BR112019027889A2 - método de tratamento e formas de dosagem do mesmo - Google Patents
método de tratamento e formas de dosagem do mesmo Download PDFInfo
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- BR112019027889A2 BR112019027889A2 BR112019027889-3A BR112019027889A BR112019027889A2 BR 112019027889 A2 BR112019027889 A2 BR 112019027889A2 BR 112019027889 A BR112019027889 A BR 112019027889A BR 112019027889 A2 BR112019027889 A2 BR 112019027889A2
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- buprenorphine
- oxycodone
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4748—Quinolines; Isoquinolines forming part of bridged ring systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
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- A—HUMAN NECESSITIES
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- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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Landscapes
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- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
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- Pain & Pain Management (AREA)
- Dermatology (AREA)
- Addiction (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| US201762527337P | 2017-06-30 | 2017-06-30 | |
| US62/527,337 | 2017-06-30 | ||
| PCT/US2018/040460 WO2019006404A1 (en) | 2017-06-30 | 2018-06-29 | METHOD OF TREATMENT AND DOSAGE FORMS |
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| BR112019027889A2 true BR112019027889A2 (pt) | 2020-07-07 |
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| BR112019027889-3A BR112019027889A2 (pt) | 2017-06-30 | 2018-06-29 | método de tratamento e formas de dosagem do mesmo |
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| US4785000A (en) | 1986-06-18 | 1988-11-15 | The Rockefeller University | Method of treating patients suffering from chronic pain or chronic cough |
| US4769372A (en) | 1986-06-18 | 1988-09-06 | The Rockefeller University | Method of treating patients suffering from chronic pain or chronic cough |
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| US9211293B2 (en) | 2011-12-15 | 2015-12-15 | Alkermes Pharma Ireland Limited | Opioid agonist antagonist combinations |
| IN2014DN09238A (enExample) | 2012-04-17 | 2015-07-10 | Purdue Pharma Lp | |
| RU2012122945A (ru) | 2012-06-04 | 2013-12-10 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Санкт-Петербургский государственный медицинский университет имени академика И.П. Павлова" Министерства здравоохранения и социального развития Российской Федерации | Аналгетическое средство |
| TW201613590A (en) * | 2014-09-12 | 2016-04-16 | Purdue Pharma Lp | Systems and methods for attenuating opioid-induced euphoria |
| US9849124B2 (en) * | 2014-10-17 | 2017-12-26 | Purdue Pharma L.P. | Systems and methods for treating an opioid-induced adverse pharmacodynamic response |
-
2018
- 2018-06-29 BR BR112019027889-3A patent/BR112019027889A2/pt not_active Application Discontinuation
- 2018-06-29 CA CA3068036A patent/CA3068036A1/en active Pending
- 2018-06-29 JP JP2019572473A patent/JP2020526500A/ja not_active Withdrawn
- 2018-06-29 AU AU2018291397A patent/AU2018291397A1/en not_active Abandoned
- 2018-06-29 EP EP18823900.8A patent/EP3645000A4/en active Pending
- 2018-06-29 KR KR1020207002939A patent/KR20200022026A/ko not_active Withdrawn
- 2018-06-29 US US16/625,011 patent/US12201629B2/en active Active
- 2018-06-29 WO PCT/US2018/040460 patent/WO2019006404A1/en not_active Ceased
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2019
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2023
- 2023-05-09 JP JP2023077065A patent/JP2023109829A/ja active Pending
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2024
- 2024-06-14 US US18/743,430 patent/US20240408078A1/en active Pending
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|---|---|
| JP2020526500A (ja) | 2020-08-31 |
| AU2018291397A1 (en) | 2020-01-16 |
| EP3645000A1 (en) | 2020-05-06 |
| US20200215052A1 (en) | 2020-07-09 |
| WO2019006404A1 (en) | 2019-01-03 |
| KR20200022026A (ko) | 2020-03-02 |
| US12201629B2 (en) | 2025-01-21 |
| CA3068036A1 (en) | 2019-01-03 |
| JP2023109829A (ja) | 2023-08-08 |
| EP3645000A4 (en) | 2021-03-24 |
| US20240408078A1 (en) | 2024-12-12 |
| IL271727A (en) | 2020-02-27 |
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