BR0202681A - Compostos de octaidro-2h-pirido[1,2a]pirazina, um processo para sua preparação e composições farmacêuticas contendo-as - Google Patents

Compostos de octaidro-2h-pirido[1,2a]pirazina, um processo para sua preparação e composições farmacêuticas contendo-as

Info

Publication number
BR0202681A
BR0202681A BR0202681-3A BR0202681A BR0202681A BR 0202681 A BR0202681 A BR 0202681A BR 0202681 A BR0202681 A BR 0202681A BR 0202681 A BR0202681 A BR 0202681A
Authority
BR
Brazil
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
compounds
octahydro
Prior art date
Application number
BR0202681-3A
Other languages
English (en)
Portuguese (pt)
Inventor
Solo Goldstein
Guillaume Poissonet
Jean-Gilles Parmentier
Pierre Lestage
Brian Lockhart
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of BR0202681A publication Critical patent/BR0202681A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR0202681-3A 2001-07-12 2002-07-11 Compostos de octaidro-2h-pirido[1,2a]pirazina, um processo para sua preparação e composições farmacêuticas contendo-as BR0202681A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0109260A FR2827288B1 (fr) 2001-07-12 2001-07-12 Nouveaux derives d'octahydro-2h-pyrido[1,2-a]pyrazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
BR0202681A true BR0202681A (pt) 2003-05-06

Family

ID=8865405

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0202681-3A BR0202681A (pt) 2001-07-12 2002-07-11 Compostos de octaidro-2h-pirido[1,2a]pirazina, um processo para sua preparação e composições farmacêuticas contendo-as

Country Status (24)

Country Link
US (1) US6992085B2 (cg-RX-API-DMAC7.html)
EP (1) EP1275647B1 (cg-RX-API-DMAC7.html)
JP (1) JP3950018B2 (cg-RX-API-DMAC7.html)
KR (1) KR100485020B1 (cg-RX-API-DMAC7.html)
CN (1) CN1197863C (cg-RX-API-DMAC7.html)
AR (1) AR036166A1 (cg-RX-API-DMAC7.html)
AT (1) ATE254124T1 (cg-RX-API-DMAC7.html)
AU (1) AU2002300094B2 (cg-RX-API-DMAC7.html)
BR (1) BR0202681A (cg-RX-API-DMAC7.html)
CA (1) CA2394027C (cg-RX-API-DMAC7.html)
DE (1) DE60200089T2 (cg-RX-API-DMAC7.html)
DK (1) DK1275647T3 (cg-RX-API-DMAC7.html)
EA (1) EA005160B1 (cg-RX-API-DMAC7.html)
ES (1) ES2210219T3 (cg-RX-API-DMAC7.html)
FR (1) FR2827288B1 (cg-RX-API-DMAC7.html)
HU (1) HUP0202282A3 (cg-RX-API-DMAC7.html)
MX (1) MXPA02006699A (cg-RX-API-DMAC7.html)
NO (1) NO322966B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ520120A (cg-RX-API-DMAC7.html)
PL (1) PL355034A1 (cg-RX-API-DMAC7.html)
PT (1) PT1275647E (cg-RX-API-DMAC7.html)
SI (1) SI1275647T1 (cg-RX-API-DMAC7.html)
TR (1) TR200302001T4 (cg-RX-API-DMAC7.html)
ZA (1) ZA200205596B (cg-RX-API-DMAC7.html)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1611902A4 (en) * 2003-04-03 2006-04-12 Kyowa Hakko Kogyo Kk MEANS FOR THE PREVENTION AND / OR TREATMENT OF NEUROPATHIC PAIN
MY141255A (en) * 2003-12-11 2010-03-31 Memory Pharm Corp Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs
FR2866647B1 (fr) * 2004-02-20 2006-10-27 Servier Lab Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2006000914A1 (en) * 2004-06-22 2006-01-05 Pfizer Products Inc. Diazabicyclic histamine-3 receptor antagonists
EP2233470B1 (en) * 2005-07-04 2011-12-07 High Point Pharmaceuticals, LLC Histamine H3 receptor antagonists
RU2442775C2 (ru) * 2005-07-04 2012-02-20 Хай Пойнт Фармасьютикалс, ЛЛС Антагонисты гистаминовых н3-рецепторов
US7795262B2 (en) * 2006-03-10 2010-09-14 Neurogen Corporation Piperazinyl oxoalkyl tetrahydroisoquinolines and related analogues
KR100871691B1 (ko) 2006-10-16 2008-12-05 삼성전자주식회사 병렬 비트 테스트 방법 및 그 방법을 사용하는 반도체메모리 장치
JP7015092B2 (ja) 2016-07-28 2022-02-02 塩野義製薬株式会社 ドーパミンｄ３受容体拮抗作用を有する含窒素縮環化合物
CN111801330B (zh) 2018-01-26 2024-04-05 盐野义制药株式会社 具有多巴胺d3受体拮抗作用的稠环化合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3388128A (en) * 1965-09-03 1968-06-11 Allan R. Day Substituted 1, 4-diazabicyclo [4. 4. 9] decanes
GB8518236D0 (en) * 1985-07-19 1985-08-29 Beecham Group Plc Compounds
WO1994006794A1 (en) * 1992-09-24 1994-03-31 National Institutes Of Health Aralkyl diazabicycloalkane derivatives for cns disorders
US6231833B1 (en) * 1999-08-05 2001-05-15 Pfizer Inc 2,7-substituted octahydro-1H-pyrido[1,2-A]pyrazine derivatives as ligands for serotonin receptors
WO1996010570A1 (en) * 1994-09-30 1996-04-11 Pfizer Inc. NEUROLEPTIC 2,7-DISUBSTITUTED PERHYDRO-1H-PYRIDO[1,2-a]PYRAZINES
AU773317B2 (en) * 1999-07-19 2004-05-20 Merck Canada Inc. Pyrazinones, compositions containing such compounds

