BE860773A - Beta-lactames monocycliques, leur procede de preparation et leur application en therapeutique - Google Patents

Beta-lactames monocycliques, leur procede de preparation et leur application en therapeutique

Info

Publication number
BE860773A
BE860773A BE182574A BE182574A BE860773A BE 860773 A BE860773 A BE 860773A BE 182574 A BE182574 A BE 182574A BE 182574 A BE182574 A BE 182574A BE 860773 A BE860773 A BE 860773A
Authority
BE
Belgium
Prior art keywords
lactames
preparation process
therapeutic application
monocyclic beta
monocyclic
Prior art date
Application number
BE182574A
Other languages
English (en)
French (fr)
Original Assignee
Smithkline Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Corp filed Critical Smithkline Corp
Publication of BE860773A publication Critical patent/BE860773A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE182574A 1976-11-15 1977-11-14 Beta-lactames monocycliques, leur procede de preparation et leur application en therapeutique BE860773A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/742,149 US4144333A (en) 1976-11-15 1976-11-15 Monocyclic beta-lactams with antibacterial activity

Publications (1)

Publication Number Publication Date
BE860773A true BE860773A (fr) 1978-05-16

Family

ID=24983681

Family Applications (1)

Application Number Title Priority Date Filing Date
BE182574A BE860773A (fr) 1976-11-15 1977-11-14 Beta-lactames monocycliques, leur procede de preparation et leur application en therapeutique

Country Status (22)

Country Link
US (1) US4144333A (no)
JP (1) JPS5363370A (no)
AU (1) AU514506B2 (no)
BE (1) BE860773A (no)
CA (1) CA1120935A (no)
CH (2) CH638781A5 (no)
DE (1) DE2751041A1 (no)
DK (1) DK497677A (no)
ES (2) ES464008A1 (no)
FI (1) FI773383A (no)
FR (1) FR2392006A1 (no)
GB (2) GB1594003A (no)
IE (1) IE45982B1 (no)
IL (1) IL53342A (no)
IT (1) IT1088885B (no)
LU (1) LU78497A1 (no)
NL (1) NL7712508A (no)
NO (1) NO150040C (no)
PH (1) PH22249A (no)
PT (1) PT67251B (no)
SE (1) SE7712645L (no)
ZA (1) ZA776131B (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4257947A (en) * 1977-08-03 1981-03-24 Smithkline Corporation 3-Amino-2-hydroxy, halo or mercaptomethyl-4-oxoazetidines
ATE9584T1 (de) * 1980-02-14 1984-10-15 Beecham Group Plc Antibakterielle beta-lactam-verbindungen, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen.
EP0187355A1 (en) 1981-09-23 1986-07-16 E.R. Squibb & Sons, Inc. Process for preparing beta-lactam antibiotics
FR2515182B1 (fr) * 1981-10-23 1986-05-09 Roussel Uclaf Nouveaux produits derives de l'acide 3-amino 2-oxo azetidine 1-sulfamique, leur procede de preparation, leur application comme medicaments et les produits intermediaires necessaires a leur preparation
US7425541B2 (en) * 1998-12-11 2008-09-16 Medarex, Inc. Enzyme-cleavable prodrug compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH563396A5 (no) * 1970-06-05 1975-06-30 Ciba Geigy Ag
US3943123A (en) * 1971-04-30 1976-03-09 Koninklijke Nederlandsche Gist-En Spiritusfabriek N.V. Novel beta-lactams and novel process
US3840556A (en) * 1971-05-28 1974-10-08 Lilly Co Eli Penicillin conversion by halogen electrophiles and anti-bacterials derived thereby
DE2204105A1 (de) * 1972-01-28 1973-08-02 Beecham Group Ltd Seco-penicilline und verfahren zu ihrer herstellung
US3920696A (en) * 1973-04-02 1975-11-18 Lilly Co Eli 2s-carboxyalkylthio-3r-imidoazetidin-4-ones and compounds useful in their preparation
US3917644A (en) * 1973-08-03 1975-11-04 Lilly Co Eli Azetidinesulfenic acids
US3901880A (en) * 1974-09-11 1975-08-26 Hoffmann La Roche (s)-alanyl-3-(+60 -(s)-chloro-3-(s)-hydroxy-2-oxo-azetidinylmethyl)-(s)-alanine
US4000154A (en) * 1975-09-03 1976-12-28 Smithkline Corporation 3-Substituted-6β-(amino- and acylamino)-7-oxo-1,3-diazabicyclo[3.2.0]-h

Also Published As

Publication number Publication date
NL7712508A (nl) 1978-05-17
ES464000A1 (es) 1978-07-16
IL53342A (en) 1981-07-31
FR2392006A1 (fr) 1978-12-22
FR2392006B1 (no) 1981-07-24
US4144333A (en) 1979-03-13
NO150040C (no) 1984-08-15
CA1120935A (en) 1982-03-30
IE45982B1 (en) 1983-01-12
PH22249A (en) 1988-07-01
GB1594003A (en) 1981-07-30
AU3058677A (en) 1979-05-17
AU514506B2 (en) 1981-02-12
CH638781A5 (de) 1983-10-14
IT1088885B (it) 1985-06-10
GB1594004A (en) 1981-07-30
CH641448A5 (de) 1984-02-29
PT67251B (en) 1979-04-16
LU78497A1 (no) 1978-03-20
PT67251A (en) 1977-12-01
ES464008A1 (es) 1978-08-01
DK497677A (da) 1978-05-16
NO150040B (no) 1984-04-30
FI773383A (fi) 1978-05-16
NO773900L (no) 1978-05-18
DE2751041A1 (de) 1978-05-24
SE7712645L (sv) 1978-05-16
IE45982L (en) 1978-05-15
ZA776131B (en) 1978-06-28
JPS5363370A (en) 1978-06-06
IL53342A0 (en) 1978-01-31
JPS6324990B2 (no) 1988-05-23

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: SMITHKLINE CORP.

Effective date: 19881130