BG105384A - CRYSTALLINE FORMS OF Et02C-CH2-(R)Cgl-Aze-Pab-OH - Google Patents
CRYSTALLINE FORMS OF Et02C-CH2-(R)Cgl-Aze-Pab-OHInfo
- Publication number
- BG105384A BG105384A BG105384A BG10538401A BG105384A BG 105384 A BG105384 A BG 105384A BG 105384 A BG105384 A BG 105384A BG 10538401 A BG10538401 A BG 10538401A BG 105384 A BG105384 A BG 105384A
- Authority
- BG
- Bulgaria
- Prior art keywords
- aze
- cgl
- pab
- et02c
- crystalline forms
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9802974A SE9802974D0 (sv) | 1998-09-03 | 1998-09-03 | New crystalline forms |
| PCT/SE1999/001514 WO2000014110A1 (en) | 1998-09-03 | 1999-09-02 | CRYSTALLINE FORMS OF EtO2C-CH2-(R)Cgl-Aze-Pab-OH |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG105384A true BG105384A (en) | 2001-11-30 |
Family
ID=20412468
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG105384A BG105384A (en) | 1998-09-03 | 2001-03-26 | CRYSTALLINE FORMS OF Et02C-CH2-(R)Cgl-Aze-Pab-OH |
Country Status (39)
| Country | Link |
|---|---|
| US (5) | US6225287B1 (ru) |
| EP (1) | EP1107980B1 (ru) |
| JP (2) | JP3493341B2 (ru) |
| KR (1) | KR100629825B1 (ru) |
| CN (1) | CN1204143C (ru) |
| AP (1) | AP1520A (ru) |
| AR (1) | AR029312A1 (ru) |
| AT (1) | ATE231521T1 (ru) |
| AU (1) | AU763421B2 (ru) |
| BG (1) | BG105384A (ru) |
| BR (1) | BR9913464A (ru) |
| CA (1) | CA2341259A1 (ru) |
| CU (1) | CU23015A3 (ru) |
| CZ (1) | CZ2001775A3 (ru) |
| DE (1) | DE69905054T2 (ru) |
| DK (1) | DK1107980T3 (ru) |
| EA (1) | EA003264B1 (ru) |
| EE (1) | EE200100135A (ru) |
| ES (1) | ES2192101T3 (ru) |
| HK (1) | HK1034721A1 (ru) |
| HR (1) | HRP20010132B1 (ru) |
| HU (1) | HUP0104330A2 (ru) |
| ID (1) | ID28779A (ru) |
| IL (1) | IL141433A0 (ru) |
| IS (1) | IS1942B (ru) |
| MY (1) | MY121394A (ru) |
| NO (1) | NO20011083L (ru) |
| NZ (2) | NZ510070A (ru) |
| OA (1) | OA11908A (ru) |
| PL (1) | PL346544A1 (ru) |
| SA (1) | SA99200682B1 (ru) |
| SE (1) | SE9802974D0 (ru) |
| SK (1) | SK2802001A3 (ru) |
| TR (1) | TR200100700T2 (ru) |
| TW (1) | TWI247013B (ru) |
| UA (1) | UA66869C2 (ru) |
| WO (1) | WO2000014110A1 (ru) |
| YU (1) | YU17301A (ru) |
| ZA (1) | ZA200101763B (ru) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9802974D0 (sv) * | 1998-09-03 | 1998-09-03 | Astra Ab | New crystalline forms |
| SE9900070D0 (sv) | 1999-01-13 | 1999-01-13 | Astra Ab | New use |
| SE9902550D0 (sv) | 1999-07-02 | 1999-07-02 | Astra Ab | New crystalline forms |
| US20020115603A1 (en) * | 2000-06-22 | 2002-08-22 | Chiron Corporation | Methods and compositions for the treatment of peripheral artery disease |
| GB0015981D0 (en) * | 2000-06-29 | 2000-08-23 | Glaxo Group Ltd | Novel process for preparing crystalline particles |
| JP4275407B2 (ja) * | 2000-10-12 | 2009-06-10 | 中外製薬株式会社 | 新規な結晶構造を有するエリスロマイシン誘導体及びその製造方法 |
| US7129233B2 (en) * | 2000-12-01 | 2006-10-31 | Astrazeneca Ab | Mandelic acid derivatives and their use as thrombin inhibitors |
| AR035216A1 (es) * | 2000-12-01 | 2004-05-05 | Astrazeneca Ab | Derivados de acido mandelico ,derivados farmaceuticamente aceptables, uso de estos derivados para la fabricacion de medicamentos, metodos de tratamiento ,procesos para la preparacion de estos derivados, y compuestos intermediarios |
