BR112012008128B8 - processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula || - Google Patents
processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula ||Info
- Publication number
- BR112012008128B8 BR112012008128B8 BR112012008128A BR112012008128A BR112012008128B8 BR 112012008128 B8 BR112012008128 B8 BR 112012008128B8 BR 112012008128 A BR112012008128 A BR 112012008128A BR 112012008128 A BR112012008128 A BR 112012008128A BR 112012008128 B8 BR112012008128 B8 BR 112012008128B8
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- formula
- preparation
- processes
- regioselective alkylation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23013409P | 2009-07-31 | 2009-07-31 | |
| US36157010P | 2010-07-06 | 2010-07-06 | |
| US61/230,134 | 2010-07-06 | ||
| PCT/EP2010/060884 WO2011012620A2 (en) | 2009-07-31 | 2010-07-27 | Processes for the alkylation of pyrazoles |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| BR112012008128A2 BR112012008128A2 (pt) | 2015-09-22 |
| BR112012008128B1 BR112012008128B1 (pt) | 2017-10-31 |
| BR112012008128B8 true BR112012008128B8 (pt) | 2019-07-16 |
Family
ID=42782270
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012008128A BR112012008128B8 (pt) | 2009-07-31 | 2010-07-27 | processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula || |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8563747B2 (https=) |
| EP (1) | EP2459538B1 (https=) |
| JP (1) | JP5956334B2 (https=) |
| CN (1) | CN102471279A (https=) |
| AR (1) | AR077332A1 (https=) |
| BR (1) | BR112012008128B8 (https=) |
| DK (1) | DK2459538T3 (https=) |
| ES (1) | ES2525489T3 (https=) |
| IL (1) | IL217387A (https=) |
| MX (1) | MX2012001067A (https=) |
| TW (1) | TW201107296A (https=) |
| WO (1) | WO2011012620A2 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2602003T3 (es) | 2009-07-28 | 2017-02-17 | Syngenta Participations Ag | Procedimientos relacionados con la alquilación de pirazoles |
| PT2603494T (pt) * | 2010-08-10 | 2017-02-03 | Syngenta Participations Ag | Processo para a preparação de 3-haloalquilopirazóis |
| JP5140776B1 (ja) * | 2012-09-05 | 2013-02-13 | タマ化学工業株式会社 | １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 |
| ES2750353T3 (es) * | 2014-08-19 | 2020-03-25 | Bayer Animal Health Gmbh | Procedimiento de preparación de 5-fluoro-1H-pirazoles partiendo de hexafluoropropeno |
| WO2024014780A1 (ko) * | 2022-07-11 | 2024-01-18 | 주식회사 엘지에너지솔루션 | 리튬 이차전지용 비수 전해액 및 이를 포함하는 리튬 이차전지 |
| CN119823045B (zh) * | 2024-12-18 | 2025-10-17 | 湖南化工研究院有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-甲酸乙酯的合成方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0759560B2 (ja) * | 1987-10-19 | 1995-06-28 | 三井東圧化学株式会社 | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| GB9405229D0 (en) | 1994-03-17 | 1994-04-27 | Rhone Poulenc Agriculture | Compositions of matter |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| JP2000044541A (ja) * | 1998-08-03 | 2000-02-15 | Mitsui Chemicals Inc | １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法 |
| JP4568404B2 (ja) | 2000-05-17 | 2010-10-27 | 三井化学アグロ株式会社 | ピラゾールカルボン酸エステル誘導体の製造法 |
| KR100818540B1 (ko) | 2002-03-05 | 2008-04-01 | 신젠타 파티서페이션즈 아게 | Ｏ-사이클로프로필-카복스아닐리드 및 이를 포함하는 살진균 조성물 |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| US20080108686A1 (en) * | 2004-06-18 | 2008-05-08 | Basf Aktiengesellschaft | N-(Ortho-Phenyl)-1-Methyl-3-Difluoromethylpyrazole-4-Carboxanilides And Their Use As Fungicides |
| EA010851B1 (ru) * | 2004-10-21 | 2008-12-30 | Зингента Партисипейшнс Аг | Способ получения пиразолов |
| CN101133031B (zh) * | 2005-02-25 | 2010-07-21 | 财团法人相模中央化学研究所 | 1-取代-3-氟代烷基吡唑-4-羧酸酯的制造方法 |
| EA014297B1 (ru) * | 2005-10-25 | 2010-10-29 | Зингента Партисипейшнс Аг | Гетероциклические амиды, применимые в качестве микробиоцидов |
| GB0526044D0 (en) | 2005-12-21 | 2006-02-01 | Syngenta Ltd | Novel herbicides |
| WO2008053044A2 (de) * | 2006-11-03 | 2008-05-08 | Basf Se | Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen |
| CA2679408C (en) | 2007-03-16 | 2016-05-03 | Syngenta Limited | Novel solid forms of a microbiocide |
| ES2395872T3 (es) | 2007-05-11 | 2013-02-15 | Eli Lilly And Company | 2-[4-(Pirazol-4-ilalquil)piperazin-1-il]-3-fenil pirazinas y piridinas y 3-[4-(pirazol-4-ilalquil)piperazin-1-il]-2-fenil piridinas como antagonistas del receptor de 5-HT7 |
| US8124787B2 (en) | 2007-05-31 | 2012-02-28 | Syngenta Crop Protection, Inc. | Process for the production of pyrazoles |
| BRPI0912383A2 (pt) | 2008-05-08 | 2015-07-28 | Basf Se | Processo para preparar aril carboxamidas |
