BE855412A - Derives nouveaux de 4-hydroxy-aporphine et leur mode de preparation - Google Patents

Derives nouveaux de 4-hydroxy-aporphine et leur mode de preparation

Info

Publication number
BE855412A
BE855412A BE6046041A BE6046041A BE855412A BE 855412 A BE855412 A BE 855412A BE 6046041 A BE6046041 A BE 6046041A BE 6046041 A BE6046041 A BE 6046041A BE 855412 A BE855412 A BE 855412A
Authority
BE
Belgium
Prior art keywords
aporphine
hydroxy
preparation
new derivatives
derivatives
Prior art date
Application number
BE6046041A
Other languages
English (en)
Inventor
Johannes Hartenstein
Gerhard Satzinger
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of BE855412A publication Critical patent/BE855412A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • C07D221/18Ring systems of four or more rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/18Aralkyl radicals
    • C07D217/20Aralkyl radicals with oxygen atoms directly attached to the aromatic ring of said aralkyl radical, e.g. papaverine
BE6046041A 1976-06-04 1977-06-03 Derives nouveaux de 4-hydroxy-aporphine et leur mode de preparation BE855412A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2625116A DE2625116C2 (de) 1976-06-04 1976-06-04 Verfahren zur Herstellung von 4-Hydroxy-aporphin-Derivaten

Publications (1)

Publication Number Publication Date
BE855412A true BE855412A (fr) 1977-12-05

Family

ID=5979808

Family Applications (1)

Application Number Title Priority Date Filing Date
BE6046041A BE855412A (fr) 1976-06-04 1977-06-03 Derives nouveaux de 4-hydroxy-aporphine et leur mode de preparation

Country Status (14)

Country Link
US (1) US4120964A (fr)
JP (1) JPS535169A (fr)
AU (1) AU508171B2 (fr)
BE (1) BE855412A (fr)
CH (1) CH629782A5 (fr)
DE (1) DE2625116C2 (fr)
DK (1) DK248277A (fr)
ES (1) ES459504A1 (fr)
FR (1) FR2353534A1 (fr)
GB (1) GB1521020A (fr)
IE (1) IE44937B1 (fr)
LU (1) LU77482A1 (fr)
NL (1) NL7706180A (fr)
SE (1) SE433212B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2412534A1 (fr) * 1977-12-22 1979-07-20 Warner Lambert Co Preparation de derives de 1-hydroxyaporphines

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2757335C3 (de) * 1977-12-22 1982-03-25 Gödecke AG, 1000 Berlin Verfahren zur O-Methylierung von Hydroxyaporphinen
FI68813C (fi) * 1978-08-21 1985-11-11 Dow Chemical Co Foerfarande foer framstaellning av terapeutiskt effektiva 1- och d,1-glausinfosfatsalter
DE3324090A1 (de) * 1983-07-05 1985-01-17 Basf Ag, 6700 Ludwigshafen Elektrophotographische aufzeichnungsmaterialien mit verbesserter photoempfindlichkeit
DE3324089A1 (de) * 1983-07-05 1985-01-17 Basf Ag, 6700 Ludwigshafen Elektrophotographische aufzeichnungsmaterialien mit verbesserter photoempfindlichkeit
US5156847A (en) * 1990-09-20 1992-10-20 Walter H. Lewis Wound-healing composition
US5474782A (en) * 1994-05-20 1995-12-12 Woundfast Pharmaceuticals, Inc. Wound-healing composition and method
US5659037A (en) * 1994-08-18 1997-08-19 Abbott Laboratories Process for preparing chiral tetracyclic dopaminergic compounds
DE19535762A1 (de) * 1995-09-26 1997-03-27 Basf Ag Verfahren zur Racematspaltung
US5932617A (en) * 1998-02-06 1999-08-03 Woundfast Pharmaceuticals Inc. Wound-treating composition and method
US6210680B1 (en) 1999-06-11 2001-04-03 Univera Pharmaceuticals, Inc. Method for the prevention and treatment of chronic venous insufficiency
US20030187011A1 (en) * 2001-12-20 2003-10-02 Lashuel Hilal A. Apomorphine inhibitors of amyloid-beta (Abeta) fibril formation and their use in amyloidosis based disease
TWI404536B (zh) * 2008-06-20 2013-08-11 Standard Chem & Pharm Co Ltd 阿朴芬化合物及其醫藥用途
CN105315208A (zh) * 2014-07-17 2016-02-10 中国科学院兰州化学物理研究所 阿朴菲类生物碱及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3131191A (en) * 1962-08-08 1964-04-28 Smith Kline French Lab Process for the preparation of noraporphines

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2412534A1 (fr) * 1977-12-22 1979-07-20 Warner Lambert Co Preparation de derives de 1-hydroxyaporphines

Also Published As

Publication number Publication date
CH629782A5 (de) 1982-05-14
AU508171B2 (en) 1980-03-13
DE2625116C2 (de) 1984-01-26
FR2353534B1 (fr) 1980-03-07
SE7706488L (sv) 1977-12-05
JPS535169A (en) 1978-01-18
AU2580977A (en) 1978-12-07
IE44937B1 (en) 1982-05-19
DE2625116A1 (de) 1977-12-22
US4120964A (en) 1978-10-17
IE44937L (en) 1977-12-04
ES459504A1 (es) 1978-05-01
FR2353534A1 (fr) 1977-12-30
SE433212B (sv) 1984-05-14
GB1521020A (en) 1978-08-09
DK248277A (da) 1977-12-05
NL7706180A (nl) 1977-12-06
LU77482A1 (fr) 1977-09-22

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: WARNER-LAMBERT CY

Effective date: 19850603