BG17800A3 - Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини - Google Patents

Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини

Info

Publication number
BG17800A3
BG17800A3 BG017732A BG1773270A BG17800A3 BG 17800 A3 BG17800 A3 BG 17800A3 BG 017732 A BG017732 A BG 017732A BG 1773270 A BG1773270 A BG 1773270A BG 17800 A3 BG17800 A3 BG 17800A3
Authority
BG
Bulgaria
Prior art keywords
thieno
pyrimidines
furyl
nitro
preparation
Prior art date
Application number
BG017732A
Other languages
Bulgarian (bg)
English (en)
Inventor
Eberhard Woitun
Wolfgang Reuter
Original Assignee
Dr. Karl Thomae Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691959403 external-priority patent/DE1959403A1/de
Priority claimed from DE19702050814 external-priority patent/DE2050814A1/de
Priority claimed from DE19702050815 external-priority patent/DE2050815A1/de
Priority claimed from DE19702050816 external-priority patent/DE2050816A1/de
Application filed by Dr. Karl Thomae Gmbh filed Critical Dr. Karl Thomae Gmbh
Publication of BG17800A3 publication Critical patent/BG17800A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
BG017732A 1969-11-26 1970-11-17 Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини BG17800A3 (bg)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19691959403 DE1959403A1 (de) 1969-11-26 1969-11-26 Neue 2-(5-Nitro-2-furyl)-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702050814 DE2050814A1 (de) 1970-10-16 1970-10-16 Neue Verfahren zur Herstellung von 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidinen
DE19702050815 DE2050815A1 (de) 1970-10-16 1970-10-16 Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine
DE19702050816 DE2050816A1 (de) 1970-10-16 1970-10-16 Neue 2-(Nitro-2-furyl>thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine

Publications (1)

Publication Number Publication Date
BG17800A3 true BG17800A3 (bg) 1973-12-25

Family

ID=27430978

Family Applications (2)

Application Number Title Priority Date Filing Date
BG017732A BG17800A3 (bg) 1969-11-26 1970-11-17 Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини
BG016080A BG17799A3 (bg) 1969-11-26 1970-11-17 Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG016080A BG17799A3 (bg) 1969-11-26 1970-11-17 Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини

Country Status (13)

Country Link
US (1) US3661908A (enExample)
BE (1) BE759493A (enExample)
BG (2) BG17800A3 (enExample)
CA (1) CA926865A (enExample)
CH (3) CH568324A5 (enExample)
DK (1) DK128781B (enExample)
FR (1) FR2073416B1 (enExample)
GB (1) GB1321316A (enExample)
IE (1) IE34765B1 (enExample)
IL (1) IL35729A (enExample)
NL (1) NL7017210A (enExample)
NO (1) NO129954B (enExample)
SE (1) SE377938B (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3932642A (en) * 1971-04-10 1976-01-13 Boehringer Ingelheim Gmbh Biocidal compositions containing a 2- (5'-nitro-2'-furyl)-thieno(2,3-d) pyrimidine and methods of use
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
US6608053B2 (en) * 2000-04-27 2003-08-19 Yamanouchi Pharmaceutical Co., Ltd. Fused heteroaryl derivatives
US20040138238A1 (en) * 2002-08-08 2004-07-15 Dhanoa Dale S. Substituted aminopyrimidine compounds as neurokinin antagonists
GB0423653D0 (en) * 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
AU2007243466B2 (en) * 2006-04-26 2012-01-19 F. Hoffmann-La Roche Ag Phosphoinositide 3-kinase inhibitor compounds and pharmaceutical compositions containing them
KR101533461B1 (ko) 2006-04-26 2015-07-02 에프. 호프만-라 로슈 아게 Pi3k저해제로 유용한 티에노[3,2-d]피리미딘 유도체
PL2041139T3 (pl) 2006-04-26 2012-05-31 Hoffmann La Roche Związki farmaceutyczne
CA2671845C (en) * 2006-12-07 2015-03-24 Genentech, Inc. Phosphoinositide 3-kinase inhibitor compounds and methods of use
PE20081679A1 (es) * 2006-12-07 2008-12-18 Hoffmann La Roche Compuestos del inhibidor de fosfoinositida 3-cinasa y metodos de uso
ATE510841T1 (de) * 2007-06-12 2011-06-15 Hoffmann La Roche Thiazoliopyrimidine und ihre verwendung als hemmer der phosphatidylinositol-3 kinase
CN101932587A (zh) * 2007-09-24 2010-12-29 吉宁特有限公司 噻唑并嘧啶pi3k抑制剂化合物及使用方法
WO2009055730A1 (en) 2007-10-25 2009-04-30 Genentech, Inc. Process for making thienopyrimidine compounds
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
JP5709766B2 (ja) 2009-03-12 2015-04-30 ジェネンテック, インコーポレイテッド 造血器腫瘍の治療のためのホスホイノシチド3キナーゼ阻害剤化合物と化学療法剤の併用
SG182247A1 (en) * 2009-05-27 2012-08-30 Hoffmann La Roche Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
MX2011012520A (es) 2009-05-27 2011-12-12 Hoffmann La Roche Compuestos inhibidores de pi3k de pirimidina biciclicos selectivos para p110 delta y metodos de uso de los mismos.
AU2010314287A1 (en) * 2009-10-12 2012-05-03 F. Hoffmann-La Roche Ag Combinations of a PI3K inhibitor and a MEK inhibitor
KR20130058672A (ko) 2010-04-16 2013-06-04 제넨테크, 인크. PI3K/AKT 키나제 경로 억제제 효능에 대한 예측 바이오마커로서의 FOXO3a
US20140004209A1 (en) 2010-12-22 2014-01-02 Genentech, Inc. Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms
RU2015140573A (ru) 2013-02-25 2017-03-30 Дженентек, Инк. Способы и композиции для обнаружения и лечения устойчивого к лекарственным средствам мутанта акт

