BE834051A - NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINES - Google Patents
NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINESInfo
- Publication number
- BE834051A BE834051A BE160578A BE160578A BE834051A BE 834051 A BE834051 A BE 834051A BE 160578 A BE160578 A BE 160578A BE 160578 A BE160578 A BE 160578A BE 834051 A BE834051 A BE 834051A
- Authority
- BE
- Belgium
- Prior art keywords
- new
- imidazolidines
- phenylimino
- disubstituted
- medicines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE2446758A DE2446758C3 (en) | 1974-10-01 | 1974-10-01 | 2- (2-Fluoro-6-trifluoromethylphenylimino) -imidazolidine, its acid addition salts, processes for the preparation of these compounds and their use in combating hypertension |
Publications (1)
Publication Number | Publication Date |
---|---|
BE834051A true BE834051A (en) | 1976-03-30 |
Family
ID=5927202
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE160578A BE834051A (en) | 1974-10-01 | 1975-09-30 | NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINES |
Country Status (27)
Country | Link |
---|---|
JP (1) | JPS6018653B2 (en) |
AT (1) | AT344159B (en) |
BE (1) | BE834051A (en) |
BG (2) | BG25220A3 (en) |
CA (1) | CA1056836A (en) |
CH (5) | CH620682A5 (en) |
CS (1) | CS193524B2 (en) |
DD (1) | DD123602A5 (en) |
DE (1) | DE2446758C3 (en) |
DK (1) | DK441875A (en) |
ES (4) | ES441385A1 (en) |
FI (1) | FI61883C (en) |
FR (1) | FR2286649A1 (en) |
GB (1) | GB1515019A (en) |
HU (1) | HU178469B (en) |
IE (1) | IE42130B1 (en) |
IL (1) | IL48214A (en) |
LU (1) | LU73472A1 (en) |
NL (1) | NL7511490A (en) |
NO (1) | NO143459C (en) |
NZ (1) | NZ178810A (en) |
PH (1) | PH13653A (en) |
PL (2) | PL98984B1 (en) |
SE (1) | SE418497B (en) |
SU (1) | SU575026A3 (en) |
YU (1) | YU230281A (en) |
ZA (1) | ZA756185B (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2630060C2 (en) * | 1976-07-03 | 1984-04-19 | C.H. Boehringer Sohn, 6507 Ingelheim | 2- (2-Bromo-6-fluoro-phenylimino) -imidazolidine, its acid addition salts, medicaments containing them and processes for their preparation |
DE2806775A1 (en) * | 1978-02-17 | 1979-08-30 | Boehringer Sohn Ingelheim | NEW SUBSTITUTED 2-PHENYLIMINO IMIDAZOLIDINE THEIR ACID ADDITION SALTS, MEDICINAL PRODUCTS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF |
DE2806811A1 (en) * | 1978-02-17 | 1979-08-23 | Boehringer Sohn Ingelheim | NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME |
CA1138451A (en) * | 1979-04-03 | 1982-12-28 | Ikuo Ueda | 2-imidazoline derivatives, process for the preparation thereof and the pharmaceutical composition of the same |
HU192986B (en) * | 1984-05-23 | 1987-08-28 | Egyt Gyogyszervegyeszeti Gyar | Process for production of imidasodiline derivatives |
AU2007213887A1 (en) * | 2006-01-27 | 2007-08-16 | F. Hoffmann-La Roche Ag | Use of 2-imidazoles for the treatment of CNS disorders |
CA2675221C (en) | 2007-02-02 | 2016-02-23 | F. Hoffmann-La Roche Ag | Novel 2-aminooxazolines as taar1 ligands |
KR101222412B1 (en) | 2007-02-15 | 2013-01-15 | 에프. 호프만-라 로슈 아게 | 2-aminooxazolines as taar1 ligands |
US8242153B2 (en) | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
US8354441B2 (en) | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
