BE834051A - NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINES - Google Patents

NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINES

Info

Publication number
BE834051A
BE834051A BE160578A BE160578A BE834051A BE 834051 A BE834051 A BE 834051A BE 160578 A BE160578 A BE 160578A BE 160578 A BE160578 A BE 160578A BE 834051 A BE834051 A BE 834051A
Authority
BE
Belgium
Prior art keywords
new
imidazolidines
phenylimino
disubstituted
medicines
Prior art date
Application number
BE160578A
Other languages
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE834051A publication Critical patent/BE834051A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • C07D233/50Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BE160578A 1974-10-01 1975-09-30 NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINES BE834051A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2446758A DE2446758C3 (en) 1974-10-01 1974-10-01 2- (2-Fluoro-6-trifluoromethylphenylimino) -imidazolidine, its acid addition salts, processes for the preparation of these compounds and their use in combating hypertension

Publications (1)

Publication Number Publication Date
BE834051A true BE834051A (en) 1976-03-30

Family

ID=5927202

Family Applications (1)

Application Number Title Priority Date Filing Date
BE160578A BE834051A (en) 1974-10-01 1975-09-30 NEW 2-PHENYLIMINO-IMIDAZOLIDINES, DISUBSTITUTED IN 2 AND 6, THEIR ADDITIONAL SALTS WITH ACIDS, MEDICINAL PRODUCTS BASED ON THESE NEW COMPOUNDS AND METHODS FOR MANUFACTURING THESE MEDICINES

Country Status (27)

Country Link
JP (1) JPS6018653B2 (en)
AT (1) AT344159B (en)
BE (1) BE834051A (en)
BG (2) BG25220A3 (en)
CA (1) CA1056836A (en)
CH (5) CH620682A5 (en)
CS (1) CS193524B2 (en)
DD (1) DD123602A5 (en)
DE (1) DE2446758C3 (en)
DK (1) DK441875A (en)
ES (4) ES441385A1 (en)
FI (1) FI61883C (en)
FR (1) FR2286649A1 (en)
GB (1) GB1515019A (en)
HU (1) HU178469B (en)
IE (1) IE42130B1 (en)
IL (1) IL48214A (en)
LU (1) LU73472A1 (en)
NL (1) NL7511490A (en)
NO (1) NO143459C (en)
NZ (1) NZ178810A (en)
PH (1) PH13653A (en)
PL (2) PL98984B1 (en)
SE (1) SE418497B (en)
SU (1) SU575026A3 (en)
YU (1) YU230281A (en)
ZA (1) ZA756185B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2630060C2 (en) * 1976-07-03 1984-04-19 C.H. Boehringer Sohn, 6507 Ingelheim 2- (2-Bromo-6-fluoro-phenylimino) -imidazolidine, its acid addition salts, medicaments containing them and processes for their preparation
DE2806775A1 (en) * 1978-02-17 1979-08-30 Boehringer Sohn Ingelheim NEW SUBSTITUTED 2-PHENYLIMINO IMIDAZOLIDINE THEIR ACID ADDITION SALTS, MEDICINAL PRODUCTS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF
DE2806811A1 (en) * 1978-02-17 1979-08-23 Boehringer Sohn Ingelheim NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME
CA1138451A (en) * 1979-04-03 1982-12-28 Ikuo Ueda 2-imidazoline derivatives, process for the preparation thereof and the pharmaceutical composition of the same
HU192986B (en) * 1984-05-23 1987-08-28 Egyt Gyogyszervegyeszeti Gyar Process for production of imidasodiline derivatives
AU2007213887A1 (en) * 2006-01-27 2007-08-16 F. Hoffmann-La Roche Ag Use of 2-imidazoles for the treatment of CNS disorders
CA2675221C (en) 2007-02-02 2016-02-23 F. Hoffmann-La Roche Ag Novel 2-aminooxazolines as taar1 ligands
KR101222412B1 (en) 2007-02-15 2013-01-15 에프. 호프만-라 로슈 아게 2-aminooxazolines as taar1 ligands
US8242153B2 (en) 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
US8354441B2 (en) 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
AU2017234042B2 (en) 2016-03-17 2020-11-19 F. Hoffmann-La Roche Ag 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of TAAR

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3236857A (en) * 1961-10-09 1966-02-22 Boehringer Sohn Ingelheim 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products
DE1670807A1 (en) * 1967-02-17 1971-03-11 Bayer Ag Process for the preparation of cyclic guanidines
DE1670918A1 (en) * 1967-09-07 1971-04-08 Bayer Ag Process for the preparation of 2-aryl-amino-substituted nitrogen-containing heterocycles
BE787683A (en) * 1971-08-20 1973-02-19 Boehringer Sohn Ingelheim 2-PHENYLIMINO-IMIDAZOLIDINES, THEIR ADDITIONAL SALTS WITH ACIDS AND METHODS FOR MAKING THEM

Also Published As

Publication number Publication date
SU575026A3 (en) 1977-09-30
JPS5159863A (en) 1976-05-25
DE2446758A1 (en) 1976-04-22
ES444898A1 (en) 1977-05-16
LU73472A1 (en) 1977-05-16
FI61883C (en) 1982-10-11
FI752728A (en) 1976-04-02
CH627453A5 (en) 1982-01-15
CH626352A5 (en) 1981-11-13
NO143459B (en) 1980-11-10
HU178469B (en) 1982-05-28
DE2446758B2 (en) 1978-05-18
CS193524B2 (en) 1979-10-31
BG25220A3 (en) 1978-08-10
ATA722875A (en) 1977-11-15
PL98984B1 (en) 1978-06-30
CH627452A5 (en) 1982-01-15
ZA756185B (en) 1977-06-29
JPS6018653B2 (en) 1985-05-11
ES444901A1 (en) 1977-04-16
DK441875A (en) 1976-04-02
PL97003B1 (en) 1978-01-31
AU8529875A (en) 1977-04-07
NO143459C (en) 1981-02-18
IL48214A0 (en) 1975-11-25
IE42130B1 (en) 1980-06-04
CH620682A5 (en) 1980-12-15
NO753314L (en) 1976-04-02
NZ178810A (en) 1978-04-03
GB1515019A (en) 1978-06-21
ES444900A1 (en) 1977-04-16
SE7511028L (en) 1976-04-02
FR2286649B1 (en) 1979-09-14
BG25221A3 (en) 1978-08-10
YU230281A (en) 1982-02-28
FR2286649A1 (en) 1976-04-30
FI61883B (en) 1982-06-30
NL7511490A (en) 1976-04-05
ES441385A1 (en) 1977-08-01
AT344159B (en) 1978-07-10
CH627454A5 (en) 1982-01-15
DE2446758C3 (en) 1979-01-04
PH13653A (en) 1980-08-21
IL48214A (en) 1979-10-31
CA1056836A (en) 1979-06-19
SE418497B (en) 1981-06-09
IE42130L (en) 1976-04-01
DD123602A5 (en) 1977-01-05

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: C.H. BOEHRINGER SOHN

Effective date: 19880930