Also Published As

Publication number Publication date
BE759493A (fr) 1971-05-25
IL35729A0 (en) 1971-01-28
SE377938B (enExample) 1975-08-04
NO129954B (enExample) 1974-06-17
CH559210A5 (enExample) 1975-02-28
US3661908A (en) 1972-05-09
NL7017210A (enExample) 1971-05-28
FR2073416B1 (enExample) 1975-04-18
FR2073416A1 (enExample) 1971-10-01
DK128781B (da) 1974-07-01
CH567029A5 (enExample) 1975-09-30
IE34765L (en) 1971-05-26
IL35729A (en) 1974-01-14
GB1321316A (en) 1973-06-27
IE34765B1 (en) 1975-08-06
CA926865A (en) 1973-05-22
BG17799A3 (bg) 1973-12-25
CH568324A5 (enExample) 1975-10-31

Similar Documents

Publication Publication Date Title
BE758910A (fr) Preparation de dimethyl-2, 2-propanediol-1, 3
BG20593A3 (bg) Метод за получаване на тиено<3,2-д>пиримидини
BG17799A3 (bg) Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини
BG17591A3 (bg) Метод за получаване на нови 2- аминоалкил амино- тиено /3,2-д пиримидини
BG18599A3 (bg) Метод за получаване на бета-арил-2-аминоалкоксистироли
BG17749A3 (bg) Метод за получаване на фенокси-2-хидрокси -3- циклоалкиламинопропани
BE745432A (fr) Procede pour la preparation de methionine
BG19166A3 (bg) Метод за получаване на тиено(3,2-д)-пиримидини
BG19597A3 (bg) Метод за получаване на перидо/ 3,2-д/ пиримидини
BG17798A3 (bg) Метод за получаване на нови 2-аминоалкил-аминотиено (3,2-d)пиримидини
BG17560A3 (bg) Метод за получаане на 4,20, 22- буфатриеноли- драмнозид- етери
CH550152A (fr) Procede de preparation de nouvelles iodomethylsulfones.
FI52216C (fi) Menetelmä gamma-piperidinobutyrofenonijohdannaisten valmistamiseksi.
ZA707999B (en) Improvements relating to 2-(5-nitro-2-furyl)-thieno(3,2-d)pyrimidines
SU446967A3 (ru) Способ получения -замещенных2-(5-нитро-2-фурил)-4-аминотиено (2,3- )пиримидинов
BG18603A3 (bg) Метод за непрекъснато получаване на циклохексаноноксим
BE750991A (fr) Procede pour la preparation de tetrahydrothiophene
BG20578A3 (bg) Метод за получаване на карденолид-3-<2,3,-дидезоксигликозиди>
BE750384A (fr) Procede de preparation de 5-(l'-alcenyl-)-2-norbornene
BG19164A3 (bg) Метод за получаване на 2-(5-нитро-2-фурил)-тиеро(3,2-алфа)пиримидин
BE779136R (fr) Procede de preparation d'acetoxy-1-methyl-3-butene-2-al-4
BG17971A3 (bg) Метод за получаване на нови 2- аминоалкиламино тиено/ 3,2-д/ пиримидини
DK125394B (da) Analogifremgangsmåde til fremstilling af benzofuranderivater.
FI49980C (fi) Menetelmä (alempi)alkyyli-5-(5-nitro-2-furyyli)-3-metyyli-isoksatsoli- 4-karboksylaattien valmistamiseksi.
BG17562A3 (bg) Метод за получаване на з- карбамоил -3- метил-6,7 диметокси-1- тиаизохроман -1,1- двуокис