BR112021020320A2 - Processo para produção contínua de um granulado de substância ativa - Google Patents
Processo para produção contínua de um granulado de substância ativaInfo
- Publication number
- BR112021020320A2 BR112021020320A2 BR112021020320A BR112021020320A BR112021020320A2 BR 112021020320 A2 BR112021020320 A2 BR 112021020320A2 BR 112021020320 A BR112021020320 A BR 112021020320A BR 112021020320 A BR112021020320 A BR 112021020320A BR 112021020320 A2 BR112021020320 A2 BR 112021020320A2
- Authority
- BR
- Brazil
- Prior art keywords
- active substance
- solid particles
- continuous production
- granulate
- process space
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 8
- 239000013543 active substance Substances 0.000 title abstract 6
- 239000008187 granular material Substances 0.000 title abstract 4
- 238000010924 continuous production Methods 0.000 title abstract 3
- 239000002245 particle Substances 0.000 abstract 5
- 239000007787 solid Substances 0.000 abstract 5
- 239000007788 liquid Substances 0.000 abstract 3
- XZWYZXLIPXDOLR-UHFFFAOYSA-N metformin Chemical compound CN(C)C(=N)NC(N)=N XZWYZXLIPXDOLR-UHFFFAOYSA-N 0.000 abstract 2
- 229960003105 metformin Drugs 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 239000007921 spray Substances 0.000 abstract 2
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical compound Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 abstract 1
- 238000009825 accumulation Methods 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Glanulating (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19168673.2A EP3721870A1 (de) | 2019-04-11 | 2019-04-11 | Verfahren zur kontinuierlichen herstellung eines wirkstoffgranulats |
| PCT/EP2020/060277 WO2020208201A1 (de) | 2019-04-11 | 2020-04-09 | Verfahren zur kontinuierlichen herstellung eines wirkstoffgranulats |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112021020320A2 true BR112021020320A2 (pt) | 2021-12-14 |
Family
ID=66105201
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112021020320A BR112021020320A2 (pt) | 2019-04-11 | 2020-04-09 | Processo para produção contínua de um granulado de substância ativa |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20220323361A1 (enExample) |
| EP (2) | EP3721870A1 (enExample) |
| JP (1) | JP7620565B2 (enExample) |
| CN (1) | CN114126591A (enExample) |
| AU (1) | AU2020272151B2 (enExample) |
| BR (1) | BR112021020320A2 (enExample) |
| CA (1) | CA3136529A1 (enExample) |
| IL (1) | IL287126A (enExample) |
| WO (1) | WO2020208201A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3721871A1 (de) * | 2019-04-11 | 2020-10-14 | ADD Advanced Drug Delivery Technologies, Ltd. | Verfahren zur kontinuierlichen herstellung eines wirkstoffgranulats |
| KR102857295B1 (ko) | 2020-11-24 | 2025-09-08 | 나노폼 핀란드 오와이제이 | 입자 생성을 위한 시스템, 장치, 기기 및 방법 |
| CN116422227B (zh) * | 2022-12-09 | 2024-01-30 | 山东奥诺能源科技股份有限公司 | 一种流化床造粒机 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19514187C1 (de) * | 1995-04-21 | 1996-05-15 | Degussa | Verfahren und Vorrichtung zur Herstellung von Granulaten durch Wirbelschicht-Sprühgranulation |
| US6117451A (en) | 1998-08-25 | 2000-09-12 | Pharmalogix, Inc. | Direct compression metformin hydrochloride tablets |
| DE10004939C1 (de) | 2000-02-05 | 2001-08-23 | Lothar Moerl | Steuerbare Gasanströmeinrichtung für Strahlschichtapparate |
| EP1238662B1 (en) | 2001-03-07 | 2006-05-31 | Dainippon Sumitomo Pharma Co., Ltd. | Method for manufacturing drug granules, the drug granules and pharmaceutical preparation containing the drug granules |
| US6667054B2 (en) | 2001-12-05 | 2003-12-23 | Bernard Charles Sherman | Metformin hydrochloride tablets |
| DE10322062A1 (de) | 2003-05-15 | 2004-12-02 | Glatt Ingenieurtechnik Gmbh | Verfahren und Vorrichtung zum Aufbringen von Flüssigkeiten in eine Feststoffströmung eines Strahlschichtapparates |
| PT1638678E (pt) | 2003-06-11 | 2012-01-05 | Glatt Ingtech Gmbh | Método para produção de granulados enzimáticos e granulados enzimáticos assim obtidos |
| EP1781253A1 (en) * | 2004-07-01 | 2007-05-09 | Warner-Lambert Company LLC | Preparation of pharmaceutical compositions containing nanoparticles |
| DE102007012105A1 (de) | 2007-03-13 | 2008-09-18 | Add Advanced Drug Delivery Technologies Ltd. | Pellets enthaltend pharmazeutische Substanz, Verfahren zu deren Herstellung und deren Verwendung |
| CN102970981A (zh) * | 2010-07-06 | 2013-03-13 | 詹森药业有限公司 | 糖尿病协同治疗制剂 |
| WO2013143688A1 (en) * | 2012-03-26 | 2013-10-03 | Glatt Ag | Taste-masked ibuprofen granules |
| WO2015012365A1 (ja) * | 2013-07-25 | 2015-01-29 | 株式会社 三和化学研究所 | 医薬製剤 |
| KR101642193B1 (ko) | 2014-10-13 | 2016-07-25 | 씨제이헬스케어 주식회사 | 메트포르민 서방성 제제 및 그의 제조방법 |
| WO2018034627A1 (en) * | 2016-08-18 | 2018-02-22 | İlko Ilaç Sanayi Ve Ticaret Anonim Şirketi | Pharmaceutical composition of antidiabetic tablet |
-
2019
- 2019-04-11 EP EP19168673.2A patent/EP3721870A1/de active Pending
-
2020
- 2020-04-09 CA CA3136529A patent/CA3136529A1/en active Pending
- 2020-04-09 WO PCT/EP2020/060277 patent/WO2020208201A1/de not_active Ceased
- 2020-04-09 AU AU2020272151A patent/AU2020272151B2/en active Active
- 2020-04-09 EP EP20722226.6A patent/EP3952843B1/de active Active
- 2020-04-09 US US17/602,356 patent/US20220323361A1/en active Pending
- 2020-04-09 CN CN202080042850.1A patent/CN114126591A/zh active Pending
- 2020-04-09 JP JP2021560695A patent/JP7620565B2/ja active Active
- 2020-04-09 BR BR112021020320A patent/BR112021020320A2/pt unknown
-
2021
- 2021-10-10 IL IL287126A patent/IL287126A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL287126A (en) | 2022-01-01 |
| EP3721870A1 (de) | 2020-10-14 |
| WO2020208201A1 (de) | 2020-10-15 |
| CA3136529A1 (en) | 2020-10-15 |
| JP7620565B2 (ja) | 2025-01-23 |
| EP3952843B1 (de) | 2025-08-06 |
| EP3952843A1 (de) | 2022-02-16 |
| CN114126591A (zh) | 2022-03-01 |
| AU2020272151A1 (en) | 2021-12-09 |
| AU2020272151B2 (en) | 2025-07-03 |
| JP2022528570A (ja) | 2022-06-14 |
| US20220323361A1 (en) | 2022-10-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06W | Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette] |