainen | |
| CH517703A (de) | Verfahren zur Herstellung von Glycyl-L-tryptophyl-L-methionyl-glycinamiden | |
| AT296251B (de) | Verfahren zur Herstellung von Methylcyclohexenen | |
| AT290555B (de) | Verfahren zur Herstellung von Triorganosilanolen | |
| CH517758A (de) | Verfahren zur Herstellung von 1-Pyridyl-2-imidazolonen | |
| CH518290A (de) | Verfahren zur Herstellung von Hydroxyphenazin-di-N-oxiden | |
| AT291577B (de) | Verfahren zur Herstellung von Polyacyloxamidrazonen | |
| CH521333A (de) | Verfahren zur Herstellung von 9a-Fluor-16-methylen-prednisolon-21-acetat | |
| CH514524A (de) | Verfahren zur Herstellung von Cyclopent-2-enyl-phenolen | |
| CH487927A (de) | Verfahren zur Herstellung von 7-Triazolyl-cumarinen |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ELJ | Ceased due to non-payment of the annual fee |