BE847011A - Pyrido (2,1-b) quinazolin-ones et leur procede de preparation - Google Patents
Pyrido (2,1-b) quinazolin-ones et leur procede de preparationInfo
- Publication number
- BE847011A BE847011A BE6045706A BE6045706A BE847011A BE 847011 A BE847011 A BE 847011A BE 6045706 A BE6045706 A BE 6045706A BE 6045706 A BE6045706 A BE 6045706A BE 847011 A BE847011 A BE 847011A
- Authority
- BE
- Belgium
- Prior art keywords
- quinazolin
- pyrido
- ones
- preparation process
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/620,471 US4033961A (en) | 1975-10-07 | 1975-10-07 | Pyrido[2-1-b]quinazolin-ones and their methods of preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
BE847011A true BE847011A (fr) | 1977-04-06 |
Family
ID=24486085
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE6045706A BE847011A (fr) | 1975-10-07 | 1976-10-06 | Pyrido (2,1-b) quinazolin-ones et leur procede de preparation |
Country Status (15)
Country | Link |
---|---|
US (2) | US4033961A (sv) |
JP (1) | JPS5246099A (sv) |
AU (1) | AU500196B2 (sv) |
BE (1) | BE847011A (sv) |
CA (1) | CA1197843A (sv) |
CH (1) | CH605954A5 (sv) |
DE (1) | DE2645110C2 (sv) |
DK (1) | DK450776A (sv) |
ES (3) | ES452441A1 (sv) |
FR (1) | FR2326924A1 (sv) |
GB (1) | GB1512299A (sv) |
IE (1) | IE46232B1 (sv) |
LU (1) | LU75943A1 (sv) |
NL (1) | NL7611126A (sv) |
SE (1) | SE434398B (sv) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4395549A (en) | 1981-10-02 | 1983-07-26 | Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. | 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2557425C2 (de) * | 1975-12-19 | 1987-03-19 | C.H. Boehringer Sohn, 6507 Ingelheim | 11-Oxo-11-H-pyrido[2,1-b]-chinazolin-2-carbonsäure und ihre Salze, Verfahren zu ihrer Herstellung und Arzneimittel |
US4066767A (en) * | 1976-11-01 | 1978-01-03 | Warner-Lambert Company | 8-(1H-Tetrazol-5-yl)-11H-pyrido[2,1-b]quinazolin-11-ones and method of treating bronchial asthma using them |
DE2720085A1 (de) * | 1977-05-05 | 1978-11-16 | Hoechst Ag | Pyrimido(6,1-a)isochinolin-2-on- derivate |
FR2384770A1 (fr) * | 1977-03-24 | 1978-10-20 | Hoffmann La Roche | Nouveaux derives de quinazoline utiles comme medicaments |
HU182009B (en) * | 1977-08-19 | 1983-12-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing substituted pirido-square bracket-1,2-a-square bracket closed-pyrimidines, pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines |
DE2739020A1 (de) | 1977-08-26 | 1979-03-01 | Schering Ag | Pyrido eckige klammer auf 2,1-b eckige klammer zu -chinazolinon-derivate, ihre herstellung und verwendung |
US4127720A (en) * | 1977-09-21 | 1978-11-28 | Bristol-Myers Company | Pyrimido[2,1-a]isoquinoline derivatives having antiallergy activity |
US4348396A (en) * | 1978-01-23 | 1982-09-07 | Hoffmann-La Roche Inc. | Substituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with them |
US4491587A (en) * | 1978-05-05 | 1985-01-01 | Mead Johnson & Company | Tetrazole derivatives |
US4223031A (en) * | 1978-05-05 | 1980-09-16 | Mead Johnson & Company | Azolopyrimidinones |
DE2845766A1 (de) * | 1978-10-18 | 1980-04-30 | Schering Ag | Pyrido eckige klammer auf 2,1-b eckige klammer zu -chinazolinon-derivate, ihre herstellung und verwendung |
US4261996A (en) * | 1980-01-11 | 1981-04-14 | Warner-Lambert Company | Pyrazolo[5,1-b]quinazolin-9-(4H)-ones and anti-allergic pharmaceutical compositions containing them |
US4261997A (en) * | 1980-01-11 | 1981-04-14 | Warner-Lambert Company | 4-Alkyl-pyrazolo[5,1-b]-quinazolin-9(4H)-ones and anti-allergic compositions containing them |
US4247555A (en) * | 1980-01-11 | 1981-01-27 | Warner-Lambert Company | 4,9-Dihydro-9-oxo-N-1H-tetrazol-5-yl-pyrazolo[5,1-b]-quinazoline-2-carboxamides and antiallergic compositions and methods using them |
JPS55134807A (en) * | 1979-04-06 | 1980-10-21 | Hitachi Ltd | Production of color filter |
JPS55138839A (en) * | 1979-04-17 | 1980-10-30 | Nec Kyushu Ltd | Method of fabricating semiconductor device |
