AU542692B2 - 1,2,4 triazol-i-yl antifungal agents - Google Patents

1,2,4 triazol-i-yl antifungal agents

Info

Publication number
AU542692B2
AU542692B2 AU17930/83A AU1793083A AU542692B2 AU 542692 B2 AU542692 B2 AU 542692B2 AU 17930/83 A AU17930/83 A AU 17930/83A AU 1793083 A AU1793083 A AU 1793083A AU 542692 B2 AU542692 B2 AU 542692B2
Authority
AU
Australia
Prior art keywords
compound
formula
salt
plc
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU17930/83A
Other languages
English (en)
Other versions
AU1793083A (en
Inventor
Kenneth Richardson
Peter John Whittle
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER CORP
Original Assignee
PFIZER
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER filed Critical PFIZER
Publication of AU1793083A publication Critical patent/AU1793083A/en
Application granted granted Critical
Publication of AU542692B2 publication Critical patent/AU542692B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/004—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reaction with organometalhalides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/04—Saturated compounds containing keto groups bound to acyclic carbon atoms
    • C07C49/16—Saturated compounds containing keto groups bound to acyclic carbon atoms containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AU17930/83A 1982-08-14 1983-08-12 1,2,4 triazol-i-yl antifungal agents Ceased AU542692B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8223459 1982-08-14
GB8223459 1982-08-14
GB8231309 1982-11-02
GB8231309 1982-11-02

Publications (2)

Publication Number Publication Date
AU1793083A AU1793083A (en) 1984-02-16
AU542692B2 true AU542692B2 (en) 1985-03-07

Family

ID=26283600

Family Applications (1)

Application Number Title Priority Date Filing Date
AU17930/83A Ceased AU542692B2 (en) 1982-08-14 1983-08-12 1,2,4 triazol-i-yl antifungal agents

Country Status (22)

Country Link
US (1) US4616027A (enExample)
EP (1) EP0104734B1 (enExample)
KR (1) KR880001046B1 (enExample)
AU (1) AU542692B2 (enExample)
CA (1) CA1249827A (enExample)
DD (1) DD207715A5 (enExample)
DE (1) DE3372481D1 (enExample)
DK (1) DK162842C (enExample)
ES (2) ES524873A0 (enExample)
FI (1) FI82933C (enExample)
GR (1) GR78905B (enExample)
HU (1) HU188943B (enExample)
IE (1) IE55845B1 (enExample)
IL (1) IL69485A (enExample)
IN (1) IN160173B (enExample)
NO (1) NO159086C (enExample)
NZ (1) NZ205243A (enExample)
PH (1) PH18645A (enExample)
PL (2) PL140540B1 (enExample)
PT (1) PT77193B (enExample)
SU (1) SU1468416A3 (enExample)
YU (1) YU42874B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU570659B2 (en) * 1982-12-14 1988-03-24 Ciba-Geigy Ag 1-azolyl-2-aryl-3-fluoroalkan-2-ols and ethers thereof

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8302498D0 (en) * 1983-01-29 1983-03-02 Pfizer Ltd Antifungal agents
US4584307A (en) * 1983-08-10 1986-04-22 Pfizer Inc. Antifungal 2-aryl-2-hydroxy perfluoro-1-(1H-1,2,4-triazol-1-yl) alkanones and alkanols
GB8322983D0 (en) * 1983-08-26 1983-09-28 Pfizer Ltd Triazole antifungal agents
FR2622582B1 (fr) * 1987-10-29 1990-01-19 Rhone Poulenc Agrochimie Composes a groupe imidazole ou triazole, utilisation de ceux-ci a titre de fongicide, procede de preparation
IT1186784B (it) * 1985-11-04 1987-12-16 Montedison Spa Azoliderivati ad attivita' antufungina
IT1196528B (it) * 1986-07-21 1988-11-16 Donegani Guido Ist Azolilderivati ad attivita' antifungina
IT1198240B (it) * 1986-12-23 1988-12-21 Agrimont Spa Azolilderivati fungicidi
US4935436A (en) * 1989-01-23 1990-06-19 The Dow Chemical Company Substituted triazoles and their use as fungicides
EP0470466A3 (en) * 1990-08-09 1992-07-29 Bayer Ag Halogenalkyl-azolyl derivatives
US5262434A (en) * 1990-08-09 1993-11-16 Bayer Aktiengesellschaft Halogenoalkyl-azolyl derivatives
JP3471831B2 (ja) * 1991-12-09 2003-12-02 富山化学工業株式会社 新規なトリアゾール誘導体およびその塩
US5611210A (en) * 1993-03-05 1997-03-18 Ikon Corporation Fluoroiodocarbon blends as CFC and halon replacements
US6270689B1 (en) 1998-03-26 2001-08-07 Ikon Corporation Blend compositions of trifluoroiodomethane, tetrafluoroethane and difluoroethane
US20110262517A1 (en) * 2007-04-05 2011-10-27 The Johns Hopkins University Chirally pure isomers of itraconazole and inhibitors of lanosterol 14a-demethylase for use as angiogenesis inhibitors
US9095589B2 (en) 2007-04-05 2015-08-04 Johns Hopkins University Chirally pure isomers of itraconazole for use as angiogenesis inhibitors
EP3181558A1 (en) 2012-12-19 2017-06-21 Basf Se Substituted [1,2,4]triazole compounds and their use as fungicides

