BR0308857A - Composições farmacêuticas contendo promedicamentos de propofol, solúveis em água, e métodos de administrar os mesmos - Google Patents

Composições farmacêuticas contendo promedicamentos de propofol, solúveis em água, e métodos de administrar os mesmos

Info

Publication number
BR0308857A
BR0308857A BR0308857-0A BR0308857A BR0308857A BR 0308857 A BR0308857 A BR 0308857A BR 0308857 A BR0308857 A BR 0308857A BR 0308857 A BR0308857 A BR 0308857A
Authority
BR
Brazil
Prior art keywords
methods
pharmaceutical compositions
compositions containing
soluble
administering
Prior art date
Application number
BR0308857-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Peggy Wingard
Eric S Burak
Ekaterina Gibianski
James J Vornov
Original Assignee
Guilford Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29254399&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0308857(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Guilford Pharm Inc filed Critical Guilford Pharm Inc
Publication of BR0308857A publication Critical patent/BR0308857A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A61P39/06—Free radical scavengers or antioxidants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Otolaryngology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Pulmonology (AREA)
  • Anesthesiology (AREA)
  • Dermatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR0308857-0A 2002-04-08 2003-04-08 Composições farmacêuticas contendo promedicamentos de propofol, solúveis em água, e métodos de administrar os mesmos BR0308857A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US37024502P 2002-04-08 2002-04-08
US37021302P 2002-04-08 2002-04-08
PCT/US2003/010540 WO2003086413A1 (en) 2002-04-08 2003-04-08 Pharmaceutical compositions containing water-soluble prodrugs of propofol and methods of administering same

Publications (1)

Publication Number Publication Date
BR0308857A true BR0308857A (pt) 2005-01-04

Family

ID=29254399

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0308857-0A BR0308857A (pt) 2002-04-08 2003-04-08 Composições farmacêuticas contendo promedicamentos de propofol, solúveis em água, e métodos de administrar os mesmos

Country Status (17)

Country Link
US (1) US20050203068A1 (ko)
EP (2) EP2281565A3 (ko)
JP (2) JP5188003B2 (ko)
KR (2) KR20070087004A (ko)
CN (1) CN1649597A (ko)
AU (2) AU2003224851B2 (ko)
BR (1) BR0308857A (ko)
CA (1) CA2480881C (ko)
HU (1) HUP0600241A2 (ko)
IL (2) IL164217A0 (ko)
MX (1) MXPA04009703A (ko)
NO (1) NO20044152L (ko)
NZ (1) NZ535484A (ko)
PL (1) PL373850A1 (ko)
RU (1) RU2297216C2 (ko)
WO (1) WO2003086413A1 (ko)
ZA (1) ZA200407804B (ko)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1569912E (pt) 2002-12-03 2015-09-15 Pharmacyclics Llc Derivados 2-(2-hidroxibifenil-3-il)-1h-benzoimidazole-5- carboxamidina como inibidores do fator viia
US8729117B2 (en) 2004-06-02 2014-05-20 Pharmacyclics, Inc. Factor VIIa inhibitor
EP1791521A4 (en) * 2004-09-17 2009-10-21 Eisai Corp North America METHODS OF ADMINISTERING PROPOFOL PROMOTERS WITH WATER SOLUBLE
US20090221532A1 (en) * 2005-07-12 2009-09-03 Mgi Gp, Inc. Methods Of Dosing Propofol Prodrugs For Inducing Mild To Moderate Levels Of Sedation
WO2007131070A2 (en) * 2006-05-04 2007-11-15 Xenoport, Inc. Compositions, dosage forms and methods of treating emesis
KR100755872B1 (ko) * 2006-10-02 2007-09-05 충남대학교산학협력단 미다졸람을 함유하는 염증 예방 및 치료용 약제학적 조성물
KR20090059136A (ko) * 2006-10-05 2009-06-10 에이자이 코포레이션 오브 노쓰아메리카 프로포폴의 수용성 프로드럭의 수성 약제학적 제제
US20080161400A1 (en) * 2006-10-26 2008-07-03 Xenoport, Inc. Use of forms of propofol for treating diseases associated with oxidative stress
BRPI0811284A2 (pt) 2007-05-09 2015-01-20 Pharmacofore Inc Compostos terapêuticos
US8071818B2 (en) 2007-05-09 2011-12-06 Pharmacofore, Inc. Therapeutic compounds
US20090005444A1 (en) * 2007-06-21 2009-01-01 Xenoport, Inc. Use of propofol prodrugs for treating alcohol withdrawal, central pain, anxiety or pruritus
WO2009036322A1 (en) * 2007-09-14 2009-03-19 Xenoport, Inc. Use of propofol prodrugs for treating neuropathic pain
CA2702970A1 (en) 2007-10-16 2009-04-23 Pharmacyclics, Inc. Manufacture, compositions and uses of coagulation factor viia modulator
UY34072A (es) 2011-05-17 2013-01-03 Novartis Ag Derivados sustituidos de indol
CN102397246A (zh) * 2011-11-18 2012-04-04 陕西合成药业有限公司 一种注射用磷丙泊酚钠及其制备方法和用途
CN103172658B (zh) * 2011-12-26 2016-01-20 宜昌人福药业有限责任公司 一种适合药用的前体药物晶型、制备方法及药用组合物
CN102552291A (zh) * 2012-01-04 2012-07-11 陕西合成药业有限公司 一种磷丙泊酚钠静脉给药制剂及其制备方法和用途
RU2535001C1 (ru) * 2013-07-11 2014-12-10 Общество с ограниченной ответственностью "ВИК-здоровье животных" Микроколлоидный раствор пропофола для анестезии
JP2018523705A (ja) * 2015-07-28 2018-08-23 ベータ・キャット・ファーマシューティカルズ・インコーポレイテッド アントラセン−９，１０−ジオンジオキシム化合物プロドラッグ及びその使用
US9585867B2 (en) * 2015-08-06 2017-03-07 Charles Everett Ankner Cannabinod formulation for the sedation of a human or animal
US11439653B1 (en) 2021-03-30 2022-09-13 Epalex Corporation Fospropofol formulations
US11478490B1 (en) 2021-03-30 2022-10-25 Epalex Corporation Fospropofol formulations
US11628178B2 (en) 2019-03-26 2023-04-18 Epalex Corporation Fospropofol methods and compositions
US11547714B2 (en) 2020-02-05 2023-01-10 Epalex Corporation Fospropofol salts, methods and compositions
CN111135304A (zh) * 2020-01-19 2020-05-12 李启芳 治疗慢性、顽固性或原发性失眠症的联合用药物及其应用

