BR0207066A - Derivados do 2h-1-benzopirano - processos para sua preparação e composições farmacêuticas a partir deles - Google Patents

Derivados do 2h-1-benzopirano - processos para sua preparação e composições farmacêuticas a partir deles

Info

Publication number
BR0207066A
BR0207066A BR0207066-9A BR0207066A BR0207066A BR 0207066 A BR0207066 A BR 0207066A BR 0207066 A BR0207066 A BR 0207066A BR 0207066 A BR0207066 A BR 0207066A
Authority
BR
Brazil
Prior art keywords
preparation
processes
pharmaceutical compositions
benzopyran derivatives
benzopyran
Prior art date
Application number
BR0207066-9A
Other languages
English (en)
Portuguese (pt)
Inventor
Maurizio Delcanale
Gabriele Amari
Elisabetta Armani
Elisabetta Galbiati
Maurizio Civelli
Original Assignee
Chiesi Famraceutici S P A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP01101521A external-priority patent/EP1229036B1/en
Priority claimed from EP01118682A external-priority patent/EP1281710A1/en
Application filed by Chiesi Famraceutici S P A filed Critical Chiesi Famraceutici S P A
Publication of BR0207066A publication Critical patent/BR0207066A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
BR0207066-9A 2001-01-24 2002-01-21 Derivados do 2h-1-benzopirano - processos para sua preparação e composições farmacêuticas a partir deles BR0207066A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP01101521A EP1229036B1 (en) 2001-01-24 2001-01-24 2H-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
EP01118682A EP1281710A1 (en) 2001-08-03 2001-08-03 2H-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
PCT/EP2002/000567 WO2002059113A1 (en) 2001-01-24 2002-01-21 2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
BR0207066A true BR0207066A (pt) 2004-03-30

Family

ID=26076450

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0207066-9A BR0207066A (pt) 2001-01-24 2002-01-21 Derivados do 2h-1-benzopirano - processos para sua preparação e composições farmacêuticas a partir deles

Country Status (26)

Country Link
US (1) US6951883B2 (https=)
EP (1) EP1355906B1 (https=)
JP (1) JP4332349B2 (https=)
CN (1) CN1261431C (https=)
AT (1) ATE286894T1 (https=)
AU (1) AU2002237282B2 (https=)
BR (1) BR0207066A (https=)
CA (1) CA2435775A1 (https=)
CZ (1) CZ20032014A3 (https=)
DE (1) DE60202590T2 (https=)
DK (1) DK1355906T3 (https=)
DZ (1) DZ3459A1 (https=)
EA (1) EA006158B1 (https=)
ES (1) ES2236485T3 (https=)
HU (1) HUP0401018A3 (https=)
IL (2) IL157065A0 (https=)
MA (1) MA26982A1 (https=)
MX (1) MXPA03006505A (https=)
NO (1) NO327808B1 (https=)
NZ (1) NZ527144A (https=)
PL (1) PL365062A1 (https=)
PT (1) PT1355906E (https=)
SI (1) SI1355906T1 (https=)
SK (1) SK287086B6 (https=)
TN (1) TNSN03043A1 (https=)
WO (1) WO2002059113A1 (https=)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8080675B2 (en) 2004-09-21 2011-12-20 Marshall Edwards, Inc. Chroman derivatives, medicaments and use in therapy
JP4976649B2 (ja) * 2004-09-21 2012-07-18 マーシャル エドワーズ，インク． 化合物
JP4913056B2 (ja) * 2004-09-21 2012-04-11 マーシャル エドワーズ，インコーポレーテッド 置換クロマン誘導体、医薬品、および治療における使用
EP2436680B1 (en) * 2004-09-21 2016-05-18 Marshall Edwards, Inc. Chroman derivatives, medicaments and use in therapy
CA2581316C (en) 2004-09-21 2013-09-10 Novogen Research Pty Ltd Substituted chroman derivatives, medicaments and use in therapy
AU2005201855B2 (en) * 2004-09-21 2012-03-29 Marshall Edwards, Inc. Chroman derived compounds and formulations thereof for use in therapy
CN101444499B (zh) * 2007-11-26 2012-12-05 湘北威尔曼制药股份有限公司 一种化合物及其组合物的新用途
EP2635273B1 (en) 2010-11-01 2020-01-08 MEI Pharma, Inc. Isoflavonoid compositions and methods for the treatment of cancer
EA031077B1 (ru) 2013-06-19 2018-11-30 Серагон Фармасьютикалз, Инк. Модулятор рецептора эстрогена и его применения
CN116139125A (zh) 2015-02-02 2023-05-23 梅制药公司 联合治疗
ES3039455T3 (en) * 2016-11-17 2025-10-21 Sanofi Sa Novel substituted n-(3-fluoropropyl)-pyrrolidine compounds, processes for their preparation and therapeutic uses thereof
WO2019051562A1 (en) * 2017-09-15 2019-03-21 Norbio No. 1 Pty Ltd TREATMENT OF EXCITOTOXICITY
CN112225716A (zh) * 2020-10-30 2021-01-15 陕西嘉禾生物科技股份有限公司 一种鹰嘴豆牙素a的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3374245A (en) * 1964-04-01 1968-03-19 Ciba Geigy Corp Unsaturated oxacycles
DE1518002C3 (de) * 1965-01-02 1975-01-23 Merck Patent Gmbh, 6100 Darmstadt Isoflavane und Isoflavene und Verfahren zu Ihrer Herstellung sowie diese enthaltende Arzneimittel
US5280040A (en) 1993-03-11 1994-01-18 Zymogenetics, Inc. Methods for reducing bone loss using centchroman derivatives
AU744403B2 (en) * 1996-10-28 2002-02-21 Novo Nordisk A/S Novel trans-3,4-chroman derivatives useful in the prevention or treatment of estrogen related diseases or syndromes
US5985306A (en) * 1996-10-28 1999-11-16 Novo Nordisk A/S (+)-enantiomers of cis-3,4-chroman derivatives useful in prevention or treatment of estrogen diseases or syndromes
US6153768A (en) 1996-12-13 2000-11-28 C & C Research Laboratories Benzopyran derivatives
KR20000001793A (ko) * 1998-06-13 2000-01-15 이경하 신규한 벤조피란 또는 티오벤조피란 유도체
DK1140889T3 (da) 1998-12-30 2003-12-22 Signal Pharm Inc Forbindelser og metoder til modulation af estrogen-receptorer