| AR034517A1 (es) * | 2001-06-21 | 2004-02-25 | Astrazeneca Ab | Formulacion farmaceutica |
| WO2003076391A2 (de) | 2002-03-11 | 2003-09-18 | Curacyte Ag | Hemmstoffe der urokinase, ihre herstellung und verwendung |
| SE0201659D0 (sv) * | 2002-05-31 | 2002-05-31 | Astrazeneca Ab | Modified release pharmaceutical formulation |
| SE0201661D0 (sv) | 2002-05-31 | 2002-05-31 | Astrazeneca Ab | New salts |
| DE10301300B4 (de) | 2003-01-15 | 2009-07-16 | Curacyte Chemistry Gmbh | Verwendung von acylierten 4-Amidino- und 4-Guanidinobenzylaminen zur Inhibierung von Plasmakallikrein |
| US7781424B2 (en) * | 2003-05-27 | 2010-08-24 | Astrazeneca Ab | Modified release pharmaceutical formulation |
| DE10342108A1 (de) | 2003-09-11 | 2005-04-14 | Curacyte Chemistry Gmbh | Basisch-substituierte Benzylaminanaloga als Inhibitoren des Gerinnungsfaktors Xa, ihre Herstellung und Verwendung |
| WO2005031397A2 (en) * | 2003-09-26 | 2005-04-07 | Zetetic Institute | Catoptric and catadioptric imaging systems with pellicle and aperture-array beam-splitters and non-adaptive and adaptive catoptric surfaces |
| US20050209211A1 (en) * | 2004-03-16 | 2005-09-22 | Devalina Law | Trihemihydrate, anhydrate and novel hydrate forms of Cefdinir |
| WO2005091696A1 (fr) * | 2004-03-29 | 2005-10-06 | Quanta Display Inc. | Structure a cadres pour module retroeclaire |
| US7524354B2 (en) * | 2005-07-07 | 2009-04-28 | Research Foundation Of State University Of New York | Controlled synthesis of highly monodispersed gold nanoparticles |
| DE102006050672A1 (de) | 2006-10-24 | 2008-04-30 | Curacyte Discovery Gmbh | Hemmstoffe des Plasmins und des Plasmakallikreins |
| TW200827336A (en) * | 2006-12-06 | 2008-07-01 | Astrazeneca Ab | New crystalline forms |
| US20090061000A1 (en) * | 2007-08-31 | 2009-03-05 | Astrazeneca Ab | Pharmaceutical formulation use 030 |
| ES2420989T3 (es) * | 2010-02-26 | 2013-08-28 | Biedermann Technologies Gmbh & Co. Kg | Implante para estabilizar huesos o vértebras |
| US9550585B2 (en) | 2014-06-09 | 2017-01-24 | Space Systems/Loral, Llc | Highly inclined elliptical orbit de-orbit techniques |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1075277B (it) * | 1977-02-11 | 1985-04-22 | Erba Carlo Spa | Derivati insaturi e epossidici dell'acio 7-acilamido-3-cefem-4-carbossilico e procedimento per la loro preparazione |
| US4315011A (en) * | 1978-07-12 | 1982-02-09 | Richter Gedeon Vegyeszeti Gyar Rt. | 1-Alkyl-9-bromohexahydroindolo quinolizium salts and use thereof to increase blood flow |
| DE3169094D1 (en) * | 1980-11-20 | 1985-03-28 | Beecham Group Plc | Secondary amines |
| SE9301916D0 (sv) * | 1993-06-03 | 1993-06-03 | Ab Astra | New peptides derivatives |
| SE504185C2 (sv) * | 1994-11-08 | 1996-12-02 | Astra Ab | Lagringsstabil vattenlösning för infusion av trombininhibitorer |
| AR005245A1 (es) | 1995-12-21 | 1999-04-28 | Astrazeneca Ab | Prodrogas de inhibidores de trombina, una formulación farmaceutica que las comprende, el uso de dichas prodrogas para la manufactura de un medicamento y un procedimiento para su preparacion |
| US5830805A (en) * | 1996-11-18 | 1998-11-03 | Cornell Research Foundation | Electroless deposition equipment or apparatus and method of performing electroless deposition |
| SE9802974D0 (sv) * | 1998-09-03 | 1998-09-03 | Astra Ab | New crystalline forms |
