AR220794A1 - Procedimiento de preparacion de derivados de la i-(benzoxatiolilmetil)-4-heterociclil piperazina - Google Patents

Procedimiento de preparacion de derivados de la i-(benzoxatiolilmetil)-4-heterociclil piperazina

Info

Publication number
AR220794A1
AR220794A1 AR278947A AR27894779A AR220794A1 AR 220794 A1 AR220794 A1 AR 220794A1 AR 278947 A AR278947 A AR 278947A AR 27894779 A AR27894779 A AR 27894779A AR 220794 A1 AR220794 A1 AR 220794A1
Authority
AR
Argentina
Prior art keywords
benzoxatiolyl
heterociclil
piperazine
derivatives
methyl
Prior art date
Application number
AR278947A
Other languages
English (en)
Original Assignee
Medicale Rech France
Science Union & Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medicale Rech France, Science Union & Cie filed Critical Medicale Rech France
Application granted granted Critical
Publication of AR220794A1 publication Critical patent/AR220794A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D327/00Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR278947A 1977-11-09 1979-11-29 Procedimiento de preparacion de derivados de la i-(benzoxatiolilmetil)-4-heterociclil piperazina AR220794A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4664677 1977-11-09

Publications (1)

Publication Number Publication Date
AR220794A1 true AR220794A1 (es) 1980-11-28

Family

ID=10442057

Family Applications (3)

Application Number Title Priority Date Filing Date
AR274381A AR220730A1 (es) 1977-11-09 1978-11-08 Procedimiento para la preparacion de nuevos derivados de la i-((benzoxatiolil)-metil)-4-heterociclil-piperazina
AR278946A AR220793A1 (es) 1977-11-09 1979-11-19 Procedimiento de preparacion de derivados de la i-(benzoxatiolilmetil)-4-heterociclil piperazina
AR278947A AR220794A1 (es) 1977-11-09 1979-11-29 Procedimiento de preparacion de derivados de la i-(benzoxatiolilmetil)-4-heterociclil piperazina

Family Applications Before (2)

Application Number Title Priority Date Filing Date
AR274381A AR220730A1 (es) 1977-11-09 1978-11-08 Procedimiento para la preparacion de nuevos derivados de la i-((benzoxatiolil)-metil)-4-heterociclil-piperazina
AR278946A AR220793A1 (es) 1977-11-09 1979-11-19 Procedimiento de preparacion de derivados de la i-(benzoxatiolilmetil)-4-heterociclil piperazina

Country Status (14)

Country Link
US (1) US4260610A (es)
JP (1) JPS5481284A (es)
AR (3) AR220730A1 (es)
AU (1) AU4140778A (es)
BE (1) BE871857A (es)
CA (1) CA1117944A (es)
DE (1) DE2848139A1 (es)
ES (1) ES474896A1 (es)
FR (1) FR2408605A1 (es)
IL (1) IL55894A (es)
IT (1) IT1109266B (es)
NL (1) NL7811135A (es)
OA (1) OA06083A (es)
ZA (1) ZA786262B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3321969A1 (de) * 1983-06-18 1984-12-20 Troponwerke GmbH & Co KG, 5000 Köln 2-pyrimidinyl-1-piperazin-derivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE3902316A1 (de) * 1989-01-26 1990-08-02 Lentia Gmbh Neue piperazinylalkyl-3(2h)-pyridazinone, verfahren zu ihrer herstellung und ihre verwendung als blutdrucksenkende mittel
US4988699A (en) * 1989-03-14 1991-01-29 Warner-Lambert Company Substituted tetrahydrobenzothiazoles as dopaminergic agents
US4954503A (en) * 1989-09-11 1990-09-04 Hoechst-Roussel Pharmaceuticals, Inc. 3-(1-substituted-4-piperazinyl)-1H-indazoles
FR2671350A1 (fr) * 1991-01-08 1992-07-10 Adir Nouveaux derives de benzisoxazole et de benzisothiazole, leur procede de preparation, et les compositions pharmaceutiques les renfermant.
US5859246A (en) * 1997-01-30 1999-01-12 Neurogen Corporation 1-phenyl-4-benzylpiperazines: dopamine receptor subtype specific ligands
RU2576037C1 (ru) * 2014-11-28 2016-02-27 Закрытое акционерное общество "Исследовательский институт Химического разнообразия" ЗАО "ИИХР" Замещенные 4-{ [4-(3,3-диоксидо-1,3-бензоксатиол-6-ил)арилокси]метил} пиперидины как агонисты рецепторов gpr119, фармацевтическая композиция, способы их получения и применения
FI3468967T3 (fi) * 2016-06-09 2023-10-26 Pramana Pharmaceuticals Inc Bentso[d][1,3]oksatiolia, bentso[d][1,3]oksatioli-3-oksidia tai bentso[d][1,3]oksatioli-3,3-dioksidia sisältäviä yhdisteitä ja menetelmiä niitä varten ja niiden käyttösovelluksia G-proteiinikytkentäisen reseptorin 119 agonisteina
US11358956B2 (en) 2017-11-30 2022-06-14 Pramana Pharmaceuticals Inc. Compounds containing polysubstituted benzo[d][1,3]oxathiole, benzo[d][1,3]oxathiole 3-oxide or benzo[d][1,3]oxathiole 3,3-dioxide and methods/uses thereof as agonists of G protein-coupled receptor 119

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2459367A (en) * 1947-11-12 1949-01-18 American Cyanamid Co 1,4-di (heterocyclic substituted) piperazines
US2561036A (en) * 1948-06-07 1951-07-17 Noel S Sodders Thread-cutting sheet metal nut
NL127996C (es) * 1963-11-19
DE1595923A1 (de) * 1965-02-20 1969-11-27 Merck Ag E 1-Aralkyl-4-(thiazolyl-2)-piperazine und Verfahren zu ihrer Herstellung
GB1187680A (en) * 1967-11-15 1970-04-15 Science Union & Cie New Heterocyclic Substituted Piperazines
GB1407552A (en) * 1973-04-02 1975-09-24 Science Union & Cie Disubstituted piperazines processes for their preparation and pharmaceutical compositions containing them
GB1432660A (en) * 1973-10-30 1976-04-22 Science Union & Cie Piperazine derivatives processes for their preparation and and pharamacueitcal compositions containing them

Also Published As

Publication number Publication date
US4260610A (en) 1981-04-07
IT1109266B (it) 1985-12-16
IT7851814A0 (it) 1978-11-08
AR220730A1 (es) 1980-11-28
CA1117944A (fr) 1982-02-09
FR2408605B1 (es) 1982-02-05
BE871857A (fr) 1979-05-08
IL55894A (en) 1981-09-13
JPS6136755B2 (es) 1986-08-20
OA06083A (fr) 1981-06-30
DE2848139A1 (de) 1979-05-10
JPS5481284A (en) 1979-06-28
NL7811135A (nl) 1979-05-11
FR2408605A1 (fr) 1979-06-08
AR220793A1 (es) 1980-11-28
ZA786262B (en) 1979-10-31
IL55894A0 (en) 1979-01-31
AU4140778A (en) 1979-05-17
ES474896A1 (es) 1979-03-16

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