BR0307352A - Processos para a preparação de um composto e para a preparação de propionato de fluticasona, composto, e, processo para a preparação de um sal de imidazol do composto - Google Patents

Processos para a preparação de um composto e para a preparação de propionato de fluticasona, composto, e, processo para a preparação de um sal de imidazol do composto

Info

Publication number
BR0307352A
BR0307352A BR0307352-1A BR0307352A BR0307352A BR 0307352 A BR0307352 A BR 0307352A BR 0307352 A BR0307352 A BR 0307352A BR 0307352 A BR0307352 A BR 0307352A
Authority
BR
Brazil
Prior art keywords
compound
preparation
processes
fluticasone propionate
imidazole salt
Prior art date
Application number
BR0307352-1A
Other languages
English (en)
Inventor
Steven John Coote
Rosalyn Kay Nice
Mark David Wipperman
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of BR0307352A publication Critical patent/BR0307352A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"PROCESSOS PARA A PREPARAçãO DE UM COMPOSTO E PARA A PREPARAçãO DE PROPIONATO DE FLUTICASONA, COMPOSTO, E, PROCESSO PARA A PREPARAçãO DE UM SAL DE IMIDAZOL DO COMPOSTO". é descrito um processo para a preparação de um composto de fórmula (II) ou um sal deste.
BR0307352-1A 2002-02-04 2003-02-03 Processos para a preparação de um composto e para a preparação de propionato de fluticasona, composto, e, processo para a preparação de um sal de imidazol do composto BR0307352A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0202563.3A GB0202563D0 (en) 2002-02-04 2002-02-04 Process
PCT/EP2003/001116 WO2003066654A1 (en) 2002-02-04 2003-02-03 Process for the production of 6.alpha.,9.alpha-difluoro-17.alpha.-(1-oxopropoxy-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4-diene-17.beta.-carbothioic acid

Publications (1)

Publication Number Publication Date
BR0307352A true BR0307352A (pt) 2004-12-14

Family

ID=9930365

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0307352-1A BR0307352A (pt) 2002-02-04 2003-02-03 Processos para a preparação de um composto e para a preparação de propionato de fluticasona, composto, e, processo para a preparação de um sal de imidazol do composto

Country Status (22)

Country Link
US (1) US20050080065A1 (pt)
EP (1) EP1472271A1 (pt)
JP (1) JP2005521680A (pt)
KR (1) KR20040088050A (pt)
CN (1) CN1628125A (pt)
AR (1) AR038389A1 (pt)
AU (1) AU2003206837B2 (pt)
BR (1) BR0307352A (pt)
CA (1) CA2473753A1 (pt)
CO (1) CO5611116A2 (pt)
GB (1) GB0202563D0 (pt)
IL (1) IL162919A0 (pt)
IS (1) IS7350A (pt)
MX (1) MXPA04007529A (pt)
MY (1) MY140446A (pt)
NO (1) NO20043665L (pt)
NZ (1) NZ534044A (pt)
PL (1) PL372217A1 (pt)
RU (1) RU2333217C2 (pt)
TW (1) TW200307689A (pt)
WO (1) WO2003066654A1 (pt)
ZA (1) ZA200405515B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL153462A0 (en) * 2002-12-16 2003-07-06 Chemagis Ltd Thiocarboxylic acid organic salts and processes utilizing the same
PT103202B (pt) * 2004-10-19 2011-01-27 Hovione Farmaciencia S A Processo para a esterificação de um ácido carbotiótico
CN100560598C (zh) * 2005-07-26 2009-11-18 上海奥锐特国际贸易有限公司 氟替卡松丙酸酯的合成方法
NO331891B1 (no) 2007-03-20 2012-04-30 Clavis Pharma Asa Kjemiske forbindelser, et farmasoytisk preparat inneholdende slike forbindelser, samt anvendelse derav for behandling av kreft, inflammasjon og KOLS
US9303060B1 (en) * 2014-10-03 2016-04-05 Amphaster Pharmaceuticals, Inc. Methods of preparing intermediate of fluticasone propionate

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2852505A (en) * 1955-10-31 1958-09-16 American Cyanamid Co Aminodeoxyglycosidopurines
US3288781A (en) * 1964-12-18 1966-11-29 Upjohn Co Process for deacylating anhydro-lyxofuranosyl with nitrogen base
US4500711A (en) * 1977-03-21 1985-02-19 Burroughs Wellcome Co. Synthesis of leucovorin
JPS56138200A (en) * 1980-02-15 1981-10-28 Glaxo Group Ltd Androstane carbothioate compound
EP1059283B1 (en) * 1999-06-11 2003-05-28 F. Hoffmann-La Roche Ag Process for preparing neuraminidase inhibitor ro-64-0796

Also Published As

Publication number Publication date
AR038389A1 (es) 2005-01-12
CO5611116A2 (es) 2006-02-28
IL162919A0 (en) 2005-11-20
GB0202563D0 (en) 2002-03-20
AU2003206837B2 (en) 2008-11-13
NZ534044A (en) 2006-10-27
WO2003066654A1 (en) 2003-08-14
PL372217A1 (en) 2005-07-11
MXPA04007529A (es) 2004-11-10
RU2333217C2 (ru) 2008-09-10
RU2004121675A (ru) 2005-05-27
NO20043665L (no) 2004-09-01
ZA200405515B (en) 2005-07-12
CA2473753A1 (en) 2003-08-14
IS7350A (is) 2004-07-09
JP2005521680A (ja) 2005-07-21
MY140446A (en) 2009-12-31
CN1628125A (zh) 2005-06-15
US20050080065A1 (en) 2005-04-14
KR20040088050A (ko) 2004-10-15
EP1472271A1 (en) 2004-11-03
AU2003206837A1 (en) 2003-09-02
TW200307689A (en) 2003-12-16

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A(S) 8A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2112 DE 28/06/2011.