BR112014000428A2 - formulação ativa para uso em produtos de alimentação - Google Patents

formulação ativa para uso em produtos de alimentação

Info

Publication number
BR112014000428A2
BR112014000428A2 BR112014000428A BR112014000428A BR112014000428A2 BR 112014000428 A2 BR112014000428 A2 BR 112014000428A2 BR 112014000428 A BR112014000428 A BR 112014000428A BR 112014000428 A BR112014000428 A BR 112014000428A BR 112014000428 A2 BR112014000428 A2 BR 112014000428A2
Authority
BR
Brazil
Prior art keywords
formula
coo
active compound
salt
carrier
Prior art date
Application number
BR112014000428A
Other languages
English (en)
Other versions
BR112014000428B1 (pt
Inventor
Nikolaos Vogiatzis
Symone Kok
Original Assignee
Purac Biochem Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Purac Biochem Bv filed Critical Purac Biochem Bv
Publication of BR112014000428A2 publication Critical patent/BR112014000428A2/pt
Publication of BR112014000428B1 publication Critical patent/BR112014000428B1/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/23Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin of acids having a carboxyl group bound to a chain of seven or more carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/105Aliphatic or alicyclic compounds
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/158Fatty acids; Fats; Products containing oils or fats
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/20Inorganic substances, e.g. oligoelements
    • A23K20/24Compounds of alkaline earth metals, e.g. magnesium
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K40/00Shaping or working-up of animal feeding-stuffs
    • A23K40/10Shaping or working-up of animal feeding-stuffs by agglomeration; by granulation, e.g. making powders
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K50/00Feeding-stuffs specially adapted for particular animals
    • A23K50/70Feeding-stuffs specially adapted for particular animals for birds
    • A23K50/75Feeding-stuffs specially adapted for particular animals for birds for poultry
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Animal Husbandry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Emergency Medicine (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fodder In General (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

abstract active formulation for use in feed products the invention pertains to a free-flowing particulate powder comprising 2-90 wt.% of an active compound on a carrier, wherein the carrier has a d(v,0.1) of at least 100 microns, with the active compound being selected from lactylate in accordance with formula 1, formula 1 r2-coo-[-ch(ch3)-coo]n-r1 or a na, k, ca, mg, fe(ii), zn, nh4, or cu(ii) salt thereof, a glycolylate of formula 2, formula 2: r2-coo-[-ch2-coo]n-r1 or a na, k, ca, mg, fe(ii), zn, nh4, or cu(ii) salt thereof a lactate ester of formula 3, formula 3: ho-ch(ch3)-coo-r2 and/or a glycolic acid ester of formula 4, formula 4: ho-ch2-coo-r2 wherein in the above formulae r1 is selected from h, n stands for an integer with a value of 1-10, and r2 stands for a c1-c35 alkyl or alkenyl chain which may be branched or unbranched. the powder allows easy provision of the active compound to feed compositions. ___________________________________________________________________________________ tradução do resumo resumo patente de invenção: "formulação ativa para uso em produtos de alimentação". a invenção pertence a um pulverizado em partículas de escoamento livre compreendendo2-90% em peso de um composto ativo sobre um carreador, onde o carreador tem um d (v, 0,1) de pelo menos 100 micra, com o composto ativo sendo selecionado de lactilato de acordo com fórmula (1), fórmula (1): r2-coo-[-ch(ch3)-coo]n-r1 ou um seu sal de na, k, ca, mg, fe(ii), zn, nh4 ou cu(ii), um glicolato de fórmula (2), fórmula (2): r2-coo-[-ch2-coo]n-r1 ou um seu sal de na, k, ca, mg, fe(ii), zn, nh4 ou cu(ii); um éster de lactato de fórmula (3), fórmula (#): ho-ch(ch3)-coo-r2 e/ou um éster de ácido glicólico de fórmula (4), fórmula (4): ho-ch2-coo-r2 onde nas fórmulas acima r1 é selecionado de h, n representa um inteiro com um valor de 1-10, e r2 representa uma cadeia c1-35 alquila ou alquenila que pode ser ramificada ou não-ramificada. o pulverizado permite fácil provisão do composto ativo para composições de alimentação.
BR112014000428-5A 2011-07-08 2012-07-03 Pulverizado, processo para fabricação e uso do mesmo, e composição de nutrição animal BR112014000428B1 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161505810P 2011-07-08 2011-07-08
EP11173177 2011-07-08
US61/505,810 2011-07-08
EP11173177.4 2011-07-08
PCT/EP2012/062926 WO2013007558A2 (en) 2011-07-08 2012-07-03 Active formulation for use in feed products