JPS574012A (en) * | 1980-06-09 | 1982-01-09 | Canon Inc | Production of color filter |
JPS587608A (ja) * | 1981-07-08 | 1983-01-17 | Hitachi Ltd | カラ−フイルタの製造方法 |
ES8406476A1 (es) * | 1982-04-29 | 1984-07-01 | Erba Farmitalia | Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas. |
US4551460A (en) * | 1982-05-10 | 1985-11-05 | Hoffmann-La Roche Inc. | Pyrido[2,1-b]quinazoline derivatives useful as agents for treatment of allergic conditions and vascular disorders involving thrombosis |
ES524262A0 (es) * | 1982-08-05 | 1984-11-16 | Erba Farmitalia | "procedimiento para preparar derivados de quinazolina" |
JPS5950411A (ja) * | 1982-09-17 | 1984-03-23 | Matsushita Electric Ind Co Ltd | 色フイルタの製造方法 |
FR2533567A1 (fr) * | 1982-09-23 | 1984-03-30 | Ki I Farmakologii | 2-(orthocarboxyphenylamino)-6h-pyrimido (2,1-b)-quinazolone-6 et ses derives, leur procede de preparation et leur application therapeutique |
DE3300477A1 (de) * | 1983-01-08 | 1984-07-12 | Boehringer Ingelheim KG, 6507 Ingelheim | Neue heterocyclische verbindungen, ihre herstellung und verwendung |
GB8331228D0 (en) * | 1983-11-23 | 1983-12-29 | Fujisawa Pharmaceutical Co | Pyrimidoisoquinoline derivatives |
US5914327A (en) * | 1996-11-26 | 1999-06-22 | American Cyanamid Company | Biaryl-pyridoquinazolinone derivatives as anti-cancer agents |
US5908840A (en) * | 1996-11-26 | 1999-06-01 | American Cyanamid Company | Hetero-biaryl-pyridoquinazolinone derivatives as anti-cancer agents |
JP2018019062A (ja) * | 2016-07-27 | 2018-02-01 | サムソン エレクトロ−メカニックス カンパニーリミテッド. | インダクタ |
-
1975
- 1975-10-07 US US05/620,471 patent/US4033961A/en not_active Expired - Lifetime
-
1976
- 1976-09-28 IE IE2143/76A patent/IE46232B1/en unknown
- 1976-10-06 GB GB41459/76A patent/GB1512299A/en not_active Expired
- 1976-10-06 AU AU18420/76A patent/AU500196B2/en not_active Expired
- 1976-10-06 DE DE2645110A patent/DE2645110C2/de not_active Expired
- 1976-10-06 BE BE6045706A patent/BE847011A/xx not_active IP Right Cessation
- 1976-10-06 LU LU75943A patent/LU75943A1/xx unknown
- 1976-10-06 DK DK450776A patent/DK450776A/da not_active Application Discontinuation
- 1976-10-06 FR FR7630050A patent/FR2326924A1/fr active Granted
- 1976-10-07 CA CA000263758A patent/CA1197843A/en not_active Expired
- 1976-10-07 NL NL7611126A patent/NL7611126A/xx not_active Application Discontinuation
- 1976-10-07 SE SE7611169A patent/SE434398B/sv unknown
- 1976-10-07 JP JP51120800A patent/JPS5246099A/ja active Granted
- 1976-10-07 CH CH1270776A patent/CH605954A5/xx not_active IP Right Cessation
- 1976-10-15 ES ES452441A patent/ES452441A1/es not_active Expired
-
1977
- 1977-03-07 US US05/775,015 patent/US4104389A/en not_active Expired - Lifetime
-
1978
- 1978-03-31 ES ES468447A patent/ES468447A1/es not_active Expired
- 1978-03-31 ES ES468448A patent/ES468448A1/es not_active Expired
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4395549A (en) | 1981-10-02 | 1983-07-26 | Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. | 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones |
Also Published As
Publication number | Publication date |
---|---|
ES468448A1 (es) | 1978-12-16 |
SE434398B (sv) | 1984-07-23 |
US4033961A (en) | 1977-07-05 |
CH605954A5 (sv) | 1978-10-13 |
FR2326924B1 (sv) | 1980-07-04 |
ES468447A1 (es) | 1978-12-16 |
ES452441A1 (es) | 1978-08-16 |
AU1842076A (en) | 1978-04-13 |
DK450776A (da) | 1977-04-08 |
US4104389A (en) | 1978-08-01 |
IE46232B1 (en) | 1983-04-06 |
LU75943A1 (sv) | 1977-05-06 |
IE46232L (en) | 1977-04-07 |
DE2645110C2 (de) | 1982-11-18 |
FR2326924A1 (fr) | 1977-05-06 |
JPS5246099A (en) | 1977-04-12 |
CA1197843A (en) | 1985-12-10 |
NL7611126A (nl) | 1977-04-13 |
GB1512299A (en) | 1978-06-01 |
DE2645110A1 (de) | 1977-04-21 |
AU500196B2 (en) | 1979-05-10 |
SE7611169L (sv) | 1977-04-08 |
JPS5526144B2 (sv) | 1980-07-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: WARNER-LAMBERT CY Effective date: 19861031 |