Also Published As

Publication number Publication date
EA200200663A1 (ru) 2003-02-27
AR036166A1 (es) 2004-08-18
MXPA02006699A (es) 2005-08-16
CA2394027A1 (fr) 2003-01-12
EP1275647B1 (fr) 2003-11-12
ATE254124T1 (de) 2003-11-15
PT1275647E (pt) 2004-03-31
ES2210219T3 (es) 2004-07-01
CN1197863C (zh) 2005-04-20
CN1397557A (zh) 2003-02-19
FR2827288A1 (fr) 2003-01-17
NZ520120A (en) 2004-03-26
HUP0202282A2 (hu) 2003-03-28
KR100485020B1 (ko) 2005-04-25
JP3950018B2 (ja) 2007-07-25
PL355034A1 (en) 2003-01-13
EP1275647A1 (fr) 2003-01-15
DE60200089T2 (de) 2004-09-09
US20030195216A1 (en) 2003-10-16
KR20030007159A (ko) 2003-01-23
SI1275647T1 (en) 2004-02-29
NO20023345D0 (no) 2002-07-11
EA005160B1 (ru) 2004-12-30
FR2827288B1 (fr) 2003-10-31
TR200302001T4 (tr) 2004-01-21
DE60200089D1 (de) 2003-12-18
HK1050682A1 (en) 2003-07-04
NO20023345L (no) 2003-01-13
HU0202282D0 (cg-RX-API-DMAC7.html) 2002-09-28
CA2394027C (fr) 2008-01-08
HUP0202282A3 (en) 2003-11-28
NO322966B1 (no) 2006-12-18
DK1275647T3 (da) 2004-03-15
ZA200205596B (en) 2003-03-27
AU2002300094B2 (en) 2007-06-14
US6992085B2 (en) 2006-01-31
JP2003064081A (ja) 2003-03-05

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE 8A. ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2103 DE 26/04/2011.