AU2017234042B2 (en) | 2016-03-17 | 2020-11-19 | F. Hoffmann-La Roche Ag | 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of TAAR |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3236857A (en) * | 1961-10-09 | 1966-02-22 | Boehringer Sohn Ingelheim | 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products |
DE1670807A1 (en) * | 1967-02-17 | 1971-03-11 | Bayer Ag | Process for the preparation of cyclic guanidines |
DE1670918A1 (en) * | 1967-09-07 | 1971-04-08 | Bayer Ag | Process for the preparation of 2-aryl-amino-substituted nitrogen-containing heterocycles |
BE787683A (en) * | 1971-08-20 | 1973-02-19 | Boehringer Sohn Ingelheim | 2-PHENYLIMINO-IMIDAZOLIDINES, THEIR ADDITIONAL SALTS WITH ACIDS AND METHODS FOR MAKING THEM |
-
1974
- 1974-10-01 DE DE2446758A patent/DE2446758C3/en not_active Expired
-
1975
- 1975-09-22 AT AT722875A patent/AT344159B/en not_active IP Right Cessation
- 1975-09-23 SU SU7502174605A patent/SU575026A3/en active
- 1975-09-26 PH PH17613A patent/PH13653A/en unknown
- 1975-09-29 CS CS756573A patent/CS193524B2/en unknown
- 1975-09-29 BG BG7500031110A patent/BG25220A3/en unknown
- 1975-09-29 LU LU73472A patent/LU73472A1/xx unknown
- 1975-09-29 DD DD188613A patent/DD123602A5/xx unknown
- 1975-09-29 BG BG7500032014A patent/BG25221A3/en unknown
- 1975-09-30 PL PL1975197816A patent/PL98984B1/en unknown
- 1975-09-30 PL PL1975183670A patent/PL97003B1/en unknown
- 1975-09-30 NZ NZ178810A patent/NZ178810A/en unknown
- 1975-09-30 NO NO753314A patent/NO143459C/en unknown
- 1975-09-30 ZA ZA756185A patent/ZA756185B/en unknown
- 1975-09-30 BE BE160578A patent/BE834051A/en not_active IP Right Cessation
- 1975-09-30 DK DK441875A patent/DK441875A/en not_active Application Discontinuation
- 1975-09-30 IL IL48214A patent/IL48214A/en unknown
- 1975-09-30 CH CH1267875A patent/CH620682A5/en not_active IP Right Cessation
- 1975-09-30 CA CA236,670A patent/CA1056836A/en not_active Expired
- 1975-09-30 ES ES441385A patent/ES441385A1/en not_active Expired
- 1975-09-30 FI FI752728A patent/FI61883C/en not_active IP Right Cessation
- 1975-09-30 JP JP50118196A patent/JPS6018653B2/en not_active Expired
- 1975-09-30 GB GB40012/75A patent/GB1515019A/en not_active Expired
- 1975-09-30 HU HU75BO1573A patent/HU178469B/en unknown
- 1975-09-30 NL NL7511490A patent/NL7511490A/en not_active Application Discontinuation
- 1975-10-01 FR FR7530117A patent/FR2286649A1/en active Granted
- 1975-10-01 IE IE2150/75A patent/IE42130B1/en unknown
- 1975-10-01 SE SE7511028A patent/SE418497B/en not_active IP Right Cessation
-
1976
- 1976-02-04 ES ES444901A patent/ES444901A1/en not_active Expired
- 1976-02-04 ES ES444900A patent/ES444900A1/en not_active Expired
- 1976-02-04 ES ES444898A patent/ES444898A1/en not_active Expired
-
1980
- 1980-07-01 CH CH506280A patent/CH627452A5/en not_active IP Right Cessation
- 1980-07-01 CH CH506580A patent/CH627454A5/en not_active IP Right Cessation
- 1980-07-01 CH CH506380A patent/CH627453A5/en not_active IP Right Cessation
- 1980-07-01 CH CH506480A patent/CH626352A5/en not_active IP Right Cessation
-
1981
- 1981-09-24 YU YU02302/81A patent/YU230281A/en unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: C.H. BOEHRINGER SOHN Effective date: 19880930 |