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE45765B1 (en) * 1976-08-19 1982-11-17 Ici Ltd Triazoles and imidazoles useful as plant fungicides and growth regulating agents
DE2832234A1 (de) * 1978-07-21 1980-01-31 Bayer Ag Alpha -azolyl-keto-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
US4654332A (en) * 1979-03-07 1987-03-31 Imperial Chemical Industries Plc Heterocyclic compounds
DE2951164A1 (de) * 1979-12-19 1981-07-16 Bayer Ag, 5090 Leverkusen Substituierte triazolylmethyl-tert.-butyl-ketone, verfahren zu ihrer herstellung und ihre verwendung als pflanzenschutzmittel sowie als zwischenprodukte
EP0131684B1 (en) * 1980-08-18 1992-03-11 Imperial Chemical Industries Plc Use of triazolylethanol derivatives and their compositions as non-agricultural fungicides
AU553482B2 (en) * 1980-08-28 1986-07-17 Imperial Chemical Industries Plc Pharmaceutical compositions of fungicidal triazole derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU570659B2 (en) * 1982-12-14 1988-03-24 Ciba-Geigy Ag 1-azolyl-2-aryl-3-fluoroalkan-2-ols and ethers thereof

Also Published As

Publication number Publication date
EP0104734A1 (en) 1984-04-04
IE55845B1 (en) 1991-01-30
DK367883A (da) 1984-02-15
AU1793083A (en) 1984-02-16
PT77193B (en) 1986-03-21
SU1468416A3 (ru) 1989-03-23
HU188943B (en) 1986-05-28
DE3372481D1 (en) 1987-08-20
KR880001046B1 (ko) 1988-06-18
DD207715A5 (de) 1984-03-14
ES8600256A1 (es) 1985-10-01
DK367883D0 (da) 1983-08-12
IN160173B (enExample) 1987-06-27
PL139633B1 (en) 1987-02-28
EP0104734B1 (en) 1987-07-15
ES8601932A1 (es) 1985-11-16
YU168283A (en) 1986-02-28
IL69485A (en) 1987-09-16
NO159086B (no) 1988-08-22
NO832915L (no) 1984-02-15
NZ205243A (en) 1986-04-11
PL243409A1 (en) 1985-07-16
PL140540B1 (en) 1987-05-30
PT77193A (en) 1983-09-01
CA1249827A (en) 1989-02-07
ES540857A0 (es) 1985-11-16
KR840005719A (ko) 1984-11-15
FI832904L (fi) 1984-02-15
US4616027A (en) 1986-10-07
FI82933B (fi) 1991-01-31
DK162842C (da) 1992-05-04
YU42874B (en) 1988-12-31
IL69485A0 (en) 1983-11-30
DK162842B (da) 1991-12-16
PH18645A (en) 1985-08-23
GR78905B (enExample) 1984-10-02
IE831889L (en) 1984-02-14
FI82933C (fi) 1991-05-10
FI832904A0 (fi) 1983-08-11
NO159086C (no) 1988-11-30
PL252362A1 (en) 1985-11-19
ES524873A0 (es) 1985-10-01

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