BE901210A - Nouveaux retinoides. - Google Patents

Nouveaux retinoides.

Info

Publication number
BE901210A
BE901210A BE0/214112A BE214112A BE901210A BE 901210 A BE901210 A BE 901210A BE 0/214112 A BE0/214112 A BE 0/214112A BE 214112 A BE214112 A BE 214112A BE 901210 A BE901210 A BE 901210A
Authority
BE
Belgium
Prior art keywords
retinoids
linked
sugar
new retinoids
new
Prior art date
Application number
BE0/214112A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BE901210A publication Critical patent/BE901210A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
    • C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Nutrition Science (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cosmetics (AREA)

Abstract

Ces rétinoides répondent à la formule générale (I) dans laquelle R est le reste d'un sucre relié par une liaison ester ou d'un aminosucre relié par une liaison amide ou d'un dérivé de sucre, et n est égal à 1 ou 2. Ces composés sont des médicaments utilisables notamment pour le traitement des néoplasies, de l'acné et du psoriasis, en particulier en application topique.
BE0/214112A 1983-12-08 1984-12-05 Nouveaux retinoides. BE901210A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH6570/83A CH661516A5 (de) 1983-12-08 1983-12-08 Phenylnonatetraenoylzuckerderivate.

Publications (1)

Publication Number Publication Date
BE901210A true BE901210A (fr) 1985-06-05

Family

ID=4311671

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/214112A BE901210A (fr) 1983-12-08 1984-12-05 Nouveaux retinoides.

Country Status (14)

Country Link
US (1) US4565863A (fr)
JP (1) JPS60146896A (fr)
AU (1) AU571278B2 (fr)
BE (1) BE901210A (fr)
CA (1) CA1234107A (fr)
CH (1) CH661516A5 (fr)
DE (1) DE3444051C2 (fr)
DK (1) DK163585C (fr)
FR (1) FR2556348B1 (fr)
GB (1) GB2152498B (fr)
IT (1) IT1177263B (fr)
NL (1) NL8403554A (fr)
SE (1) SE468987B (fr)
ZA (1) ZA849364B (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5110801A (en) * 1984-08-13 1992-05-05 Leveen Harry H Treatment of acne
AT388166B (de) * 1986-06-03 1989-05-10 Oesterr Zuckerfab Evidenz Verfahren zur herstellung von neuen wasserloeslichen kohlenhydrat-derivaten
LU87035A1 (fr) * 1987-11-04 1989-06-14 Oreal Esters du type etretinique ou apparente d'antibiotiques macrolidiques et lincosamidiques,leur procede de preparation et compositions pharmaceutiques et cosmetiques les contenant
FR2644460A1 (fr) * 1989-03-16 1990-09-21 Oreal Esters retinoiques de d-desosamine, leur procede de preparation et leur utilisation en medecine humaine ou veterinaire et en cosmetique
FR2644459B1 (fr) * 1989-03-16 1994-10-28 Oreal Esters retinoiques de l-cladinose, leur procede de preparation et leur utilisation en medecine humaine ou veterinaire et en cosmetique
WO1990014092A1 (fr) * 1989-05-18 1990-11-29 Cell Genesys, Inc. Utilisation d'oligonucleotides mono-brins pour la modification axee sur le site de genes mammiferes in vivo
US5075340A (en) * 1989-05-22 1991-12-24 Iowa State University Research Foundation Retinoic acid glucuronide preparations for application to the skin
KR950013763B1 (ko) * 1989-05-22 1995-11-15 아이오아 스테이트 유니버시티 리서치 파운데이션 인코포레이티드 레티노산 글루쿠로나이드를 포함하는 약제학적 조성물
US5235076A (en) * 1991-05-28 1993-08-10 University Of Hawaii Azulenic retinoid compounds, compositions and methods
CH684092A5 (de) * 1992-04-21 1994-07-15 Ciba Geigy Ag Wasserlösliche Retinoide.
GB2282596B (en) * 1993-10-06 1998-04-15 Ciba Geigy Ag Water-soluble retinoids
US5534261A (en) * 1995-01-17 1996-07-09 University Of Southern California Retinoid-based compositions and method for preventing adhesion formation using the same
FR2768630B1 (fr) * 1997-09-22 2000-08-04 Ulice Sa Utilisation d'alkyl monoglucosides en tant que vecteurs moleculaires
FR2791679B1 (fr) * 1999-03-31 2003-04-11 Fabre Pierre Dermo Cosmetique Bioprecurseurs aptes a liberer un derive retinoique par mise a profit de l'activite enzymatique de la surface cutanee et compositions pharmaceutiques et/ou cosmetiques
US20050148534A1 (en) * 2003-09-22 2005-07-07 Castellino Angelo J. Small molecule compositions and methods for increasing drug efficiency using compositions thereof
EP1765773A2 (fr) * 2004-07-09 2007-03-28 DSMIP Assets B.V. Congugues amino, d'acides amines ou de peptides d'acide retinoique
US8003621B2 (en) * 2007-09-14 2011-08-23 Nitto Denko Corporation Drug carriers

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3219657A (en) * 1961-02-27 1965-11-23 Monsanto Co Saccharide polydicarboxylate half-esters
US4224244A (en) * 1973-03-30 1980-09-23 Hoffmann-La Roche Inc. 9-Phenyl 5,6-dimethyl-nona-2,4,6,8 tetraenal or tetraenol derivatives
CH585166A5 (fr) * 1973-03-30 1977-02-28 Hoffmann La Roche
US4215215A (en) * 1975-08-01 1980-07-29 Hoffmann-La Roche Inc. 9-Phenyl-nonate traene compounds
LU77254A1 (fr) * 1977-05-04 1979-01-18
JPS5640651A (en) * 1979-09-12 1981-04-16 Takeda Chem Ind Ltd Quinone compound and its preparation
FI67386C (fi) * 1979-06-21 1985-03-11 Hoffmann La Roche Foerfarande foer framstaellning av nya terapeutiskt anvaendbara sockerderivat

Also Published As

Publication number Publication date
CH661516A5 (de) 1987-07-31
GB2152498B (en) 1987-09-09
AU571278B2 (en) 1988-04-14
DE3444051A1 (de) 1985-06-13
SE8406138L (sv) 1985-06-09
NL8403554A (nl) 1985-07-01
GB2152498A (en) 1985-08-07
SE8406138D0 (sv) 1984-12-04
US4565863A (en) 1986-01-21
DK163585C (da) 1992-08-24
AU3514384A (en) 1985-06-13
IT1177263B (it) 1987-08-26
SE468987B (sv) 1993-04-26
JPH0524920B2 (fr) 1993-04-09
DK587384D0 (da) 1984-12-07
IT8423661A1 (it) 1986-05-20
GB8430915D0 (en) 1985-01-16
FR2556348B1 (fr) 1988-10-14
CA1234107A (fr) 1988-03-15
JPS60146896A (ja) 1985-08-02
FR2556348A1 (fr) 1985-06-14
DE3444051C2 (de) 1994-08-04
DK163585B (da) 1992-03-16
DK587384A (da) 1985-06-09
ZA849364B (en) 1985-07-31
IT8423661A0 (it) 1984-11-20

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: F. HOFFMANN-LA ROCHE A.G.

Effective date: 19951231