BR112016027819A8 - processo de preparação de derivados de tiazole - Google Patents

processo de preparação de derivados de tiazole

Info

Publication number
BR112016027819A8
BR112016027819A8 BR112016027819A BR112016027819A BR112016027819A8 BR 112016027819 A8 BR112016027819 A8 BR 112016027819A8 BR 112016027819 A BR112016027819 A BR 112016027819A BR 112016027819 A BR112016027819 A BR 112016027819A BR 112016027819 A8 BR112016027819 A8 BR 112016027819A8
Authority
BR
Brazil
Prior art keywords
thiazole derivatives
preparing thiazole
preparing
derivatives
preparation
Prior art date
Application number
BR112016027819A
Other languages
English (en)
Other versions
BR112016027819A2 (pt
BR112016027819B1 (pt
Inventor
Hömberger Günter
James Ford Mark
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR112016027819A2 publication Critical patent/BR112016027819A2/pt
Publication of BR112016027819A8 publication Critical patent/BR112016027819A8/pt
Publication of BR112016027819B1 publication Critical patent/BR112016027819B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

processo de preparação de derivados de tiazole. a presente invenção está relacionada a um novo processo de preparação de derivados de tiazole.
BR112016027819-4A 2014-05-28 2015-05-22 Processo de preparação de derivados de tiazole BR112016027819B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14170156 2014-05-28
EP14170156.5 2014-05-28
PCT/EP2015/061455 WO2015181097A1 (en) 2014-05-28 2015-05-22 Process for preparing thiazole derivatives

Publications (3)

Publication Number Publication Date
BR112016027819A2 BR112016027819A2 (pt) 2017-08-22
BR112016027819A8 true BR112016027819A8 (pt) 2021-07-20
BR112016027819B1 BR112016027819B1 (pt) 2023-05-02

Family

ID=50828732

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016027819-4A BR112016027819B1 (pt) 2014-05-28 2015-05-22 Processo de preparação de derivados de tiazole

Country Status (12)

Country Link
US (1) US10336742B2 (pt)
EP (1) EP3148993B1 (pt)
JP (1) JP6546936B2 (pt)
KR (1) KR102445983B1 (pt)
CN (1) CN106414437B (pt)
BR (1) BR112016027819B1 (pt)
DK (1) DK3148993T3 (pt)
ES (1) ES2725458T3 (pt)
IL (1) IL248565B (pt)
MX (1) MX2016015624A (pt)
TW (1) TWI660955B (pt)
WO (1) WO2015181097A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110818708B (zh) * 2018-08-14 2022-04-01 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剂
CN111848612B (zh) * 2019-07-31 2021-09-14 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剂
WO2021122752A1 (en) 2019-12-19 2021-06-24 Bayer Aktiengesellschaft Process for preparing [3-chloro-2-[3-[2-[1-(2-chloroacetyl)-4-piperidyl]thiazol-4-yl]-4,5-dihydroisoxazol-5-yl]phenyl] methanesulfonate
WO2023007427A1 (en) * 2021-07-29 2023-02-02 Pi Industries Ltd. Preparation of phenyl sulfilimines or sulfoximines containing thiazolyl-piperidinyl compounds and intermediates thereof

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2505397A1 (en) 2002-11-08 2004-05-21 Warner-Lambert Company Llc Phenylalkyl and pyridylalkyl piperazine derivatives
US7115596B2 (en) 2002-12-20 2006-10-03 Pharmacia Corporation Thiazole compounds as integrin receptor antagonists derivatives
EP1623355A1 (en) 2003-05-15 2006-02-08 Nokia Corporation Transferring content between digital rights management systems
DE602006008932D1 (de) 2005-05-25 2009-10-15 Actelion Pharmaceuticals Ltd Neue antibiotische derivate
WO2007056170A2 (en) 2005-11-02 2007-05-18 Bayer Healthcare Ag Pyrrolo[2,1-f] [1,2,4] triazin-4-ylamines igf-1r kinase inhibitors for the treatment of cancer and other hyperproliferative diseases
EP1878730A1 (en) 2006-07-12 2008-01-16 Bayer Schering Pharma Aktiengesellschaft Substituted isoxazolines, pharmaceutical compositions containing the same, methods of preparing the same, and uses of the same
WO2008013622A2 (en) 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
TWI428091B (zh) * 2007-10-23 2014-03-01 Du Pont 殺真菌劑混合物
BRPI0905758A2 (pt) * 2008-01-25 2015-07-14 Du Pont Composto, método de controle de doenças de plantas e composição fungicida
CN103965187A (zh) 2008-01-25 2014-08-06 杜邦公司 杀真菌杂环化合物
EP2141164A1 (en) 2008-07-01 2010-01-06 Mutabilis New 1,2,4-triazine derivatives and biological applications thereof
ES2624828T3 (es) 2008-07-16 2017-07-17 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros
EP2358709B1 (en) * 2008-12-02 2014-01-22 E. I. du Pont de Nemours and Company Fungicidal heterocyclic compounds
TWI508962B (zh) * 2009-04-22 2015-11-21 Du Pont 氮雜環醯胺之固體形態
KR101151415B1 (ko) 2009-07-10 2012-06-01 양지화학 주식회사 Ｃｃｒ２ 길항제로서의 피페라지닐에틸 3-아미노피롤리딘 유도체
BR112012013801A2 (pt) * 2009-12-11 2019-09-24 Du Pont composto,método para inibir a atividade de hidrolase de amida de ácido graxo em um indivíduo,composição farmacêutica e método para tratar um individuo com dor
US8759527B2 (en) * 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
AU2012280508A1 (en) 2011-07-01 2013-12-12 Bayer Intellectual Property Gmbh Hydroxymethylaryl-substituted pyrrolotriazines as ALK1 inhibitors
DK2921484T3 (en) * 2011-12-27 2018-11-12 Bayer Cropscience Ag oxazole

Also Published As

Publication number Publication date
IL248565B (en) 2019-05-30
CN106414437A (zh) 2017-02-15
IL248565A0 (en) 2016-12-29
EP3148993B1 (en) 2019-02-27
JP6546936B2 (ja) 2019-07-17
DK3148993T3 (da) 2019-05-20
BR112016027819A2 (pt) 2017-08-22
JP2017516780A (ja) 2017-06-22
MX2016015624A (es) 2017-02-27
BR112016027819B1 (pt) 2023-05-02
TWI660955B (zh) 2019-06-01
EP3148993A1 (en) 2017-04-05
ES2725458T3 (es) 2019-09-24
US20170240541A1 (en) 2017-08-24
TW201625604A (zh) 2016-07-16
KR102445983B1 (ko) 2022-09-21
WO2015181097A1 (en) 2015-12-03
KR20170012307A (ko) 2017-02-02
US10336742B2 (en) 2019-07-02
CN106414437B (zh) 2019-06-21

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 22/05/2015, OBSERVADAS AS CONDICOES LEGAIS