| GB0812028D0 (en) | 2008-07-01 | 2008-08-06 | Syngenta Participations Ag | Fungicidal compositions |
-
2010
- 2010-07-27 US US13/388,246 patent/US8563747B2/en active Active
- 2010-07-27 DK DK10736729.4T patent/DK2459538T3/en active
- 2010-07-27 BR BR112012008128A patent/BR112012008128B8/pt active IP Right Grant
- 2010-07-27 AR ARP100102714A patent/AR077332A1/es unknown
- 2010-07-27 ES ES10736729.4T patent/ES2525489T3/es active Active
- 2010-07-27 MX MX2012001067A patent/MX2012001067A/es not_active Application Discontinuation
- 2010-07-27 TW TW099124617A patent/TW201107296A/zh unknown
- 2010-07-27 CN CN2010800339701A patent/CN102471279A/zh active Pending
- 2010-07-27 EP EP10736729.4A patent/EP2459538B1/en active Active
- 2010-07-27 JP JP2012522152A patent/JP5956334B2/ja active Active
- 2010-07-27 WO PCT/EP2010/060884 patent/WO2011012620A2/en not_active Ceased
-
2012
- 2012-01-05 IL IL217387A patent/IL217387A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011012620A2 (en) | 2011-02-03 |
| IL217387A (en) | 2016-02-29 |
| JP2013500945A (ja) | 2013-01-10 |
| IL217387A0 (en) | 2012-02-29 |
| US8563747B2 (en) | 2013-10-22 |
| CN102471279A (zh) | 2012-05-23 |
| MX2012001067A (es) | 2012-03-16 |
| AR077332A1 (es) | 2011-08-17 |
| EP2459538B1 (en) | 2014-10-15 |
| BR112012008128A2 (pt) | 2015-09-22 |
| US20120130085A1 (en) | 2012-05-24 |
| TW201107296A (en) | 2011-03-01 |
| EP2459538A2 (en) | 2012-06-06 |
| DK2459538T3 (en) | 2015-01-05 |
| ES2525489T3 (es) | 2014-12-23 |
| JP5956334B2 (ja) | 2016-07-27 |
| WO2011012620A3 (en) | 2011-06-09 |
| BR112012008128B1 (pt) | 2017-10-31 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BR112012007085B8 (pt) | processos para a preparação de derivados de benzil-benzeno substituídos com glicopiranosila | |
| BR112012008128B8 (pt) | processos para a preparação de um composto da fórmula | e processo para a alquilação regiosseletiva de um composto da fórmula || | |
| MA34644B1 (fr) | Dérivés de pyrazole aminopyrimidine en tant que modulateurs du lrrk2 | |
| BRPI0813284A8 (pt) | Processo para a preparação de um composto da fórmula (i) e composto | |
| BR112013006720A2 (pt) | processo para preparação de inibidores de pan-cdk da fórmula (i) e intermediários da preparação | |
| BR112012021556A2 (pt) | processo para a preparação de peptídeos prolila substituídos e peptidomiméticos similares | |
| BR122017022221B8 (pt) | Processo para preparação de 2-amino-5,8-alcóxi[1,2,4]triazol[l,5-c]pirimidinas | |
| BR112014000471A2 (pt) | processo para preparo de derivados de diamida de ácido antranílico substituídos com tetrazol por meio da reação de ácidos pirazóis com ésteres antranílicos | |
| CO6410257A2 (es) | Herbicidas novedosos | |
| BR122018074319B8 (pt) | Método para preparar um composto de fórmula 14 | |
| BR112014004210A2 (pt) | processo para a preparação de derivados de diamida do ácido antranílico substituídos com tetrazole por reação de benzoxazinonas com aminas | |
| BRPI1014802B8 (pt) | profármacos de triptolida. | |
| BR112014031616A2 (pt) | compostos de fenoxietil piperidina | |
| BR112013028486A2 (pt) | método para promover crescimento de planta | |
| BRPI0803636A2 (pt) | processo para a sìntese de ranelato de estrÈncio e seus hidratos | |
| CO6480992A2 (es) | Derivados de pirazoles, su preparacion y su aplicacion terapeutica | |
| BR112014026198A2 (pt) | compostos pirazol como inibidores de sglt1 | |
| BR112014009266A2 (pt) | processo para a preparação de ácidos isoxazolil-metóxi-nicotínicos | |
| SG194727A1 (en) | Method for modification of organic molecules | |
| BR112014015430A8 (pt) | formulação oftálmica | |
| BR112013028789A2 (pt) | processo | |
| BR112013027395A2 (pt) | inibidores de 17alfa-hidroxilase/c17,20-liase | |
| BR112012009611A2 (pt) | ''processo para a preparação de um composto de fómula (i)'' | |
| BRPI0808570B8 (pt) | processo para a preparação de inibidores de glyt-1 | |
| BR102012013573A2 (pt) | processo de sÍntese, e forma cristalina de cloridrato de 4-{3-[cis-hexa-hidrociclopenta[c]pirrol-2(1h)-il]propà xi}benzamida e composiÇÕes farmacÊuticas contendo o mesmo |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] | ||
| B16C | Correction of notification of the grant [chapter 16.3 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 27/07/2010, OBSERVADAS AS CONDICOES LEGAIS. (CO) REF. 2443 DE 31/10/2017 QUANTO AO ITEM (30) PRIORIDADE UNIONISTA. |
|
| B25G | Requested change of headquarter approved | ||
| B25A | Requested transfer of rights approved |