-
1998
- 1998-09-03 SE SE9802974A patent/SE9802974D0/xx unknown
-
1999
- 1999-08-24 TW TW088114464A patent/TWI247013B/zh not_active IP Right Cessation
- 1999-09-01 MY MYPI99003779A patent/MY121394A/en unknown
- 1999-09-02 US US09/424,770 patent/US6225287B1/en not_active Expired - Fee Related
- 1999-09-02 IL IL14143399A patent/IL141433A0/xx unknown
- 1999-09-02 TR TR2001/00700T patent/TR200100700T2/xx unknown
- 1999-09-02 CU CU20010061A patent/CU23015A3/es unknown
- 1999-09-02 BR BR9913464-0A patent/BR9913464A/pt not_active IP Right Cessation
- 1999-09-02 DK DK99968671T patent/DK1107980T3/da active
- 1999-09-02 YU YU17301A patent/YU17301A/sh unknown
- 1999-09-02 EA EA200100194A patent/EA003264B1/ru not_active IP Right Cessation
- 1999-09-02 AR ARP990104422A patent/AR029312A1/es unknown
- 1999-09-02 NZ NZ510070A patent/NZ510070A/xx not_active IP Right Cessation
- 1999-09-02 JP JP2000568867A patent/JP3493341B2/ja not_active Expired - Fee Related
- 1999-09-02 ES ES99968671T patent/ES2192101T3/es not_active Expired - Lifetime
- 1999-09-02 AU AU60147/99A patent/AU763421B2/en not_active Ceased
- 1999-09-02 AP APAP/P/2001/002078A patent/AP1520A/en active
- 1999-09-02 ID IDW20010492A patent/ID28779A/id unknown
- 1999-09-02 KR KR1020017002730A patent/KR100629825B1/ko not_active IP Right Cessation
- 1999-09-02 AT AT99968671T patent/ATE231521T1/de active
- 1999-09-02 PL PL99346544A patent/PL346544A1/xx not_active Application Discontinuation
- 1999-09-02 CZ CZ2001775A patent/CZ2001775A3/cs unknown
- 1999-09-02 HU HU0104330A patent/HUP0104330A2/hu unknown
- 1999-09-02 DE DE69905054T patent/DE69905054T2/de not_active Expired - Lifetime
- 1999-09-02 SK SK280-2001A patent/SK2802001A3/sk unknown
- 1999-09-02 CN CNB998128384A patent/CN1204143C/zh not_active Expired - Fee Related
- 1999-09-02 EP EP99968671A patent/EP1107980B1/en not_active Expired - Lifetime
- 1999-09-02 UA UA2001021083A patent/UA66869C2/ru unknown
- 1999-09-02 OA OA00100056A patent/OA11908A/en unknown
- 1999-09-02 EE EEP200100135A patent/EE200100135A/xx unknown
- 1999-09-02 CA CA002341259A patent/CA2341259A1/en not_active Abandoned
- 1999-09-02 NZ NZ524486A patent/NZ524486A/en not_active IP Right Cessation
- 1999-09-02 WO PCT/SE1999/001514 patent/WO2000014110A1/en active IP Right Grant
- 1999-10-18 SA SA99200682A patent/SA99200682B1/ar unknown
-
2001
- 2001-01-04 US US09/753,655 patent/US6440939B2/en not_active Expired - Fee Related
- 2001-02-23 HR HR20010132A patent/HRP20010132B1/xx not_active IP Right Cessation
- 2001-02-28 IS IS5870A patent/IS1942B/is unknown
- 2001-03-01 ZA ZA200101763A patent/ZA200101763B/en unknown
- 2001-03-02 NO NO20011083A patent/NO20011083L/no not_active Application Discontinuation
- 2001-03-26 BG BG105384A patent/BG105384A/xx unknown
- 2001-08-02 HK HK01105394A patent/HK1034721A1/xx not_active IP Right Cessation
-
2002
- 2002-05-20 US US10/147,908 patent/US6888007B2/en not_active Expired - Fee Related
-
2003
- 2003-08-26 JP JP2003300959A patent/JP2004075687A/ja active Pending
-
2005
- 2005-03-11 US US11/077,210 patent/US20050153901A1/en not_active Abandoned
-
2006
- 2006-08-22 US US11/507,513 patent/US20060287249A1/en not_active Abandoned
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