AU8215098A - Composition comprising 5-(4-(2-(N-methyl-N-2-pyridyl)amino) ethoxy)benzyl)thiazolidine-2,4-dione - Google Patents

Composition comprising 5-(4-(2-(N-methyl-N-2-pyridyl)amino) ethoxy)benzyl)thiazolidine-2,4-dione Download PDF

Info

Publication number
AU8215098A
AU8215098A AU82150/98A AU8215098A AU8215098A AU 8215098 A AU8215098 A AU 8215098A AU 82150/98 A AU82150/98 A AU 82150/98A AU 8215098 A AU8215098 A AU 8215098A AU 8215098 A AU8215098 A AU 8215098A
Authority
AU
Australia
Prior art keywords
pharmaceutically acceptable
compound
composition
acceptable form
composition according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU82150/98A
Other languages
English (en)
Inventor
Jeffrey Roger Granett
Jai Patel
Robin Price
Hamish Ross
Paul Nigel Wray
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Ltd
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9712851.6A external-priority patent/GB9712851D0/en
Application filed by SmithKline Beecham Ltd, SmithKline Beecham Corp filed Critical SmithKline Beecham Ltd
Publication of AU8215098A publication Critical patent/AU8215098A/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
AU82150/98A 1997-06-05 1998-06-02 Composition comprising 5-(4-(2-(N-methyl-N-2-pyridyl)amino) ethoxy)benzyl)thiazolidine-2,4-dione Abandoned AU8215098A (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB9711683.4A GB9711683D0 (en) 1997-06-05 1997-06-05 Composition
GB9711683 1997-06-05
GBGB9712851.6A GB9712851D0 (en) 1997-06-18 1997-06-18 Composition
GB9712851 1997-06-18
PCT/EP1998/003478 WO1998055122A1 (en) 1997-06-05 1998-06-02 Composition comprising 5-[4-[2-(n-methyl-n-2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU95134/01A Division AU9513401A (en) 1997-06-05 2001-11-29 Composition comprising 5-(4-(2-(N-methyl-N-2-pyridyl) amino)ethoxy)benzyl)thiazolidine-2,4-dione

Publications (1)

Publication Number Publication Date
AU8215098A true AU8215098A (en) 1998-12-21

Family

ID=26311662

Family Applications (1)

Application Number Title Priority Date Filing Date
AU82150/98A Abandoned AU8215098A (en) 1997-06-05 1998-06-02 Composition comprising 5-(4-(2-(N-methyl-N-2-pyridyl)amino) ethoxy)benzyl)thiazolidine-2,4-dione

Country Status (29)

Country Link
EP (1) EP0998284A1 (es)
JP (1) JP2001521553A (es)
KR (1) KR20010013410A (es)
CN (3) CN1526391A (es)
AP (1) AP1214A (es)
AR (2) AR008198A1 (es)
AU (1) AU8215098A (es)
BG (1) BG104048A (es)
BR (1) BR9810405A (es)
CA (2) CA2333352A1 (es)
CO (1) CO4940400A1 (es)
DZ (1) DZ2510A1 (es)
EA (1) EA002384B1 (es)
GB (1) GB9711683D0 (es)
HU (1) HUP0004070A3 (es)
ID (1) ID24264A (es)
IL (1) IL133074A0 (es)
MX (1) MXPA99011322A (es)
NO (2) NO995938L (es)
NZ (2) NZ523725A (es)
OA (1) OA11306A (es)
PE (1) PE78899A1 (es)
PL (1) PL337201A1 (es)
SK (1) SK164899A3 (es)
TR (2) TR200002790T2 (es)
TW (1) TW570797B (es)
UY (1) UY25032A1 (es)
WO (1) WO1998055122A1 (es)
ZA (2) ZA9811572B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2203453T3 (es) * 1999-04-23 2004-04-16 Smithkline Beecham Plc Polimorfo de sal del acido maleico de 5-(4-(2-(n-metil-n-(2-piridil)amino)etoxi)bentil)tiazolidina-2,4-diona.
PT1173434E (pt) 1999-04-23 2003-12-31 Smithkline Beecham Plc Novo produto farmaceutico
US20040248945A1 (en) 1999-04-23 2004-12-09 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
GB0021978D0 (en) 2000-09-07 2000-10-25 Smithkline Beecham Plc Novel pharmaceutical
GB0127805D0 (en) * 2001-11-20 2002-01-09 Smithkline Beecham Plc Pharmaceutical composition
AU2002350965A1 (en) * 2001-12-13 2003-06-23 Smithkline Beecham Plc Toluenesulfonate hydrates of a thiazolidinedione derivative
GB0129876D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB0129871D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB0130509D0 (en) * 2001-12-20 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
US7435741B2 (en) 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
EP2270007A1 (en) * 2006-05-09 2011-01-05 Teva Pharmaceutical Industries Ltd. 2-N-{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2-4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
WO2015008234A1 (en) * 2013-07-17 2015-01-22 Glenmark Pharmaceuticals S.A. Bicyclic heterocyclic compounds as ror gamma modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE186724T1 (de) * 1987-09-04 1999-12-15 Beecham Group Plc Substituierte thiazolidindionderivate
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
CA2182986A1 (en) * 1994-02-10 1995-08-17 Smithkline Beecham P.L.C. Use of insulin sensitisers for treating renal diseases
JPH11510508A (ja) * 1995-08-10 1999-09-14 ワーナー−ランバート・コンパニー インシュリン非依存性真性糖尿病患者に投与される外来インシュリンの量を減らす方法
WO1997018811A1 (en) * 1995-11-17 1997-05-29 Warner-Lambert Company A method of treating myotonic dystrophy
NZ314406A (en) * 1996-03-18 2000-12-22 Sankyo Co Treatment or prophylaxis of pancreatitis with a medicament containing an insulin sensitiser including oxazoles and thiazoles
PL331148A1 (en) * 1996-07-12 1999-06-21 Smithkline Beecham Plc Novel method of treating the leptin immunity