Publications (2)

Publication Number Publication Date
BR112014000428A2 true BR112014000428A2 (pt) 2017-01-10
BR112014000428B1 BR112014000428B1 (pt) 2019-09-17

Family

ID=47506621

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014000428-5A BR112014000428B1 (pt) 2011-07-08 2012-07-03 Pulverizado, processo para fabricação e uso do mesmo, e composição de nutrição animal

Country Status (11)

Country Link
US (2) US9849105B2 (pt)
EP (1) EP2729015B1 (pt)
JP (1) JP6460791B2 (pt)
KR (1) KR102196004B1 (pt)
CN (1) CN103732077B (pt)
BR (1) BR112014000428B1 (pt)
CA (1) CA2841149C (pt)
MX (1) MX357070B (pt)
PL (1) PL2729015T3 (pt)
RU (1) RU2603915C2 (pt)
WO (1) WO2013007558A2 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3536163A1 (en) 2013-10-30 2019-09-11 Purac Biochem B.V. Method for manufacturing a feed product
CN110290710B (zh) * 2017-02-14 2023-12-19 帝斯曼知识产权资产管理有限公司 水分散性制剂
CN110381747A (zh) * 2017-02-14 2019-10-25 帝斯曼知识产权资产管理有限公司 贮存稳定的配制物
CN109744362B (zh) * 2018-11-19 2022-03-29 浙江海洋大学 罗非鱼混合型饲料添加剂
CN115867145A (zh) * 2020-07-03 2023-03-28 普拉克生化公司 稳定的液体动物饲料成分

