BE871857A - Nouvelles piperazines disubstituees, leur procedes de preparation et les compositions pharmaceutiques les renfermant - Google Patents

Nouvelles piperazines disubstituees, leur procedes de preparation et les compositions pharmaceutiques les renfermant

Info

Publication number
BE871857A
BE871857A BE191610A BE191610A BE871857A BE 871857 A BE871857 A BE 871857A BE 191610 A BE191610 A BE 191610A BE 191610 A BE191610 A BE 191610A BE 871857 A BE871857 A BE 871857A
Authority
BE
Belgium
Prior art keywords
disubstitled
piperazines
preparation
new
methods
Prior art date
Application number
BE191610A
Other languages
English (en)
French (fr)
Original Assignee
Science Union & Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Science Union & Cie filed Critical Science Union & Cie
Publication of BE871857A publication Critical patent/BE871857A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D327/00Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
BE191610A 1977-11-09 1978-11-08 Nouvelles piperazines disubstituees, leur procedes de preparation et les compositions pharmaceutiques les renfermant BE871857A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4664677 1977-11-09

Publications (1)

Publication Number Publication Date
BE871857A true BE871857A (fr) 1979-05-08

Family

ID=10442057

Family Applications (1)

Application Number Title Priority Date Filing Date
BE191610A BE871857A (fr) 1977-11-09 1978-11-08 Nouvelles piperazines disubstituees, leur procedes de preparation et les compositions pharmaceutiques les renfermant

Country Status (14)

Country Link
US (1) US4260610A (nl)
JP (1) JPS5481284A (nl)
AR (3) AR220730A1 (nl)
AU (1) AU4140778A (nl)
BE (1) BE871857A (nl)
CA (1) CA1117944A (nl)
DE (1) DE2848139A1 (nl)
ES (1) ES474896A1 (nl)
FR (1) FR2408605A1 (nl)
IL (1) IL55894A (nl)
IT (1) IT1109266B (nl)
NL (1) NL7811135A (nl)
OA (1) OA06083A (nl)
ZA (1) ZA786262B (nl)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3321969A1 (de) * 1983-06-18 1984-12-20 Troponwerke GmbH & Co KG, 5000 Köln 2-pyrimidinyl-1-piperazin-derivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE3902316A1 (de) * 1989-01-26 1990-08-02 Lentia Gmbh Neue piperazinylalkyl-3(2h)-pyridazinone, verfahren zu ihrer herstellung und ihre verwendung als blutdrucksenkende mittel
US4988699A (en) * 1989-03-14 1991-01-29 Warner-Lambert Company Substituted tetrahydrobenzothiazoles as dopaminergic agents
US4954503A (en) * 1989-09-11 1990-09-04 Hoechst-Roussel Pharmaceuticals, Inc. 3-(1-substituted-4-piperazinyl)-1H-indazoles
FR2671350A1 (fr) * 1991-01-08 1992-07-10 Adir Nouveaux derives de benzisoxazole et de benzisothiazole, leur procede de preparation, et les compositions pharmaceutiques les renfermant.
US5859246A (en) 1997-01-30 1999-01-12 Neurogen Corporation 1-phenyl-4-benzylpiperazines: dopamine receptor subtype specific ligands
RU2576037C1 (ru) * 2014-11-28 2016-02-27 Закрытое акционерное общество "Исследовательский институт Химического разнообразия" ЗАО "ИИХР" Замещенные 4-{ [4-(3,3-диоксидо-1,3-бензоксатиол-6-ил)арилокси]метил} пиперидины как агонисты рецепторов gpr119, фармацевтическая композиция, способы их получения и применения
US10906894B2 (en) * 2016-06-09 2021-02-02 Pramana Pharmaceuticals Inc. Compounds containing benzo[d][1,3]oxathiole, benzo[d][1,3]oxathiole 3-oxide or benzo[d][1,3]oxathiole 3,3-dioxide and methods/uses thereof as agonists of g protein-coupled receptor 119
WO2019104418A1 (en) 2017-11-30 2019-06-06 Pramana Pharmaceuticals Inc. Compounds containing polysubstituted benzo[d][1,3]oxathiole, benzo[d][1,3]oxathiole 3-oxide or benzo[d][1,3]oxathiole 3,3-dioxide and methods/uses thereof as agonists of g protein-coupled receptor 119

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2459367A (en) * 1947-11-12 1949-01-18 American Cyanamid Co 1,4-di (heterocyclic substituted) piperazines
US2561036A (en) * 1948-06-07 1951-07-17 Noel S Sodders Thread-cutting sheet metal nut
NL127996C (nl) * 1963-11-19
DE1595923A1 (de) * 1965-02-20 1969-11-27 Merck Ag E 1-Aralkyl-4-(thiazolyl-2)-piperazine und Verfahren zu ihrer Herstellung
GB1187680A (en) * 1967-11-15 1970-04-15 Science Union & Cie New Heterocyclic Substituted Piperazines
GB1407552A (en) * 1973-04-02 1975-09-24 Science Union & Cie Disubstituted piperazines processes for their preparation and pharmaceutical compositions containing them
GB1432660A (en) * 1973-10-30 1976-04-22 Science Union & Cie Piperazine derivatives processes for their preparation and and pharamacueitcal compositions containing them

Also Published As

Publication number Publication date
IT7851814A0 (it) 1978-11-08
FR2408605B1 (nl) 1982-02-05
OA06083A (fr) 1981-06-30
JPS5481284A (en) 1979-06-28
NL7811135A (nl) 1979-05-11
ES474896A1 (es) 1979-03-16
AR220794A1 (es) 1980-11-28
AR220730A1 (es) 1980-11-28
CA1117944A (fr) 1982-02-09
AR220793A1 (es) 1980-11-28
AU4140778A (en) 1979-05-17
DE2848139A1 (de) 1979-05-10
IL55894A (en) 1981-09-13
IL55894A0 (en) 1979-01-31
FR2408605A1 (fr) 1979-06-08
IT1109266B (it) 1985-12-16
JPS6136755B2 (nl) 1986-08-20
US4260610A (en) 1981-04-07
ZA786262B (en) 1979-10-31

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: SCIENCE UNION ET CIE SOC. FRANCAISE DE RECHERCHE

Effective date: 19861130