Also Published As

Publication number Publication date
CA2435775A1 (en) 2002-08-01
AU2002237282B2 (en) 2007-02-15
PT1355906E (pt) 2005-05-31
WO2002059113A1 (en) 2002-08-01
DE60202590D1 (de) 2005-02-17
PL365062A1 (en) 2004-12-27
DZ3459A1 (fr) 2002-08-01
ATE286894T1 (de) 2005-01-15
NZ527144A (en) 2005-03-24
MA26982A1 (fr) 2004-12-20
SK287086B6 (sk) 2009-11-05
JP4332349B2 (ja) 2009-09-16
HUP0401018A2 (hu) 2004-09-28
ES2236485T3 (es) 2005-07-16
JP2004517151A (ja) 2004-06-10
EP1355906A1 (en) 2003-10-29
NO20033318L (no) 2003-09-24
EA006158B1 (ru) 2005-10-27
CN1261431C (zh) 2006-06-28
NO20033318D0 (no) 2003-07-23
CZ20032014A3 (cs) 2003-12-17
IL157065A0 (en) 2004-02-08
IL157065A (en) 2010-05-17
US6951883B2 (en) 2005-10-04
CN1487934A (zh) 2004-04-07
TNSN03043A1 (en) 2005-12-23
DK1355906T3 (da) 2005-05-30
EP1355906B1 (en) 2005-01-12
HUP0401018A3 (en) 2007-05-29
EA200300727A1 (ru) 2004-02-26
MXPA03006505A (es) 2004-04-21
NO327808B1 (no) 2009-09-28
HK1060558A1 (en) 2004-08-13
US20040106595A1 (en) 2004-06-03
SI1355906T1 (en) 2005-06-30
DE60202590T2 (de) 2005-12-29
SK9392003A3 (en) 2003-12-02

Similar Documents

Publication Publication Date Title
BR0209580A (pt) Derivados de ciclohexan-1, 4 diamina substituìdos
SE9704545D0 (sv) Novel compounds
SE9704544D0 (sv) Novel compounds
BR0317715A (pt) Composições e processos de uso de collajolie
PT960107E (pt) Compostos de paclitaxel 6-tio-substituidos
NO20042739L (no) Farmasoytiske sammensetninger av 5,6,14-triazatetracyklo(10.3.1.0(2,11).0(4,9))-heksadeca-2(11)3,5,7,9-pentan
ATE231872T1 (de) Thiazolopyrimidinderivate
BR0207066A (pt) Derivados do 2h-1-benzopirano - processos para sua preparação e composições farmacêuticas a partir deles
ZA9610460B (en) New phenylamidine derivatives, processes for preparing them and their use as pharmaceutical compositions.
BR0114380A (pt) Derivados-1-aminobutan-3-ol-substituìdos
DE60108354D1 (de) 2H-1-Benzopyran-Derivative, Prozesse zu ihrer Herstellung und Pharmazeutische Zusammensetzungen
NO995685L (no) Nye glycosylerte ginkgolidderivater, anvendelse derav som medikamenter og farmasoeytiske blandinger
DK0787135T3 (da) Vandopløslige derivater af epipodophyllotoxin, fremgangsmåde til fremstilling deraf og anvendelse som et lægemiddel til beh
AP2001002369A0 (en) Pharmaceutical complex.
EP0937708A3 (en) sulphonamide derivatives
NO20020914L (no) Alkoksy-substituerte benzimidazolforbindelser, preparater inneholdende slike samt anvendelser derav
PT1408035E (pt) Metodo de preparacao de derivativos de 1.5-diaril-3-trifluorometilo-delta2-pirazolinas que sejam racemicos e enanciomericamente puros
AR008474A1 (es) Derivado de 9-dihidroeritromicina a 6,9; 11,12-diciclocarbonato, composicion farmaceutica y preparacion bactericida que lo contienen y su uso
BR0114459A (pt) Derivados substituìdos de 5-amino-1-penten-3-ol substituidos
CA2420056A1 (en) 1-amino-alkylcyclohexanes as trypanocidal agents
ITMI992457A0 (it) Procedimento per la preparazione di (s)-n-terbutil-1,2,3,4-tetraidrois ochinolin-3-carbossiammide
UY27406A1 (es) Derivados de 2h-1-benzopirano, procesos para su preparación y composiciones farmacéuticas que los contienen
SE9902673D0 (sv) New composition
IT1318986B1 (it) Procedimento per la preparazione di (s)-n-terbutil-1,2,3,4-tetraidroisochinolin-3-carbossiammide.
WO2002100342A3 (en) (s, s'), (s, r')-amphetaminil, compositions and uses thereof

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A(S) 9A ANUIDADE(S)

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2103 DE 26/04/2011.