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3081154A (en) * 1959-11-17 1963-03-12 Grace W R & Co Process for preparing fine size silica
US3284209A (en) * 1960-10-06 1966-11-08 Grace W R & Co Re-expanding compressed exfoliated vermiculite
GB1581744A (en) * 1976-03-22 1980-12-17 Unilever Ltd Edible composition
JPS57123102A (en) * 1981-01-12 1982-07-31 Odeitsusei Ekusupooto Co Ltd Mildew preventive composition for feed
US4603143A (en) * 1983-05-02 1986-07-29 Basf Corporation Free-flowing, high density, fat soluble vitamin powders with improved stability
US5002780A (en) * 1987-07-31 1991-03-26 Caola Kozmetikai Es Haztartasvegyipari Vallalat Magnesium salt of a fatty acid acyl lactylate
FR2631620B1 (fr) * 1988-05-19 1990-07-27 Rhone Poulenc Chimie Nouvelle silice precipitee absorbante et composition a base de cette s ilice
JPH04214801A (ja) * 1990-02-22 1992-08-05 Kawasaki Steel Corp 粉末冶金用金属造粒粉末及びそれを使用する焼結体の製造方法
IT1251937B (it) * 1991-10-17 1995-05-27 Donegani Guido Ist Xerogels di silice ad alta porosita` e processo per la loro preparazione.
CH687053A5 (fr) * 1993-10-05 1996-09-13 Crina Additifs pour l'alimentation animale et procédé pour leur préparation.
FR2776537B1 (fr) * 1998-03-30 2000-05-05 Rhodia Chimie Sa Composition comprenant un liquide absorbe sur un support a base de silice precipitee
US6303167B1 (en) * 1998-11-09 2001-10-16 Archer-Daniels-Midland Company Method of producing vitamin powders
JP2002012505A (ja) * 2000-04-28 2002-01-15 Daicel Chem Ind Ltd 固形化ギ酸、黴・細菌汚染防止飼料及びその製造方法
EP1551570A4 (en) * 2002-08-14 2008-04-09 Du Pont SOLID FLUID POWDER HAVING A HIGH LIQUID LOAD
EP1483975A1 (en) * 2003-06-05 2004-12-08 PURAC Biochem BV Antimicrobial composition comprising a mixture of lactic acid or a derivative thereof and an inorganic acid
KR101327700B1 (ko) * 2005-07-05 2013-11-11 론자 아게 건조 카르니틴 분말 또는 과립을 제조하는 분무-건조 방법
KR20080098586A (ko) * 2005-12-22 2008-11-11 바스프 에스이 비타민 e-흡착물의 제조 방법
CN100364551C (zh) * 2006-04-12 2008-01-30 浙江大学 负载型超细锌粉的补锌剂及制备方法和用途
FI20070521L (fi) * 2006-11-10 2008-05-11 Atacama Labs Oy Rakeita, tabletteja ja rakeistusmenetelmä
EP2082739A1 (en) * 2008-01-25 2009-07-29 PURAC Biochem BV Lactylates for the prevention and treatment of infections caused by gram-positive bacteria in animals
JP5890097B2 (ja) * 2008-02-08 2016-03-22 ピュラック バイオケム ビー. ブイ. 金属ラクテート粉及び製造方法
DE102008000290A1 (de) * 2008-02-13 2009-08-20 Evonik Degussa Gmbh Lagerstabile Produktsyteme für Prämixformulierungen
JP2009270130A (ja) * 2008-04-30 2009-11-19 Aida Kagaku Kogyo Kk 銀粉末または銀合金粉末、銀または銀合金の造形体の製造方法並びに銀または銀合金の造形体
EA201171282A1 (ru) * 2009-04-24 2012-05-30 Айсьютика Пти Лтд. Способ производства коммерческих порошков, содержащих нано- и микрочастицы
WO2011026796A1 (en) * 2009-09-01 2011-03-10 Basf Se Synergistic fungicidal mixtures comprising lactylates and method for combating phytopathogenic fungi
EP2335495A1 (en) * 2009-12-11 2011-06-22 Lonza Ltd. Carnitine granulate and methods for its production
CN101828584B (zh) * 2010-06-17 2012-06-27 郑州天地人面粉实业有限公司 速冻面点粉用改良剂、速冻面点粉和其制备方法
US8754054B2 (en) * 2010-07-09 2014-06-17 Albany Molecular Research, Inc. Antibacterial compounds, methods of making them, and uses thereof
CN101973744B (zh) * 2010-07-30 2011-10-26 许庆华 红色凹凸棒软陶粉
CN101973742B (zh) * 2010-07-30 2011-10-26 许庆华 蓝色凹凸棒软陶粉
CN101973737B (zh) * 2010-07-30 2011-10-26 许庆华 发光凹凸棒软陶粉
CN101973740B (zh) * 2010-07-30 2011-08-24 许庆华 黑色凹凸棒软陶粉
CN101973743B (zh) * 2010-07-30 2011-09-21 许庆华 黄色凹凸棒软陶粉

Also Published As

Publication number Publication date
CN103732077B (zh) 2016-08-17
EP2729015A2 (en) 2014-05-14
KR102196004B1 (ko) 2020-12-31
CN103732077A (zh) 2014-04-16
MX2014000321A (es) 2014-05-30
BR112014000428B1 (pt) 2019-09-17
JP6460791B2 (ja) 2019-01-30
MX357070B (es) 2018-06-22
CA2841149A1 (en) 2013-01-17
CA2841149C (en) 2019-11-05
US9849105B2 (en) 2017-12-26
RU2014102671A (ru) 2015-08-20
JP2014520518A (ja) 2014-08-25
US20180064675A1 (en) 2018-03-08
RU2603915C2 (ru) 2016-12-10
KR20140051936A (ko) 2014-05-02
WO2013007558A2 (en) 2013-01-17
US20140161864A1 (en) 2014-06-12
EP2729015B1 (en) 2019-01-02
WO2013007558A3 (en) 2013-04-04
PL2729015T3 (pl) 2019-07-31