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2829151A (en) * 1952-11-03 1958-04-01 Dow Chemical Co Chlorotoloxy-ethyl phosphates
US3271314A (en) * 1958-12-04 1966-09-06 Ethyl Corp 2, 6-diisopropylphenol
GB1146173A (en) * 1966-06-18 1969-03-19 Geigy Uk Ltd Production of triaryl phosphates
US3723578A (en) * 1970-10-13 1973-03-27 Gaf Corp Phosphate esters of ethers of thiol substituted phenols
US4171272A (en) * 1977-12-02 1979-10-16 Fmc Corporation Turbine lubricant
FR2601259B1 (fr) * 1986-07-11 1990-06-22 Rhone Poulenc Chimie Nouvelles compositions tensio-actives a base d'esters phosphoriques leur procede de preparation et leur application a la formulation de matieres actives.
MY103951A (en) * 1988-01-12 1993-10-30 Kao Corp Detergent composition
FR2638168A1 (fr) * 1988-10-21 1990-04-27 Rhone Poulenc Chimie Dispersions d'halogenures de terres rares en milieu huileux
DE3900941A1 (de) * 1989-01-14 1990-07-19 Henkel Kgaa Verfahren zur flotation von fuellstoffen aus altpapieren in gegenwart organischer phosphorsaeureester
CA2014539C (en) * 1989-04-17 2000-07-25 Shinichiro Umeda Water borne metallic coating composition
US5091211A (en) * 1989-08-17 1992-02-25 Lord Corporation Coating method utilizing phosphoric acid esters
US5110503A (en) * 1990-05-15 1992-05-05 Elliot Cohen Demulsifying
JP2869186B2 (ja) * 1990-10-17 1999-03-10 株式会社トーメン 植物における生物活性剤の吸収移行を促進する方法及び組成物
US5646176A (en) * 1992-12-24 1997-07-08 Bristol-Myers Squibb Company Phosphonooxymethyl ethers of taxane derivatives
US5731355A (en) * 1994-03-22 1998-03-24 Zeneca Limited Pharmaceutical compositions of propofol and edetate
GB9405593D0 (en) * 1994-03-22 1994-05-11 Zeneca Ltd Pharmaceutical compositions
IT1270093B (it) * 1994-09-28 1997-04-28 Zambon Spa Processo per la purificazione di 2,6-diisopropilfenolo
US5804682A (en) * 1995-11-29 1998-09-08 Henkel Corporation Aqueous dispersions of polyamides
US5637625A (en) * 1996-03-19 1997-06-10 Research Triangle Pharmaceuticals Ltd. Propofol microdroplet formulations
US5723538A (en) * 1996-06-14 1998-03-03 Henkel Corporation Aqueous dispersions of polyamides
US5746973A (en) * 1996-07-10 1998-05-05 Naraghi; Ali Method for reducing odorant depletion
PT1052975E (pt) * 1998-02-10 2007-10-29 Sicor Inc Composição de propofol que contém sulfito
AR015744A1 (es) * 1998-04-01 2001-05-16 Orion Corp Uso de dexmedetomidina para sedacion en terapia intensiva
US6254853B1 (en) * 1998-05-08 2001-07-03 Vyrex Corporation Water soluble pro-drugs of propofol
MXPA00011835A (es) * 1998-06-03 2002-10-17 Scott Lab Inc Aparato y metodo para proveer alivio del dolor de un paciente consciente y ansiedad asociada con procedimientos medicos o quirurgicos.
US6204257B1 (en) * 1998-08-07 2001-03-20 Universtiy Of Kansas Water soluble prodrugs of hindered alcohols
DK1105096T3 (da) * 1998-08-19 2004-03-08 Skyepharma Canada Inc Injicerbare vandige propofoldispersioner
EP1161226B1 (en) * 1999-02-18 2004-05-26 SuperGen, Inc. Phosphocholine linked prodrug derivatives
AU3898700A (en) * 1999-03-15 2000-10-04 John Claude Krusz Treatment of acute headaches and chronic pain using rapidly-cleared anesthetic drug at sub-anesthetic dosages
GB2359747B (en) * 2000-02-29 2002-04-24 Maelor Pharmaceuticals Ltd Anaesthetic formulations
SE0001865D0 (sv) * 2000-05-19 2000-05-19 Astrazeneca Ab Management of septic shock
WO2001097779A2 (en) * 2000-06-16 2001-12-27 Rtp Pharma Inc. Improved injectable dispersions of propofol
US6362234B1 (en) * 2000-08-15 2002-03-26 Vyrex Corporation Water-soluble prodrugs of propofol for treatment of migrane

