BR112016021034A8 - composição farmacêutica, uso da mesma e kit - Google Patents

composição farmacêutica, uso da mesma e kit

Info

Publication number
BR112016021034A8
BR112016021034A8 BR112016021034A BR112016021034A BR112016021034A8 BR 112016021034 A8 BR112016021034 A8 BR 112016021034A8 BR 112016021034 A BR112016021034 A BR 112016021034A BR 112016021034 A BR112016021034 A BR 112016021034A BR 112016021034 A8 BR112016021034 A8 BR 112016021034A8
Authority
BR
Brazil
Prior art keywords
disease
kit
pharmaceutical composition
carbidopa
antioxidant
Prior art date
Application number
BR112016021034A
Other languages
English (en)
Portuguese (pt)
Other versions
BR112016021034A2 (pt
Inventor
Yacoby-Zeevi Oron
Original Assignee
Neuroderm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53488380&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112016021034(A8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Neuroderm Ltd filed Critical Neuroderm Ltd
Publication of BR112016021034A2 publication Critical patent/BR112016021034A2/pt
Publication of BR112016021034A8 publication Critical patent/BR112016021034A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/133Amines having hydroxy groups, e.g. sphingosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/20Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR112016021034A 2014-03-13 2015-03-12 composição farmacêutica, uso da mesma e kit BR112016021034A8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461952477P 2014-03-13 2014-03-13
US201461990967P 2014-05-09 2014-05-09
PCT/IL2015/050258 WO2015136538A1 (en) 2014-03-13 2015-03-12 Dopa decarboxylase inhibitor compositions

Publications (2)

Publication Number Publication Date
BR112016021034A2 BR112016021034A2 (pt) 2017-08-15
BR112016021034A8 true BR112016021034A8 (pt) 2021-06-29

Family

ID=53488380

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016021034A BR112016021034A8 (pt) 2014-03-13 2015-03-12 composição farmacêutica, uso da mesma e kit

Country Status (19)

Country Link
US (5) US10022320B2 (https=)
EP (3) EP3777833B1 (https=)
JP (2) JP6591995B2 (https=)
CN (1) CN106413754B (https=)
AU (1) AU2015228369B2 (https=)
BR (1) BR112016021034A8 (https=)
CA (1) CA2942244C (https=)
DK (2) DK3116475T3 (https=)
ES (2) ES2967693T3 (https=)
FI (1) FI3777833T3 (https=)
HR (2) HRP20201948T1 (https=)
HU (2) HUE064818T2 (https=)
IL (1) IL247668B (https=)
MX (1) MX2016011837A (https=)
PL (2) PL3777833T3 (https=)
PT (2) PT3777833T (https=)
RS (1) RS65060B1 (https=)
RU (1) RU2684105C2 (https=)
WO (1) WO2015136538A1 (https=)

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WO2018154447A1 (en) * 2017-02-21 2018-08-30 Neuroderm Ltd Dopa decarboxylase inhibitor compositions
CN113015531A (zh) 2018-11-15 2021-06-22 艾伯维公司 用于皮下施用的药物调配物
WO2020178810A1 (en) * 2019-03-04 2020-09-10 Neuroderm, Ltd. Pharmaceutical compositions comprising levodopa amide derivatives and uses thereof
CN111701024B (zh) * 2020-05-26 2022-05-24 上海京新生物医药有限公司 一种左旋多巴制剂及其制备方法及其应用
US11844754B2 (en) 2020-11-17 2023-12-19 Neuroderm, Ltd. Methods for treatment of Parkinson's disease
US11331293B1 (en) 2020-11-17 2022-05-17 Neuroderm, Ltd. Method for treatment of Parkinson's disease
US11213502B1 (en) 2020-11-17 2022-01-04 Neuroderm, Ltd. Method for treatment of parkinson's disease
CN113396897B (zh) * 2021-07-26 2022-06-07 苏州华测生物技术有限公司 一种稳定生物基质中卡比多巴/左旋多巴的方法
US12161612B2 (en) 2023-04-14 2024-12-10 Neuroderm, Ltd. Methods and compositions for reducing symptoms of Parkinson's disease

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Also Published As

Publication number Publication date
JP6591995B2 (ja) 2019-10-16
PT3116475T (pt) 2020-12-15
JP2020011977A (ja) 2020-01-23
US20190151233A1 (en) 2019-05-23
DK3116475T3 (da) 2020-12-07
HRP20231716T1 (hr) 2024-03-15
HUE052642T2 (hu) 2021-05-28
CA2942244C (en) 2022-08-23
AU2015228369B2 (en) 2020-05-21
US20260102334A1 (en) 2026-04-16
ES2967693T3 (es) 2024-05-03
JP2017507973A (ja) 2017-03-23
HRP20201948T1 (hr) 2021-01-22
IL247668A0 (en) 2016-11-30
CA2942244A1 (en) 2015-09-17
MX2016011837A (es) 2017-04-27
CN106413754A (zh) 2017-02-15
US20210038505A1 (en) 2021-02-11
ES2836325T3 (es) 2021-06-24
EP3777833A1 (en) 2021-02-17
IL247668B (en) 2020-09-30
RS65060B1 (sr) 2024-02-29
PL3777833T3 (pl) 2024-03-25
HUE064818T2 (hu) 2024-04-28
EP3777833B1 (en) 2023-10-18
CN106413754B (zh) 2019-11-29
RU2684105C2 (ru) 2019-04-04
US20150352212A1 (en) 2015-12-10
RU2016135952A3 (https=) 2018-09-12
EP3116475A1 (en) 2017-01-18
EP3116475B1 (en) 2020-11-04
EP4299128A2 (en) 2024-01-03
WO2015136538A1 (en) 2015-09-17
EP4299128A3 (en) 2024-04-17
BR112016021034A2 (pt) 2017-08-15
DK3777833T3 (da) 2023-12-18
FI3777833T3 (fi) 2024-01-03
RU2016135952A (ru) 2018-04-13
PT3777833T (pt) 2024-01-09
JP6770158B2 (ja) 2020-10-14
US10624839B2 (en) 2020-04-21
PL3116475T3 (pl) 2021-02-08
US20230240980A1 (en) 2023-08-03
US10022320B2 (en) 2018-07-17
AU2015228369A1 (en) 2016-10-27

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