BR0008798A - L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmos - Google Patents

L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmos

Info

Publication number
BR0008798A
BR0008798A BR0008798-0A BR0008798A BR0008798A BR 0008798 A BR0008798 A BR 0008798A BR 0008798 A BR0008798 A BR 0008798A BR 0008798 A BR0008798 A BR 0008798A
Authority
BR
Brazil
Prior art keywords
processes
preparation
pharmaceutical compositions
compositions containing
arabino
Prior art date
Application number
BR0008798-0A
Other languages
English (en)
Inventor
Fabio Animati
Marco Berettoni
Mario Bigioni
Amalia Cipollone
Arlos Alberto Maggi
Original Assignee
Menarini Ricerche Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Menarini Ricerche Spa filed Critical Menarini Ricerche Spa
Publication of BR0008798A publication Critical patent/BR0008798A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/24Condensed ring systems having three or more rings
    • C07H15/252Naphthacene radicals, e.g. daunomycins, adriamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A61K31/704Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

"L-ARABINO-DISSACARìDEOS DE ANTRACICLINAS,PROCESSOS PARA SUA PREPARAçãO E COMPOSIçõESFARMACêUTICAS CONTENDO OS MESMOS". A presenteinvenção se refere a compostos de fórmula geral (I), aos saisfarmaceuticamente aceitáveis dos mesmos, aos processos parasua preparação e às composições farmacêuticas contendo osmesmos.
BR0008798-0A 1999-03-09 2000-03-08 L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmos BR0008798A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT1999FI000043A IT1307846B1 (it) 1999-03-09 1999-03-09 L-arabino disaccaridi di antracicline, loro processi di preparazione ecomposizioni farmaceutiche che li contengono.
PCT/EP2000/002006 WO2000053615A1 (en) 1999-03-09 2000-03-08 L-arabino-disaccharides of anthracyclines, processes for their preparation, and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
BR0008798A true BR0008798A (pt) 2001-12-26

Family

ID=11352829

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0008798-0A BR0008798A (pt) 1999-03-09 2000-03-08 L-arabino-dissacarìdeos de antraciclinas,processos para sua preparação e composiçõesfarmacêuticas contendo os mesmos

Country Status (23)

Country Link
US (1) US6653289B1 (pt)
EP (1) EP1169327B1 (pt)
JP (1) JP2002539133A (pt)
KR (1) KR20010105368A (pt)
CN (1) CN1150201C (pt)
AR (1) AR042571A1 (pt)
AT (1) ATE311398T1 (pt)
AU (1) AU3554500A (pt)
BG (1) BG105881A (pt)
BR (1) BR0008798A (pt)
CA (1) CA2366675A1 (pt)
CZ (1) CZ296359B6 (pt)
DE (1) DE60024428D1 (pt)
EA (1) EA003455B1 (pt)
EE (1) EE200100474A (pt)
HU (1) HUP0200208A3 (pt)
IT (1) IT1307846B1 (pt)
MX (1) MXPA01009025A (pt)
PL (1) PL353169A1 (pt)
SK (1) SK12802001A3 (pt)
TR (1) TR200102584T2 (pt)
UA (1) UA69446C2 (pt)
WO (1) WO2000053615A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7737123B2 (en) * 2005-05-12 2010-06-15 The Ohio State University Research Foundation Multidrug resistant anticancer anthracyclines

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1262565B (it) * 1993-09-30 1996-07-04 Menarini Farma Ind Disaccaridi di antracicline, loro processi di preparazione e composizioni farmaceutiche che li contengono.

Also Published As

Publication number Publication date
EE200100474A (et) 2002-12-16
SK12802001A3 (sk) 2002-01-07
PL353169A1 (en) 2003-11-03
HUP0200208A2 (hu) 2002-05-29
ATE311398T1 (de) 2005-12-15
US6653289B1 (en) 2003-11-25
EP1169327A1 (en) 2002-01-09
BG105881A (bg) 2002-06-28
CA2366675A1 (en) 2000-09-14
JP2002539133A (ja) 2002-11-19
CN1150201C (zh) 2004-05-19
ITFI990043A0 (it) 1999-03-09
IT1307846B1 (it) 2001-11-19
AR042571A1 (es) 2005-06-29
WO2000053615A1 (en) 2000-09-14
MXPA01009025A (es) 2002-10-23
HUP0200208A3 (en) 2003-08-28
EA200100953A1 (ru) 2002-02-28
CZ20013228A3 (cs) 2002-02-13
TR200102584T2 (tr) 2002-03-21
CZ296359B6 (cs) 2006-02-15
EA003455B1 (ru) 2003-06-26
DE60024428D1 (de) 2006-01-05
ITFI990043A1 (it) 2000-09-09
KR20010105368A (ko) 2001-11-28
AU3554500A (en) 2000-09-28
CN1343214A (zh) 2002-04-03
EP1169327B1 (en) 2005-11-30
UA69446C2 (uk) 2004-09-15

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A , 8A E 9A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009.