BR112012008128B8 - processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula || - Google Patents
processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula ||Info
- Publication number
- BR112012008128B8 BR112012008128B8 BR112012008128A BR112012008128A BR112012008128B8 BR 112012008128 B8 BR112012008128 B8 BR 112012008128B8 BR 112012008128 A BR112012008128 A BR 112012008128A BR 112012008128 A BR112012008128 A BR 112012008128A BR 112012008128 B8 BR112012008128 B8 BR 112012008128B8
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- formula
- preparation
- processes
- regioselective alkylation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23013409P | 2009-07-31 | 2009-07-31 | |
| US61/230,134 | 2009-07-31 | ||
| US36157010P | 2010-07-06 | 2010-07-06 | |
| PCT/EP2010/060884 WO2011012620A2 (en) | 2009-07-31 | 2010-07-27 | Processes for the alkylation of pyrazoles |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| BR112012008128A2 BR112012008128A2 (pt) | 2015-09-22 |
| BR112012008128B1 BR112012008128B1 (pt) | 2017-10-31 |
| BR112012008128B8 true BR112012008128B8 (pt) | 2019-07-16 |
Family
ID=42782270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012008128A BR112012008128B8 (pt) | 2009-07-31 | 2010-07-27 | processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula || |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8563747B2 (https=) |
| EP (1) | EP2459538B1 (https=) |
| JP (1) | JP5956334B2 (https=) |
| CN (1) | CN102471279A (https=) |
| AR (1) | AR077332A1 (https=) |
| BR (1) | BR112012008128B8 (https=) |
| DK (1) | DK2459538T3 (https=) |
| ES (1) | ES2525489T3 (https=) |
| IL (1) | IL217387A (https=) |
| MX (1) | MX2012001067A (https=) |
| TW (1) | TW201107296A (https=) |
| WO (1) | WO2011012620A2 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102471278B (zh) | 2009-07-28 | 2015-04-01 | 先正达参股股份有限公司 | 关于吡唑的烷基化方法 |
| JP5869570B2 (ja) * | 2010-08-10 | 2016-02-24 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | ３−ハロアルキルピラゾールの調製方法 |
| JP5140776B1 (ja) * | 2012-09-05 | 2013-02-13 | タマ化学工業株式会社 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| ES2750353T3 (es) | 2014-08-19 | 2020-03-25 | Bayer Animal Health Gmbh | Procedimiento de preparación de 5-fluoro-1H-pirazoles partiendo de hexafluoropropeno |
| WO2024014780A1 (ko) * | 2022-07-11 | 2024-01-18 | 주식회사 엘지에너지솔루션 | 리튬 이차전지용 비수 전해액 및 이를 포함하는 리튬 이차전지 |
| CN119823045B (zh) * | 2024-12-18 | 2025-10-17 | 湖南化工研究院有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的合成方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0759560B2 (ja) * | 1987-10-19 | 1995-06-28 | 三井東圧化学株式会社 | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| GB9405229D0 (en) * | 1994-03-17 | 1994-04-27 | Rhone Poulenc Agriculture | Compositions of matter |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| JP2000044541A (ja) | 1998-08-03 | 2000-02-15 | Mitsui Chemicals Inc | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| JP4568404B2 (ja) | 2000-05-17 | 2010-10-27 | 三井化学アグロ株式会社 | ピラゾールカルボン酸エステル誘導体の製造法 |
| MXPA04008314A (es) | 2002-03-05 | 2004-11-26 | Syngenta Participations Ag | O-ciclopropil-carboxaniluros y su uso como funguicidas. |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| US20080108686A1 (en) * | 2004-06-18 | 2008-05-08 | Basf Aktiengesellschaft | N-(Ortho-Phenyl)-1-Methyl-3-Difluoromethylpyrazole-4-Carboxanilides And Their Use As Fungicides |
