BR0008798A - L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmos - Google Patents
L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmosInfo
- Publication number
- BR0008798A BR0008798A BR0008798-0A BR0008798A BR0008798A BR 0008798 A BR0008798 A BR 0008798A BR 0008798 A BR0008798 A BR 0008798A BR 0008798 A BR0008798 A BR 0008798A
- Authority
- BR
- Brazil
- Prior art keywords
- processes
- preparation
- pharmaceutical compositions
- compositions containing
- arabino
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 229940045799 anthracyclines and related substance Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/24—Condensed ring systems having three or more rings
- C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
- A61K31/704—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
"L-ARABINO-DISSACARìDEOS DE ANTRACICLINAS,PROCESSOS PARA SUA PREPARAçãO E COMPOSIçõESFARMACêUTICAS CONTENDO OS MESMOS". A presenteinvenção se refere a compostos de fórmula geral (I), aos saisfarmaceuticamente aceitáveis dos mesmos, aos processos parasua preparação e às composições farmacêuticas contendo osmesmos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1999FI000043A IT1307846B1 (it) | 1999-03-09 | 1999-03-09 | L-arabino disaccaridi di antracicline, loro processi di preparazione ecomposizioni farmaceutiche che li contengono. |
PCT/EP2000/002006 WO2000053615A1 (en) | 1999-03-09 | 2000-03-08 | L-arabino-disaccharides of anthracyclines, processes for their preparation, and pharmaceutical compositions containing them |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0008798A true BR0008798A (pt) | 2001-12-26 |
Family
ID=11352829
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0008798-0A BR0008798A (pt) | 1999-03-09 | 2000-03-08 | L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmos |
Country Status (23)
Country | Link |
---|---|
US (1) | US6653289B1 (pt) |
EP (1) | EP1169327B1 (pt) |
JP (1) | JP2002539133A (pt) |
KR (1) | KR20010105368A (pt) |
CN (1) | CN1150201C (pt) |
AR (1) | AR042571A1 (pt) |
AT (1) | ATE311398T1 (pt) |
AU (1) | AU3554500A (pt) |
BG (1) | BG105881A (pt) |
BR (1) | BR0008798A (pt) |
CA (1) | CA2366675A1 (pt) |
CZ (1) | CZ296359B6 (pt) |
DE (1) | DE60024428D1 (pt) |
EA (1) | EA003455B1 (pt) |
EE (1) | EE200100474A (pt) |
HU (1) | HUP0200208A3 (pt) |
IT (1) | IT1307846B1 (pt) |
MX (1) | MXPA01009025A (pt) |
PL (1) | PL353169A1 (pt) |
SK (1) | SK12802001A3 (pt) |
TR (1) | TR200102584T2 (pt) |
UA (1) | UA69446C2 (pt) |
WO (1) | WO2000053615A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7737123B2 (en) * | 2005-05-12 | 2010-06-15 | The Ohio State University Research Foundation | Multidrug resistant anticancer anthracyclines |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1262565B (it) * | 1993-09-30 | 1996-07-04 | Menarini Farma Ind | Disaccaridi di antracicline, loro processi di preparazione e composizioni farmaceutiche che li contengono. |
-
1999
- 1999-03-09 IT IT1999FI000043A patent/IT1307846B1/it active
-
2000
- 2000-03-08 SK SK1280-2001A patent/SK12802001A3/sk unknown
- 2000-03-08 TR TR2001/02584T patent/TR200102584T2/xx unknown
- 2000-03-08 EP EP00914117A patent/EP1169327B1/en not_active Expired - Lifetime
- 2000-03-08 AU AU35545/00A patent/AU3554500A/en not_active Abandoned
- 2000-03-08 MX MXPA01009025A patent/MXPA01009025A/es unknown
- 2000-03-08 PL PL00353169A patent/PL353169A1/xx unknown
- 2000-03-08 EA EA200100953A patent/EA003455B1/ru not_active IP Right Cessation
- 2000-03-08 AT AT00914117T patent/ATE311398T1/de not_active IP Right Cessation
- 2000-03-08 EE EEP200100474A patent/EE200100474A/xx unknown
- 2000-03-08 CN CNB008046808A patent/CN1150201C/zh not_active Expired - Fee Related
- 2000-03-08 BR BR0008798-0A patent/BR0008798A/pt not_active IP Right Cessation
- 2000-03-08 CA CA002366675A patent/CA2366675A1/en not_active Abandoned
- 2000-03-08 WO PCT/EP2000/002006 patent/WO2000053615A1/en not_active Application Discontinuation
- 2000-03-08 DE DE60024428T patent/DE60024428D1/de not_active Expired - Lifetime
- 2000-03-08 HU HU0200208A patent/HUP0200208A3/hu unknown
- 2000-03-08 JP JP2000604050A patent/JP2002539133A/ja active Pending
- 2000-03-08 US US09/914,987 patent/US6653289B1/en not_active Expired - Fee Related
- 2000-03-08 CZ CZ20013228A patent/CZ296359B6/cs not_active IP Right Cessation
- 2000-03-08 KR KR1020017011178A patent/KR20010105368A/ko not_active Application Discontinuation
- 2000-03-09 AR ARP000101041A patent/AR042571A1/es unknown
- 2000-08-03 UA UA2001106843A patent/UA69446C2/uk unknown
-
2001
- 2001-09-05 BG BG105881A patent/BG105881A/bg unknown
Also Published As
Publication number | Publication date |
---|---|
EE200100474A (et) | 2002-12-16 |
SK12802001A3 (sk) | 2002-01-07 |
PL353169A1 (en) | 2003-11-03 |
HUP0200208A2 (hu) | 2002-05-29 |
ATE311398T1 (de) | 2005-12-15 |
US6653289B1 (en) | 2003-11-25 |
EP1169327A1 (en) | 2002-01-09 |
BG105881A (bg) | 2002-06-28 |
CA2366675A1 (en) | 2000-09-14 |
JP2002539133A (ja) | 2002-11-19 |
CN1150201C (zh) | 2004-05-19 |
ITFI990043A0 (it) | 1999-03-09 |
IT1307846B1 (it) | 2001-11-19 |
AR042571A1 (es) | 2005-06-29 |
WO2000053615A1 (en) | 2000-09-14 |
MXPA01009025A (es) | 2002-10-23 |
HUP0200208A3 (en) | 2003-08-28 |
EA200100953A1 (ru) | 2002-02-28 |
CZ20013228A3 (cs) | 2002-02-13 |
TR200102584T2 (tr) | 2002-03-21 |
CZ296359B6 (cs) | 2006-02-15 |
EA003455B1 (ru) | 2003-06-26 |
DE60024428D1 (de) | 2006-01-05 |
ITFI990043A1 (it) | 2000-09-09 |
KR20010105368A (ko) | 2001-11-28 |
AU3554500A (en) | 2000-09-28 |
CN1343214A (zh) | 2002-04-03 |
EP1169327B1 (en) | 2005-11-30 |
UA69446C2 (uk) | 2004-09-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A , 8A E 9A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009. |