BG102618A - Derivatives of 5h, 1oh-imidazo[1,2-a)inden[1,2-e]pyrazin-4-on, their preparation and their intermediate products and medicaments containing them - Google Patents

Derivatives of 5h, 1oh-imidazo[1,2-a)inden[1,2-e]pyrazin-4-on, their preparation and their intermediate products and medicaments containing them

Info

Publication number
BG102618A
BG102618A BG102618A BG10261898A BG102618A BG 102618 A BG102618 A BG 102618A BG 102618 A BG102618 A BG 102618A BG 10261898 A BG10261898 A BG 10261898A BG 102618 A BG102618 A BG 102618A
Authority
BG
Bulgaria
Prior art keywords
alk
cooh
po3h2
preparation
medicaments containing
Prior art date
Application number
BG102618A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jean-Claude Aloup
Jean Bouquerel
Dominique Damour
Jean-Claude Hardy
Patrick Jimonet
Franco Manfre
Serge Mignani
Patrick Nemecek
Original Assignee
Rhone-Poulenc Rorer S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone-Poulenc Rorer S.A. filed Critical Rhone-Poulenc Rorer S.A.
Publication of BG102618A publication Critical patent/BG102618A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG102618A 1996-01-10 1998-07-10 Derivatives of 5h, 1oh-imidazo[1,2-a)inden[1,2-e]pyrazin-4-on, their preparation and their intermediate products and medicaments containing them BG102618A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9600192A FR2743366B1 (fr) 1996-01-10 1996-01-10 Derives de 5h,10h-imidazo(1,2-a)indeno(1,2-e)pyrazine-4-one, leur preparation, leurs intermediaires et les medicaments les contenant
PCT/FR1997/000019 WO1997025328A1 (fr) 1996-01-10 1997-01-06 DERIVES DE 5H,10H-IMIDAZO(1,2-a)INDENO(1,2-e)PYRAZINE-4-ONE, LEUR PREPARATION, LEURS INTERMEDIAIRES ET LES MEDICAMENTS LES CONTENANT______________________________________________________________

Publications (1)

Publication Number Publication Date
BG102618A true BG102618A (en) 1999-09-30

Family

ID=9487995

Family Applications (1)

Application Number Title Priority Date Filing Date
BG102618A BG102618A (en) 1996-01-10 1998-07-10 Derivatives of 5h, 1oh-imidazo[1,2-a)inden[1,2-e]pyrazin-4-on, their preparation and their intermediate products and medicaments containing them

Country Status (20)

Country Link
US (2) US5990108A (de)
EP (1) EP0880522B1 (de)
JP (1) JP2000505073A (de)
KR (1) KR19990077135A (de)
AR (1) AR005424A1 (de)
AT (1) ATE205847T1 (de)
AU (1) AU1383097A (de)
BG (1) BG102618A (de)
CA (1) CA2239254A1 (de)
CZ (1) CZ216698A3 (de)
DE (1) DE69706830T2 (de)
DK (1) DK0880522T3 (de)
ES (1) ES2164323T3 (de)
FR (1) FR2743366B1 (de)
MX (1) MX9805167A (de)
PL (1) PL327942A1 (de)
PT (1) PT880522E (de)
SK (1) SK93498A3 (de)
WO (1) WO1997025328A1 (de)
ZA (1) ZA9786B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999047497A2 (en) * 1998-03-13 1999-09-23 Merck Frosst Canada & Co. Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
US6242493B1 (en) 1998-03-13 2001-06-05 Merck Frosst Canada & Co. Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
WO2003029210A2 (en) * 2001-10-04 2003-04-10 Merck & Co. Inc. Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
WO2003070722A1 (fr) * 2002-02-21 2003-08-28 Azwell Inc. Amelioration apportee a la production de derives d'imidazole et de nouveaux intermediaires de ces derives
GB0415320D0 (en) * 2004-07-08 2004-08-11 Astrazeneca Ab Novel compounds
US7649098B2 (en) * 2006-02-24 2010-01-19 Lexicon Pharmaceuticals, Inc. Imidazole-based compounds, compositions comprising them and methods of their use
TW200920355A (en) * 2007-09-06 2009-05-16 Lexicon Pharmaceuticals Inc Compositions and methods for treating immunological and inflammatory diseases and disorders
US9737531B2 (en) 2012-07-12 2017-08-22 Glytech, Llc Composition and method for treatment of depression and psychosis in humans
JP7305560B2 (ja) 2017-06-12 2023-07-10 グリテック, エルエルシー Nmdaアンタゴニスト及びd2/5ht2a又は選択的5ht2aアンタゴニストによるうつ病の治療

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2717812B1 (fr) * 1994-03-28 1996-05-10 Rhone Poulenc Rorer Sa Indeno[1,2-e]pyrazine-4-ones, leur préparation et les médicaments les contenant.
FR2732681B1 (fr) * 1995-04-05 1997-07-04 Rhone Poulenc Rorer Sa Derives de 10h-imidazo(1,2-a)indeno(1,2-e)pyrazin-4-one, leur preparation et les medicaments les contenant

Also Published As

Publication number Publication date
FR2743366B1 (fr) 1998-02-06
DE69706830T2 (de) 2002-04-25
ZA9786B (en) 1997-07-17
KR19990077135A (ko) 1999-10-25
US5990108A (en) 1999-11-23
JP2000505073A (ja) 2000-04-25
CA2239254A1 (fr) 1997-07-17
AU1383097A (en) 1997-08-01
WO1997025328A1 (fr) 1997-07-17
AR005424A1 (es) 1999-06-23
MX9805167A (es) 1998-10-31
EP0880522A1 (de) 1998-12-02
ATE205847T1 (de) 2001-10-15
SK93498A3 (en) 1998-12-02
EP0880522B1 (de) 2001-09-19
PL327942A1 (en) 1999-01-04
ES2164323T3 (es) 2002-02-16
DK0880522T3 (da) 2002-01-21
CZ216698A3 (cs) 1998-10-14
PT880522E (pt) 2002-05-31
FR2743366A1 (fr) 1997-07-11
DE69706830D1 (de) 2001-10-25
US6100264A (en) 2000-08-08

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