Similar Documents

Publication Publication Date Title
BR112014000428A2 (pt) formulação ativa para uso em produtos de alimentação
BR112014020831B8 (pt) Composição de controle de peste incluindo derivado de iminopiridina, seu uso e método para pro-teger plantas úteis de pestes
AR082252A1 (es) Composiciones farmaceuticas moduladoras de c-met
AR089673A1 (es) Formulacion de premezcla de dexmedetomidina
CA2875877C (en) Syk inhibitors
PE20130217A1 (es) Composiciones farmaceuticas y metodos para su elaboracion
BR112012030416A2 (pt) composições pesticidas
BR112014032873A2 (pt) derivado de éster de ácido 2-aminonicotínico, e, bactericida
BR112014029754A2 (pt) soluções de tensoativos contendo n-metil-n-oleilglucaminas e n-metil-n-c12-c14-acilglucaminas
BR112013006936A2 (pt) composto de amida substituída
AR072261A1 (es) Derivados piperazin-pirazolicos, composiciones farmaceuticas que los contienen y usos de los mismos como agentes anticancerigenos.
MX361618B (es) Formulaciones farmacéuticas que comprenden derivados de nitrocatecol y métodos para hacer las mismas.
BR112015032340A2 (pt) composições e artigos para cuidados pessoais
BRPI0706125A2 (pt) molho instantÂneo para uso alimentÍcio, processo para o preparo do referido molho, bem como embalagem parcial ou completamente transparente
BR112015004185A2 (pt) composições antiperspirantes em aerossol, produtos e métodos
IN2014CN04665A (pt)
BR112012029913A8 (pt) levoisovalerilespiramicina i, ii ou iii, preparações, métodos de preparação e usos dos mesmos
TR201902435T4 (tr) DGAT1 inhibitör içeren farmasötik bileşimler.
BR112015026441A2 (pt) derivados de fulereno aperfeiçoados e materiais, métodos e dispositivos relacionados
BR112017004667A2 (pt) método para preparação de um composto, composto, uso de um composto, método para preparação de gêneros alimentícios, e, produto alimentar ou aditivo alimentar.
CL2011002186A1 (es) Composición pulverulenta que contiene 1 a 50% de un derivado de astaxantina, 10 a 70% de al menos un coloide de protección y eventualmente aditivos alimentarios; procedimiento de preparación de la composición; sus usos y procedimiento de preparación de comida animal.
BR112012028456A2 (pt) composições de aerossol
AR086045A1 (es) Componente de formulacion
AR079170A1 (es) Compuesto de ciclopropil-benzamida-imidazo-benzazepina inhibidor de diacil-glicerol aciltransferasa, sal del mismo, composicion farmaceutica que lo comprende, su uso para preparar un medicamento util para el tratamiento de obesidad o para mejorar la sensibilidad a insulina y compuesto intermedio par
PE20131327A1 (es) Forma cristalina delta de la sal de arginina de perindoprilo, su procedimiento de preparacion, y las composiciones farmaceuticas que la contienen

Legal Events

Date Code Title Description
B06T Formal requirements before examination
B15K Others concerning applications: alteration of classification

Ipc: A61K 31/23 (2006.01), A23K 20/105 (2016.01), A23K

B15K Others concerning applications: alteration of classification

Ipc: A23K 20/105 (2016.01), A23K 20/158 (2016.01), A23K

B07A Technical examination (opinion): publication of technical examination (opinion)
B09A Decision: intention to grant
B16A Patent or certificate of addition of invention granted

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 03/07/2012, OBSERVADAS AS CONDICOES LEGAIS. (CO) 20 (VINTE) ANOS CONTADOS A PARTIR DE 03/07/2012, OBSERVADAS AS CONDICOES LEGAIS