Also Published As

Publication number Publication date
CA2333352A1 (en) 1998-12-10
NO20040738L (no) 2000-02-02
IL133074A0 (en) 2001-03-19
CO4940400A1 (es) 2000-07-24
TW570797B (en) 2004-01-11
ID24264A (id) 2000-07-13
PL337201A1 (en) 2000-08-14
DZ2510A1 (fr) 2003-01-25
PE78899A1 (es) 1999-10-22
EA199901116A1 (ru) 2000-06-26
NZ523725A (en) 2004-09-24
NO995938D0 (no) 1999-12-03
AP1214A (en) 2003-10-08
AR008198A1 (es) 1999-12-29
MXPA99011322A (es) 2004-12-02
SK164899A3 (en) 2000-11-07
CN1112926C (zh) 2003-07-02
JP2001521553A (ja) 2001-11-06
ZA9811572B (en) 1999-07-22
BR9810405A (pt) 2000-08-29
EP0998284A1 (en) 2000-05-10
AP9901696A0 (en) 1999-12-31
UY25032A1 (es) 1998-11-26
HUP0004070A2 (hu) 2002-02-28
AR015120A1 (es) 2001-04-18
CA2292629A1 (en) 1998-12-10
TR199902963T2 (xx) 2000-02-21
TR200002790T2 (tr) 2001-11-21
EA002384B1 (ru) 2002-04-25
CA2292629C (en) 2004-01-06
NO995938L (no) 2000-02-02
OA11306A (en) 2003-10-22
BG104048A (bg) 2000-07-31
WO1998055122A1 (en) 1998-12-10
CN1430959A (zh) 2003-07-23
CN1259050A (zh) 2000-07-05
KR20010013410A (ko) 2001-02-26
CN1526391A (zh) 2004-09-08
ZA984826B (en) 1999-08-03
NZ513922A (en) 2001-09-28
HUP0004070A3 (en) 2002-03-28
GB9711683D0 (en) 1997-08-06

Similar Documents

Publication Publication Date Title
SK286029B6 (sk) Farmaceutický prostriedok a jeho použitie
CA2292629C (en) Composition comprising 5-[4-[2-(n-methyl-n-2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione
AP1287A (en) Treatment of diabetes with rosiglitazone and insulin.
US20030187030A1 (en) Composition comprising 5-[4-[2-(N-methyl-N-2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione
EP0999845B1 (en) Treatment of diabetes with thiazolidinedione and sulphonylurea
AU743269B2 (en) Treatment of diabetes with thiazolidinedione and sulphonylurea
US20020028768A1 (en) Treatment of diabetes with rosiglitazone and insulin
SK179499A3 (en) The use of insulin sensitiser and alpha-glucosidase inhibitive antihyperglycaemic agent
AU9513401A (en) Composition comprising 5-(4-(2-(N-methyl-N-2-pyridyl) amino)ethoxy)benzyl)thiazolidine-2,4-dione
AU783539B2 (en) Treatment of diabetes with thiazolidinedione and sulphonylurea
AU778947B2 (en) Treatment of diabetes with thiazolidinedione and metformin
NZ518076A (en) 5-[4-[2-(N-methyl-N-(2- pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione (BRL49653) for treating non-insulin dependent diabetes (NIDDM)
AU1552102A (en) Treatment of diabetes with rosiglitazone and insulin
MXPA99012065A (es) Tratamiento de diabetes con rosiglitazona e insulina
MXPA99012098A (es) Tratamiento de diabetes con tiazolidinodiona e inhibidor de alfa-glucosidasa
NZ520542A (en) Treatment of diabetes with thiazolidinedione and metformin

Legal Events

Date Code Title Description
MK5 Application lapsed section 142(2)(e) - patent request and compl. specification not accepted