BR0208885A - Inibidores de integrina alfavbeta6 - Google Patents

Inibidores de integrina alfavbeta6

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Publication number
BR0208885A
BR0208885A BR0208885-1A BR0208885A BR0208885A BR 0208885 A BR0208885 A BR 0208885A BR 0208885 A BR0208885 A BR 0208885A BR 0208885 A BR0208885 A BR 0208885A
Authority
BR
Brazil
Prior art keywords
alphabeta6
novel
integrin inhibitors
integrin
inhibitors
Prior art date
Application number
BR0208885-1A
Other languages
English (en)
Inventor
Oliver Schadt
Alfred Jonczyk
Wolfgang Staehle
Simon Goodman
Original Assignee
Merck Patent Ges Mit Beschroen
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Ges Mit Beschroen filed Critical Merck Patent Ges Mit Beschroen
Publication of BR0208885A publication Critical patent/BR0208885A/pt

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    • C07C275/20Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an unsaturated carbon skeleton
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Abstract

"INIBIDORES DE INTEGRINA ALFA~ v~BETA~ 6~". A presente invenção refere-se a derivados de bifenila novos da fórmula geral 1 na qual R^ 1^, R^ 1<39>^, R^ 1"^, R^ 2^ e n são como definido na Reivindicação 1, seus estereoisómeros e seus sais ou solvatos fisiologicamente aceitáveis são novos ligandos de integrina, em particular do receptor de integrina <244>~ v~<225>~ 6~. Os novos compostos podem ser empregados como medicamentos.
BR0208885-1A 2001-04-14 2002-03-13 Inibidores de integrina alfavbeta6 BR0208885A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10118550A DE10118550A1 (de) 2001-04-14 2001-04-14 Liganden des Integrins alpha¶nu¶beta¶6¶
PCT/EP2002/002728 WO2002083627A2 (de) 2001-04-14 2002-03-13 Liganden des integrins alpha-v-beta-6

Publications (1)

Publication Number Publication Date
BR0208885A true BR0208885A (pt) 2004-06-29

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BR0208885-1A BR0208885A (pt) 2001-04-14 2002-03-13 Inibidores de integrina alfavbeta6

Country Status (16)

Country Link
US (1) US20040142877A1 (pt)
EP (1) EP1379495A2 (pt)
JP (1) JP2004528325A (pt)
KR (1) KR20030090739A (pt)
CN (1) CN1501827A (pt)
BR (1) BR0208885A (pt)
CA (1) CA2444247A1 (pt)
CZ (1) CZ20033000A3 (pt)
DE (1) DE10118550A1 (pt)
HU (1) HUP0303804A3 (pt)
MX (1) MXPA03009318A (pt)
PL (1) PL363328A1 (pt)
RU (1) RU2003130639A (pt)
SK (1) SK13732003A3 (pt)
WO (1) WO2002083627A2 (pt)
ZA (1) ZA200308857B (pt)

Families Citing this family (9)

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CA2478833C (en) 2002-03-13 2015-11-10 Biogen, Inc. Anti-.alpha.v.beta.6 antibodies
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WO2002083627A3 (de) 2003-10-09
WO2002083627A2 (de) 2002-10-24
HUP0303804A3 (en) 2005-09-28
SK13732003A3 (sk) 2004-02-03
CZ20033000A3 (cs) 2004-02-18
MXPA03009318A (es) 2004-02-12
RU2003130639A (ru) 2005-04-10
ZA200308857B (en) 2004-09-13
CA2444247A1 (en) 2002-10-24
KR20030090739A (ko) 2003-11-28
EP1379495A2 (de) 2004-01-14
JP2004528325A (ja) 2004-09-16
PL363328A1 (en) 2004-11-15
CN1501827A (zh) 2004-06-02
US20040142877A1 (en) 2004-07-22
HUP0303804A2 (hu) 2004-03-29

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