BE828440A - Procede de production de 3-oxydes de 6-amino-2,4-diamino-pyrimidines et de leurs intermediaires, et produits obtenus - Google Patents

Procede de production de 3-oxydes de 6-amino-2,4-diamino-pyrimidines et de leurs intermediaires, et produits obtenus

Info

Publication number
BE828440A
BE828440A BE155822A BE155822A BE828440A BE 828440 A BE828440 A BE 828440A BE 155822 A BE155822 A BE 155822A BE 155822 A BE155822 A BE 155822A BE 828440 A BE828440 A BE 828440A
Authority
BE
Belgium
Prior art keywords
intermediaries
diamino
pyrimidine
oxides
amino
Prior art date
Application number
BE155822A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE828440A publication Critical patent/BE828440A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/195Radicals derived from nitrogen analogues of carboxylic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms
BE155822A 1974-04-26 1975-04-25 Procede de production de 3-oxydes de 6-amino-2,4-diamino-pyrimidines et de leurs intermediaires, et produits obtenus BE828440A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US464476A US3910928A (en) 1974-04-26 1974-04-26 3-(Cyanimino)-propionitriles

Publications (1)

Publication Number Publication Date
BE828440A true BE828440A (fr) 1975-10-27

Family

ID=23844086

Family Applications (1)

Application Number Title Priority Date Filing Date
BE155822A BE828440A (fr) 1974-04-26 1975-04-25 Procede de production de 3-oxydes de 6-amino-2,4-diamino-pyrimidines et de leurs intermediaires, et produits obtenus

Country Status (16)

Country Link
US (1) US3910928A (sv)
JP (2) JPS6039670B2 (sv)
BE (1) BE828440A (sv)
CA (1) CA1038388A (sv)
CH (2) CH612924A5 (sv)
DE (1) DE2516868C2 (sv)
DK (1) DK157293C (sv)
ES (1) ES436654A1 (sv)
FR (1) FR2270250B1 (sv)
GB (1) GB1450010A (sv)
HU (2) HU172103B (sv)
IL (1) IL46897A (sv)
NL (1) NL182562C (sv)
SE (1) SE458766B (sv)
SU (2) SU645570A3 (sv)
ZA (1) ZA752076B (sv)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4032559A (en) * 1975-07-28 1977-06-28 The Upjohn Company N,2-dicyanoacetimidates
CH638216A5 (de) * 1977-02-04 1983-09-15 Hoffmann La Roche Oxadiazolopyrimidin-deriate.
US4098791A (en) * 1977-07-29 1978-07-04 The Upjohn Company Process for preparing 3-(cyanimino)-3-amino-propionitriles
CA1103245A (en) * 1978-07-21 1981-06-16 Jean-Claude Muller Process for the manufacture of novel oxadiazolopyrimidine derivatives
EP0042669A3 (en) * 1980-06-23 1982-03-24 The Upjohn Company Compounds and compositions for use in animal feeds
US4308271A (en) * 1980-06-23 1981-12-29 The Upjohn Company Animal feed and process
JPS5973573A (ja) * 1982-09-09 1984-04-25 ワ−ナ−−ランバ−ト・コンパニ− ジアミノピリミジン化合物
LU86695A1 (fr) * 1986-12-01 1988-07-14 Oreal Nouveaux derives de piperazinyl-1 pyrimidine,leur preparation et leur application en therapeutique et cosmetique
LU86960A1 (fr) * 1987-07-31 1989-03-08 Oreal Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux
US5272164A (en) * 1988-12-27 1993-12-21 Kirin Beer Kabushiki Kaisha Carboximidamide derivatives
JPH0662567B2 (ja) * 1988-12-27 1994-08-17 麒麟麦酒株式会社 ピリジンカルボキシイミダミド誘導体、その製造中間体、製造法および用途
US4959475A (en) * 1989-01-04 1990-09-25 Lonza Ltd. Process for the production of 2,4-diamino-6-piperidinyl-pyrimidine-3-N-oxide
FR2671082B1 (fr) * 1990-12-28 1993-04-16 Oreal Agent a plusieurs composants ou kit de preparation de la forme sulfo-conjuguee de composes pyrimidino- ou triazino-n-oxyde et procede de mise en óoeuvre.
EP1408025B1 (en) * 2001-06-12 2007-11-21 Ube Industries, Ltd. 3,3-dialkoxy-2-hydroxyiminopropionitriles, process for preparation thereof and process of preparing 5-amino -4-nitrosopyrazoles or salts thereof by the use of the same
CN111018838B (zh) * 2019-11-25 2022-12-27 重庆东寰科技开发有限公司 吡咯烷基二氨基嘧啶氮氧化物的合成方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3461461A (en) * 1965-11-01 1969-08-12 Upjohn Co 6-amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidines

Also Published As

Publication number Publication date
IL46897A0 (en) 1975-05-22
US3910928A (en) 1975-10-07
JPS6039670B2 (ja) 1985-09-06
JPS50148367A (sv) 1975-11-27
DE2516868C2 (de) 1986-10-23
HU172103B (hu) 1978-05-28
NL182562C (nl) 1988-04-05
CA1038388A (en) 1978-09-12
SE458766B (sv) 1989-05-08
DE2516868A1 (de) 1975-11-13
AU7981875A (en) 1976-10-07
JPH0219829B2 (sv) 1990-05-07
DK157293C (da) 1990-05-07
GB1450010A (en) 1976-09-22
ES436654A1 (es) 1977-01-01
IL46897A (en) 1979-10-31
SU584770A3 (ru) 1977-12-15
FR2270250A1 (sv) 1975-12-05
SE7504762L (sv) 1975-10-27
CH612924A5 (sv) 1979-08-31
JPS60190753A (ja) 1985-09-28
DK179675A (da) 1975-10-27
HU170090B (sv) 1977-03-28
ZA752076B (en) 1976-03-31
CH616158A5 (sv) 1980-03-14
FR2270250B1 (sv) 1979-10-05
DK157293B (da) 1989-12-04
NL7504846A (nl) 1975-10-28
SU645570A3 (ru) 1979-01-30
NL182562B (nl) 1987-11-02

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19930430