NL7511490A - PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS. - Google Patents

PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS.

Info

Publication number
NL7511490A
NL7511490A NL7511490A NL7511490A NL7511490A NL 7511490 A NL7511490 A NL 7511490A NL 7511490 A NL7511490 A NL 7511490A NL 7511490 A NL7511490 A NL 7511490A NL 7511490 A NL7511490 A NL 7511490A
Authority
NL
Netherlands
Prior art keywords
phenyliminoimidazolidins
substituted
digital
preparation
new
Prior art date
Application number
NL7511490A
Other languages
Dutch (nl)
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of NL7511490A publication Critical patent/NL7511490A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • C07D233/50Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NL7511490A 1974-10-01 1975-09-30 PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS. NL7511490A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2446758A DE2446758C3 (en) 1974-10-01 1974-10-01 2- (2-Fluoro-6-trifluoromethylphenylimino) -imidazolidine, its acid addition salts, processes for the preparation of these compounds and their use in combating hypertension

Publications (1)

Publication Number Publication Date
NL7511490A true NL7511490A (en) 1976-04-05

Family

ID=5927202

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7511490A NL7511490A (en) 1974-10-01 1975-09-30 PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS.

Country Status (27)

Country Link
JP (1) JPS6018653B2 (en)
AT (1) AT344159B (en)
BE (1) BE834051A (en)
BG (2) BG25220A3 (en)
CA (1) CA1056836A (en)
CH (5) CH620682A5 (en)
CS (1) CS193524B2 (en)
DD (1) DD123602A5 (en)
DE (1) DE2446758C3 (en)
DK (1) DK441875A (en)
ES (4) ES441385A1 (en)
FI (1) FI61883C (en)
FR (1) FR2286649A1 (en)
GB (1) GB1515019A (en)
HU (1) HU178469B (en)
IE (1) IE42130B1 (en)
IL (1) IL48214A (en)
LU (1) LU73472A1 (en)
NL (1) NL7511490A (en)
NO (1) NO143459C (en)
NZ (1) NZ178810A (en)
PH (1) PH13653A (en)
PL (2) PL97003B1 (en)
SE (1) SE418497B (en)
SU (1) SU575026A3 (en)
YU (1) YU230281A (en)
ZA (1) ZA756185B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2630060C2 (en) * 1976-07-03 1984-04-19 C.H. Boehringer Sohn, 6507 Ingelheim 2- (2-Bromo-6-fluoro-phenylimino) -imidazolidine, its acid addition salts, medicaments containing them and processes for their preparation
DE2806811A1 (en) * 1978-02-17 1979-08-23 Boehringer Sohn Ingelheim NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME
DE2806775A1 (en) * 1978-02-17 1979-08-30 Boehringer Sohn Ingelheim NEW SUBSTITUTED 2-PHENYLIMINO IMIDAZOLIDINE THEIR ACID ADDITION SALTS, MEDICINAL PRODUCTS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF
CA1138451A (en) * 1979-04-03 1982-12-28 Ikuo Ueda 2-imidazoline derivatives, process for the preparation thereof and the pharmaceutical composition of the same
HU192986B (en) * 1984-05-23 1987-08-28 Egyt Gyogyszervegyeszeti Gyar Process for production of imidasodiline derivatives
KR20080090546A (en) * 2006-01-27 2008-10-08 에프. 호프만-라 로슈 아게 Use of 2-imidazoles for the treatment of cns disorders
CA2675221C (en) 2007-02-02 2016-02-23 F. Hoffmann-La Roche Ag Novel 2-aminooxazolines as taar1 ligands
CA2676944C (en) 2007-02-15 2016-01-19 F. Hoffmann-La Roche Ag 2-aminooxazolines as taar1 ligands
US8242153B2 (en) 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
US8354441B2 (en) 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
LT3430010T (en) 2016-03-17 2020-10-12 F. Hoffmann-La Roche Ag 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3236857A (en) * 1961-10-09 1966-02-22 Boehringer Sohn Ingelheim 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products
DE1670807A1 (en) * 1967-02-17 1971-03-11 Bayer Ag Process for the preparation of cyclic guanidines
DE1670918A1 (en) * 1967-09-07 1971-04-08 Bayer Ag Process for the preparation of 2-aryl-amino-substituted nitrogen-containing heterocycles
BE787683A (en) * 1971-08-20 1973-02-19 Boehringer Sohn Ingelheim 2-PHENYLIMINO-IMIDAZOLIDINES, THEIR ADDITIONAL SALTS WITH ACIDS AND METHODS FOR MAKING THEM

Also Published As

Publication number Publication date
SE7511028L (en) 1976-04-02
FR2286649A1 (en) 1976-04-30
ES444900A1 (en) 1977-04-16
BE834051A (en) 1976-03-30
IL48214A (en) 1979-10-31
CA1056836A (en) 1979-06-19
FI752728A (en) 1976-04-02
SU575026A3 (en) 1977-09-30
ES441385A1 (en) 1977-08-01
IL48214A0 (en) 1975-11-25
DE2446758B2 (en) 1978-05-18
HU178469B (en) 1982-05-28
BG25221A3 (en) 1978-08-10
DE2446758A1 (en) 1976-04-22
YU230281A (en) 1982-02-28
ATA722875A (en) 1977-11-15
FI61883C (en) 1982-10-11
GB1515019A (en) 1978-06-21
PH13653A (en) 1980-08-21
IE42130L (en) 1976-04-01
NO143459B (en) 1980-11-10
AU8529875A (en) 1977-04-07
SE418497B (en) 1981-06-09
ES444898A1 (en) 1977-05-16
FI61883B (en) 1982-06-30
ZA756185B (en) 1977-06-29
FR2286649B1 (en) 1979-09-14
NO143459C (en) 1981-02-18
CH627454A5 (en) 1982-01-15
NZ178810A (en) 1978-04-03
ES444901A1 (en) 1977-04-16
NO753314L (en) 1976-04-02
PL97003B1 (en) 1978-01-31
JPS5159863A (en) 1976-05-25
IE42130B1 (en) 1980-06-04
CS193524B2 (en) 1979-10-31
PL98984B1 (en) 1978-06-30
DE2446758C3 (en) 1979-01-04
LU73472A1 (en) 1977-05-16
CH620682A5 (en) 1980-12-15
JPS6018653B2 (en) 1985-05-11
CH626352A5 (en) 1981-11-13
CH627452A5 (en) 1982-01-15
DK441875A (en) 1976-04-02
DD123602A5 (en) 1977-01-05
BG25220A3 (en) 1978-08-10
CH627453A5 (en) 1982-01-15
AT344159B (en) 1978-07-10

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Legal Events

Date Code Title Description
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
A85 Still pending on 85-01-01
BV The patent application has lapsed