| TWI357898B (en) | 2004-10-21 | 2012-02-11 | Syngenta Participations Ag | Process for the preparation of pyrazoles |
| US7863460B2 (en) * | 2005-02-25 | 2011-01-04 | Sagami Chemical Research Center | Process for producing 1-substituted-3-fluoroalkylpyrazole-4-carboxylate |
| US7732469B2 (en) * | 2005-10-25 | 2010-06-08 | Syngenta Crop Protection, Inc. | Heterocyclic amide derivatives useful as microbiocides |
| GB0526044D0 (en) * | 2005-12-21 | 2006-02-01 | Syngenta Ltd | Novel herbicides |
| WO2008053044A2 (de) | 2006-11-03 | 2008-05-08 | Basf Se | Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen |
| BRPI0808927B1 (pt) | 2007-03-16 | 2023-09-26 | Syngenta Participations Ag | Modificação c cristalográfica (9-isopropil-1,2,3,4- tetra-hidro-1,4- metano-naftalen-5-il)-amida racêmica syn do ácido 3-difluorometil-1-metil-1hpirazol-4- carboxílico e composição a compreendendo, bem como método para controlar doenças em plantas úteis ou no material de propagação das mesmas, causadas por agentes fitopatogênicos |
| JP5210375B2 (ja) * | 2007-05-11 | 2013-06-12 | イーライ リリー アンド カンパニー | ５−ｈｔ７受容体拮抗薬としての２−［４−（ピラゾール−４−イルアルキル）ピペラジン−１−イル］−３−フェニルピラジンおよびピリジンならびに３−［４−（ピラゾール−４−イルアルキル）ピペラジン−１−イル］−２−フェニルピリジン |
| KR20100017431A (ko) | 2007-05-31 | 2010-02-16 | 신젠타 파티서페이션즈 아게 | 피라졸의 제조 방법 |
| WO2009135860A1 (de) | 2008-05-08 | 2009-11-12 | Basf Se | Verfahren zur herstellung von arylcarboxamiden |
| GB0812028D0 (en) | 2008-07-01 | 2008-08-06 | Syngenta Participations Ag | Fungicidal compositions |
-
2010
- 2010-07-27 MX MX2012001067A patent/MX2012001067A/es not_active Application Discontinuation
- 2010-07-27 TW TW099124617A patent/TW201107296A/zh unknown
- 2010-07-27 ES ES10736729.4T patent/ES2525489T3/es active Active
- 2010-07-27 EP EP10736729.4A patent/EP2459538B1/en active Active
- 2010-07-27 JP JP2012522152A patent/JP5956334B2/ja active Active
- 2010-07-27 BR BR112012008128A patent/BR112012008128B8/pt active IP Right Grant
- 2010-07-27 WO PCT/EP2010/060884 patent/WO2011012620A2/en not_active Ceased
- 2010-07-27 DK DK10736729.4T patent/DK2459538T3/en active
- 2010-07-27 AR ARP100102714A patent/AR077332A1/es unknown
- 2010-07-27 CN CN2010800339701A patent/CN102471279A/zh active Pending
- 2010-07-27 US US13/388,246 patent/US8563747B2/en active Active
-
2012
- 2012-01-05 IL IL217387A patent/IL217387A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| IL217387A0 (en) | 2012-02-29 |
| EP2459538B1 (en) | 2014-10-15 |
| US8563747B2 (en) | 2013-10-22 |
| MX2012001067A (es) | 2012-03-16 |
| CN102471279A (zh) | 2012-05-23 |
| DK2459538T3 (en) | 2015-01-05 |
| BR112012008128B1 (pt) | 2017-10-31 |
| WO2011012620A3 (en) | 2011-06-09 |
| TW201107296A (en) | 2011-03-01 |
| IL217387A (en) | 2016-02-29 |
| BR112012008128A2 (pt) | 2015-09-22 |
| ES2525489T3 (es) | 2014-12-23 |
| EP2459538A2 (en) | 2012-06-06 |
| JP2013500945A (ja) | 2013-01-10 |
| JP5956334B2 (ja) | 2016-07-27 |
| WO2011012620A2 (en) | 2011-02-03 |
| AR077332A1 (es) | 2011-08-17 |
| US20120130085A1 (en) | 2012-05-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] | ||
| B16C | Correction of notification of the grant [chapter 16.3 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 27/07/2010, OBSERVADAS AS CONDICOES LEGAIS. (CO) REF. 2443 DE 31/10/2017 QUANTO AO ITEM (30) PRIORIDADE UNIONISTA. |
|
| B25G | Requested change of headquarter approved | ||
| B25A | Requested transfer of rights approved |