BR112012026456B1 - Process for the preparation of carboxylic pyrazole acid amides - Google Patents

Process for the preparation of carboxylic pyrazole acid amides Download PDF

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Publication number
BR112012026456B1
BR112012026456B1 BR112012026456-7A BR112012026456A BR112012026456B1 BR 112012026456 B1 BR112012026456 B1 BR 112012026456B1 BR 112012026456 A BR112012026456 A BR 112012026456A BR 112012026456 B1 BR112012026456 B1 BR 112012026456B1
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BR
Brazil
Prior art keywords
formula
compound
reacting
palladium
viii
Prior art date
Application number
BR112012026456-7A
Other languages
English (en)
Portuguese (pt)
Other versions
BR112012026456A2 (pt
Inventor
Schleth Florian
Vettiger Thomas
Rommel Michael
Tobler Hans
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of BR112012026456A2 publication Critical patent/BR112012026456A2/pt
Publication of BR112012026456B1 publication Critical patent/BR112012026456B1/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/263Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
    • C07C17/2635Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions involving a phosphorus compound, e.g. Wittig synthesis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/35Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction
    • C07C17/354Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction by hydrogenation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24Halogenated aromatic hydrocarbons with unsaturated side chains

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Catalysts (AREA)
BR112012026456-7A 2010-04-20 2011-04-14 Process for the preparation of carboxylic pyrazole acid amides BR112012026456B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10160439.5 2010-04-20
EP10160439 2010-04-20
PCT/EP2011/055870 WO2011131544A1 (en) 2010-04-20 2011-04-14 Process for the preparation of pyrazole carboxylic acid amides

Publications (2)

Publication Number Publication Date
BR112012026456A2 BR112012026456A2 (pt) 2015-09-08
BR112012026456B1 true BR112012026456B1 (pt) 2017-06-27

Family

ID=43984050

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012026456-7A BR112012026456B1 (pt) 2010-04-20 2011-04-14 Process for the preparation of carboxylic pyrazole acid amides

Country Status (13)

Country Link
US (1) US8524915B2 (https=)
EP (1) EP2560960B1 (https=)
JP (1) JP6153864B2 (https=)
CN (1) CN102858749B (https=)
AR (1) AR080923A1 (https=)
BR (1) BR112012026456B1 (https=)
ES (1) ES2458935T3 (https=)
IL (1) IL222400A (https=)
MX (1) MX2012012009A (https=)
PY (1) PY1115669A (https=)
TW (1) TWI480041B (https=)
UY (1) UY33341A (https=)
WO (1) WO2011131544A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
CN103483407B (zh) * 2013-10-10 2015-11-18 宁夏启元药业有限公司 一种硫氰酸红霉素萃取结晶用复合溶媒及萃取结晶方法
GB201403438D0 (en) * 2014-02-27 2014-04-16 Syngenta Participations Ag Polymorphs
CN105985254B (zh) * 2015-02-17 2018-03-16 上海中科绿碳化工科技有限公司 一种制备甲酰胺类化合物的方法
CN106588745B (zh) * 2016-12-02 2019-06-14 杭州百昂锐地科技有限公司 一种苯并烯氟菌唑的中间体及其制备方法和应用
KR20250036910A (ko) 2022-07-22 2025-03-14 신젠타 크롭 프로텍션 아게 이종환식 아미드 유도체의 고체 형태
PY2503719A (es) 2024-01-26 2025-08-05 Syngenta Crop Protection Ag Proceso químico

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 1―ブロモ―2―クロロ―4―フルオロベンゼンの製造法
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
US7732469B2 (en) * 2005-10-25 2010-06-08 Syngenta Crop Protection, Inc. Heterocyclic amide derivatives useful as microbiocides
IN2015DN00818A (https=) 2005-12-12 2015-07-10 Syngenta Participations Ag
CN101528034B (zh) 2006-10-25 2011-11-09 辛根塔有限公司 生产经取代的溴苯的方法
MX2010011790A (es) * 2008-05-14 2010-11-25 Syngenta Ltd Proceso para la preparacion de amidas.
BRPI0923527A2 (pt) * 2008-12-24 2016-08-09 Syngenta Ltd métodos de preparo de fungicidas
BR112012024705A2 (pt) * 2010-03-31 2016-06-07 Actelion Pharmaceuticals Ltd derivados antibacterianos de isoquinolin-3-ilureia
WO2011131546A1 (en) * 2010-04-20 2011-10-27 Syngenta Participations Ag Process for the preparation of pyrazole carboxylic acid amides
JP5684896B2 (ja) * 2010-04-20 2015-03-18 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト ピラゾールカルボン酸アミドの調製方法
JP5684895B2 (ja) * 2010-04-20 2015-03-18 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト ピラゾールカルボン酸アミドの調製方法

Also Published As

Publication number Publication date
US8524915B2 (en) 2013-09-03
AR080923A1 (es) 2012-05-16
PY1115669A (es) 2014-09-01
BR112012026456A2 (pt) 2015-09-08
US20130041160A1 (en) 2013-02-14
WO2011131544A1 (en) 2011-10-27
UY33341A (es) 2011-12-01
EP2560960A1 (en) 2013-02-27
EP2560960B1 (en) 2014-02-26
CN102858749A (zh) 2013-01-02
TWI480041B (zh) 2015-04-11
IL222400A (en) 2015-04-30
MX2012012009A (es) 2012-12-17
JP2013527840A (ja) 2013-07-04
ES2458935T3 (es) 2014-05-07
TW201210590A (en) 2012-03-16
CN102858749B (zh) 2014-07-02
JP6153864B2 (ja) 2017-06-28

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Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]
B24B Patent annual fee: requirement for complementing annual fee

Free format text: COMPLEMENTAR A RETRIBUICAO DA(S) 8A. ANUIDADE(S), DE ACORDO COM TABELA VIGENTE, REFERENTE A(S) GUIA(S) DE RECOLHIMENTO 0000921705515656.

B24E Patent annual fee: resolution cancelled
B25G Requested change of headquarter approved
B25A Requested transfer of rights approved