Also Published As

Publication number Publication date
NZ535484A (en) 2009-01-31
EP2281565A3 (en) 2011-10-26
CN1649597A (zh) 2005-08-03
PL373850A1 (en) 2005-09-19
CA2480881A1 (en) 2003-10-23
KR20070087004A (ko) 2007-08-27
AU2003224851A1 (en) 2003-10-27
JP5188003B2 (ja) 2013-04-24
EP1492544A4 (en) 2005-10-12
AU2008202880A1 (en) 2008-07-24
NO20044152L (no) 2005-01-07
IL164217A0 (en) 2005-12-18
JP2010195803A (ja) 2010-09-09
US20050203068A1 (en) 2005-09-15
MXPA04009703A (es) 2004-12-13
WO2003086413A1 (en) 2003-10-23
KR20040095352A (ko) 2004-11-12
AU2003224851B2 (en) 2008-04-03
EP1492544A1 (en) 2005-01-05
EP2281565A2 (en) 2011-02-09
IL164217A (en) 2013-02-28
RU2297216C2 (ru) 2007-04-20
ZA200407804B (en) 2005-11-30
JP2005526108A (ja) 2005-09-02
RU2004129339A (ru) 2005-05-27
HUP0600241A2 (en) 2006-07-28
CA2480881C (en) 2012-09-11

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved

Owner name: MGI GP INC. (US)

Free format text: ALTERADO DE: GUILFORD PHARMACEUTICALS INC.

B25G Requested change of headquarter approved

Owner name: MGI GP INC. (US)

Free format text: SEDE ALTERADA CONFORME SOLICITADO NA PETICAO NO 020060149192/RJ DE 27/09/2006.

B25A Requested transfer of rights approved

Owner name: EISAI CORPORATION OF NORTH AMERICA (US)

Free format text: TRANSFERIDO DE: MGI GP, INC.

B25A Requested transfer of rights approved

Owner name: EISAI INC. (US)

Free format text: TRANSFERIDO DE: EISAI CORPORATION OF NORTH AMERICA

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: PARA.INT.CI. A61K 31/66, A61P 23/00, A61P 25/20

Ipc: A61K 31/66 (2011.01), A61P 23/00 (2011.01), A61P 2

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07F Notification of approval that there is no relation to art. 229 of lpi (pipeline patents) [chapter 7.6 patent gazette]

Free format text: NOTIFICACAO DE NAO ANUENCIA RELACIONADA COM O ART. 229 DA LPI

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 12A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2307 DE 24/03/2015.